Search Results - "Zucchelli, Valeria"

Design and Synthesis of Novel Tricyclic Benzoxazines as Potent 5-HT1A/B/D Receptor Antagonists Leading to the Discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M, Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J, Granci, Enrica, Leslie, Colin P, Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M, Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of…”
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Design and Synthesis of Novel Tricyclic Benzoxazines as Potent 5-HT 1A/B/D Receptor Antagonists Leading to the Discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4 H -imidazo[5,1- c ][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M., Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J., Granci, Enrica, Leslie, Colin P., Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M., Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

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8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones: dual-acting 5-HT1 receptor antagonists and serotonin reuptake inhibitors--part II by Bromidge, Steven M, Bertani, Barbara, Borriello, Manuela, Bozzoli, Andrea, Faedo, Stefania, Gianotti, Massimo, Gordon, Laurie J, Hill, Matthew, Zucchelli, Valeria, Watson, Jeannette M, Zonzini, Laura

“…8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones have been identified as highly potent 5-HT(1A/B/D) receptor antagonists with and without…”
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6-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones : Dual-acting 5-HT1 receptor antagonists and serotonin reuptake inhibitors by BROMIDGE, Steven M, BERTANI, Barbara, MERLO, Giancarlo, VESENTINI, Alessia, WATSON, Jeannette M, ZONZINI, Laura, BORRIELLO, Manuela, FAEDO, Stefania, GORDON, Laurie J, GRANCI, Enrica, HILL, Matthew, MARSHALL, Howard R, STASI, Luigi P, ZUCCHELLI, Valeria

“…Investigation of a series 6-[2-(4-aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones has led to the discovery of potent 5-HT(1A/1B/1D) receptor antagonists…”
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5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1H)-quinolinones and 3,4-dihydro-2(1H)-quinolinones: Dual-acting 5-HT1 receptor antagonists and serotonin reuptake inhibitors. Part 3 by BROMIDGE, Steven M, ARBAN, Roberto, PASQUARELLO, Alessandra, SPADA, Simone K, WORBY, Angela, ZONZINI, Laura, ZUCCHELLI, Valeria, BERTANI, Barbara, BORRIELLO, Manuela, CAPELLI, Anna-Maria, DI-FABIO, Romano, FAEDO, Stefania, GIANOTTI, Massimo, GORDON, Laurie J, GRANCI, Enrica

“…5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1H)-quinolinones and 3,4-dihydro-2(1H)-quinolinones have been identified with different combinations of…”
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5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1H)-quinoli nones and 3,4-dihydro-2(1H)-quinolinones: Dual-acting 5-HT sub(1) receptor antagonists and serotonin reuptake inhibitors. Part 3 by Bromidge, Steven M, Arban, Roberto, Bertani, Barbara, Borriello, Manuela, Capelli, Anna-Maria, Di-Fabio, Romano, Faedo, Stefania, Gianotti, Massimo, Gordon, Laurie J, Granci, Enrica, Pasquarello, Alessandra, Spada, Simone K, Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1H)-quinoli nones and 3,4-dihydro-2(1H)-quinolinones have been identified with different combinations of…”
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5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1 H)-quinolinones and 3,4-dihydro-2(1 H)-quinolinones: Dual-acting 5-HT 1 receptor antagonists and serotonin reuptake inhibitors. Part 3 by Bromidge, Steven M., Arban, Roberto, Bertani, Barbara, Borriello, Manuela, Capelli, Anna-Maria, Di-Fabio, Romano, Faedo, Stefania, Gianotti, Massimo, Gordon, Laurie J., Granci, Enrica, Pasquarello, Alessandra, Spada, Simone K., Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…5-{2-[4-(2-Methyl-5-quinolinyl)-1-piperazinyl]ethyl}-2(1 H)-quinolinones and 3,4-dihydro-2(1 H)-quinolinones have been identified with different combinations…”
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8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones : Dual-acting 5.HT1 receptor antagonists and serotonin reuptake inhibitors-Part II by BROMIDGE, Steven M, BERTANI, Barbara, ZONZINI, Laura, BORRIELLO, Manuela, BOZZOLI, Andrea, FAEDO, Stefania, GIANOTTI, Massimo, GORDON, Laurie J, HILL, Matthew, ZUCCHELLI, Valeria, WATSON, Jeannette M

