Search Results - SP Birkhäuser Verlag Boston
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1
Potent antimalarial activity of newly synthesized substituted chalcone analogs in vitro
Published in Medicinal chemistry research (01-07-2009)“…Several new chalcone analogues were synthesized and evaluated as inhibitors of malaria parasite. Inhibitory activity was determined in vitro against a…”
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2
Molecular docking study on anticancer activity of plant-derived natural products
Published in Medicinal chemistry research (01-11-2010)“…A variety of compounds from plant sources have been reported to possess substantial anticancer properties; however, their modes of action have not been clearly…”
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3
Synthesis and pharmacological evaluation of newer thiazolo [3,2-a] pyrimidines for anti-inflammatory and antinociceptive activity
Published in Medicinal chemistry research (01-12-2010)“…A new series of thiazolo [3,2-a] pyrimidine derivatives was designed and synthesized using 4-fluoroaniline and ethylacetoacetate as starting material…”
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4
Synthesis and evaluation of 4-amino-5-phenyl-4H-[1,2,4]-triazole-3-thiol derivatives as antimicrobial agents
Published in Medicinal chemistry research (01-03-2010)“…A series of novel 1,2,4-triazole derivatives have been synthesized by condensing the methyl benzoate and methyl salicylate with various substituents; their…”
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5
Synthesis of new 2(1H)-quinoxalinone derivatives for antimicrobial and antiinflammatory evaluation
Published in Medicinal chemistry research (01-12-2009)“…New 2(1H)-quinoxalinones and their hexahydro derivatives were prepared for investigating their antimicrobial and antiinflammatory activities. The study showed…”
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6
Synthesis and biological activity studies of furan derivatives
Published in Medicinal chemistry research (01-06-2010)“…The organic compounds, 4-Ethyl-2,5,5-triphenyl-4,5-dihydrofuran-3-carbonitrile; 2,4,5-Triphenyl-5-propyl-4,5-dihydrofuran-3-carbonitrile;…”
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7
Inhibitory effect of Gymnema Montanum leaves on α-glucosidase activity and α-amylase activity and their relationship with polyphenolic content
Published in Medicinal chemistry research (01-11-2010)“…The present study was attempted to investigate the effect of G. montanum leaf extract on inhibition of α-glucosidase and α-amylase activity. The ethanol…”
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8
Piperamides and their derivatives as potential anti-trypanosomal agents
Published in Medicinal chemistry research (01-12-2009)“…We describe herein an evaluation of the trypanocidal effect of eight piperamides (1-8) isolated from Piper tuberculatum bearing dihydropyridone, piperidine,…”
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9
Design and synthesis of 2-quinolones as antioxidants and antimicrobials: a rational approach
Published in Medicinal chemistry research (01-03-2010)“…As an important class of compounds, 2-quinolones are isomeric to 4-quinolones and isosteric to coumarins. The compounds that have 2-quinolone moiety are…”
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10
Antioxidant phenolic compounds and flavonoids of Mitragyna rotundifolia (Roxb.) Kuntze in vitro
Published in Medicinal chemistry research (01-12-2010)“…Different solvent extracts of leaves and bark of Mitragyna rotundifolia (Roxb.) Kuntze were evaluated by DPPH, ABTS, and FRAP assays, respectively, for…”
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11
Anticonvulsant and sedative-hypnotic activity of some novel 3-[5-(4-substituted) phenyl-1,3,4-oxadiazole-2yl]-2-styrylquinazoline-4(3H)-ones
Published in Medicinal chemistry research (01-04-2010)“…A few novel 3-[5-(4-substituted) phenyl-1,3,4-oxadiazole-2-yl]-2-styryl quinazoline-4(3H)-ones were synthesized and evaluated for anticonvulsant,…”
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12
Extraction of water-soluble polysaccharide and the antioxidant activity from Ginkgo biloba leaves
Published in Medicinal chemistry research (01-04-2010)“…Water-soluble polysaccharide was isolated from Ginkgo biloba leaves with the method of water-dissolving and ethanol-precipitating. The optimized condition for…”
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13
Synthesis and evaluation of curcumin analogues as cytotoxic agents
Published in Medicinal chemistry research (01-06-2010)“…Seventeen curcumin analogues were prepared and evaluated for in vitro and in vivo cytotoxicity against an Ehrlich ascites carcinoma (EAC). In vitro results…”
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14
Lonazolac analogues: molecular modeling, synthesis, and in vivo anti-inflammatory activity
Published in Medicinal chemistry research (01-12-2009)“…A novel series of 1,3-diarylpyrazole derivatives (4-8), analogues to lonazolac, were designed, synthesized, and evaluated for their anti-inflammatory as well…”
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15
Synthesis and in vivo anticancer and antiangiogenic effects of novel thioxothiazolidin-4-one derivatives against transplantable mouse tumor
Published in Medicinal chemistry research (01-04-2010)“…A series of novel thioxothiazolidin-4-one derivatives 5(a-g) were synthesized by the coupling of different amines containing aliphatic, substituted aromatic,…”
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16
Design, synthesis, antifungal activity, and ADME prediction of functional analogues of terbinafine
Published in Medicinal chemistry research (01-07-2009)“…From the earlier quantitative structure-activity relationship (QSAR) and molecular modeling studies, a series of quinoline derivatives 5a-h mimicking…”
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17
Antioxidant activity of alcoholic extract of Agrimonia pilosa Ledeb
Published in Medicinal chemistry research (01-06-2010)“…Ultrasonically assisted extraction and Soxhlet extraction using 95% ethanol were performed to obtain ultrasonically assisted extract of Agrimonia pilosa (UEA)…”
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18
Antioxidant activities of Liquidambar formosana Hance leaf extracts
Published in Medicinal chemistry research (01-03-2010)“…Leaves of Liquidambar formosana Hance has been be used as a rice dye for festival food by a small group of people in Guangxi province China. This study…”
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19
Anti-inflammatory and antioxidant activities of some extracts and pure natural products isolated from Rhus tripartitum (Ucria)
Published in Medicinal chemistry research (01-04-2010)“…Chromatographic separation of Rhus tripartitum (Anacardiaceae) chemical components revealed the presence of four main natural substances: a new biflavonoid…”
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20
Extraction of essential oils from garlic (Allium sativum) using ligarine as solvent and its immunity activity in gastric cancer rat
Published in Medicinal chemistry research (01-12-2010)“…The solvent extraction (SE) of garlic essential oil (Allium sativum) was studied. A multivariate study based on a four-factor, three-level Box-Behnken design…”
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