A novel procedure for the synthesis of aziridines: application of Simmons–Smith reagents to aziridination

A novel procedure for the synthesis of aziridines: application of Simmons–Smith reagents to aziridination

The reaction of Simmons–Smith carbenoids with imines in the presence of sulfides provides N-( p-toluenesulfonyl)- and N-[(1,1,1-trimethylsilyl)ethyl]sulfonyl-substituted aziridines in high yield. Graphic

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Bibliographic Details
Published in:Tetrahedron letters Vol. 42; no. 8; pp. 1587 - 1589
Main Authors: Aggarwal, Varinder K, Stenson, Rachel A, Jones, Ray V.H, Fieldhouse, Robin, Blacker, John
Format: Journal Article
Language:English
Published: Elsevier Ltd 19-02-2001
Online Access:Get full text
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Description
Summary:The reaction of Simmons–Smith carbenoids with imines in the presence of sulfides provides N-( p-toluenesulfonyl)- and N-[(1,1,1-trimethylsilyl)ethyl]sulfonyl-substituted aziridines in high yield. Graphic
ISSN:0040-4039
1873-3581
DOI:10.1016/S0040-4039(00)02310-8