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8-[2-(4-Aryl-1-piperazinyl)ethyl]-2 H-1,4-benzoxazin-3(4 H)-ones: Dual-acting 5-HT 1 receptor antagonists and serotonin reuptake inhibitors—Part II by Bromidge, Steven M., Bertani, Barbara, Borriello, Manuela, Bozzoli, Andrea, Faedo, Stefania, Gianotti, Massimo, Gordon, Laurie J., Hill, Matthew, Zucchelli, Valeria, Watson, Jeannette M., Zonzini, Laura

“…8-[2-(4-Aryl-1-piperazinyl)ethyl]-2 H-1,4-benzoxazin-3(4 H)-ones have been identified as highly potent 5-HT 1A/B/D receptor antagonists with and without…”
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6-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones: Dual-acting 5-HT sub(1) receptor antagonists and serotonin reuptake inhibitors by Bromidge, Steven M, Bertani, Barbara, Borriello, Manuela, Faedo, Stefania, Gordon, Laurie J, Granci, Enrica, Hill, Matthew, Marshall, Howard R, Stasi, Luigi P, Zucchelli, Valeria, Merlo, Giancarlo, Vesentini, Alessia, Watson, Jeannette M, Zonzini, Laura

“…Investigation of a series 6-[2-(4-aryl-1-piperazinyl)ethyl]-2H-1,4- benzoxazin-3(4H)-ones has led to the discovery of potent 5-HT sub(1A/1B/1D) receptor…”
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2-Alkyl-4,6-dialkylamino-1,3,5-triazines via Grignard Alkylation of Cyanuric Chloride: An Aged Reaction Revisited by Menicagli, Rita, Samaritani, Simona, Zucchelli, Valeria

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6-[2-(4-Aryl-1-piperazinyl)ethyl]-2 H-1,4-benzoxazin-3(4 H)-ones: Dual-acting 5-HT 1 receptor antagonists and serotonin reuptake inhibitors by Bromidge, Steven M., Bertani, Barbara, Borriello, Manuela, Faedo, Stefania, Gordon, Laurie J., Granci, Enrica, Hill, Matthew, Marshall, Howard R., Stasi, Luigi P., Zucchelli, Valeria, Merlo, Giancarlo, Vesentini, Alessia, Watson, Jeannette M., Zonzini, Laura

“…Investigation of a series 6-[2-(4-aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones has led to the discovery of potent 5-HT 1A/1B/1D receptor antagonists…”
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Design and synthesis of novel tricyclic benzoxazines as potent 5-HT(1A/B/D) receptor antagonists leading to the discovery of 6-{2-[4-(2-methyl-5-quinolinyl)-1-piperazinyl]ethyl}-4H-imidazo[5,1-c][1,4]benzoxazine-3-carboxamide (GSK588045) by Bromidge, Steven M, Arban, Roberto, Bertani, Barbara, Bison, Silvia, Borriello, Manuela, Cavanni, Paolo, Dal Forno, Giovanna, Di-Fabio, Romano, Donati, Daniele, Fontana, Stefano, Gianotti, Massimo, Gordon, Laurie J, Granci, Enrica, Leslie, Colin P, Moccia, Luca, Pasquarello, Alessandra, Sartori, Ilaria, Sava, Anna, Watson, Jeannette M, Worby, Angela, Zonzini, Laura, Zucchelli, Valeria

“…Bioisoteric replacement of the metabolically labile N-methyl amide group of a series of benzoxazinones with small heterocyclic rings has led to novel series of…”
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Clinical Features and Long-Term Follow-Up of 20 Cases of Parakeratosis Pustulosa by Tosti, Antonella, Peluso, Anna Maria, Zucchelli, Valeria

“…: We report the clinical features and long‐term follow‐up of 20 pediatric patients with parakeratosis pustulosa (PKP). In eight children PKP was considered as…”
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Clinical features and long-term follow-up of 20 cases of parakeratosis pustulosa by TOSTI, A, PELUSO, A. M, ZUCCHELLI, V

“…We report the clinical features and long-term follow-up of 20 pediatric patients with parakeratosis pustulosa (PKP). In eight children PKP was considered as a…”
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Contact dermatitis from levobunolol and befunolol by Zucchelli, V, Silvani, S, Vezzani, C, Lorenzi, S, Tosti, A

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Allergic contact dermatitis due to phenol-formaldehyde resins in a knee-guard by Vincenzi, C, Guerra, L, Peluso, A M, Zucchelli, V

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