Search Results - "Zhao, Gui Long"

Exquisite Synthesis of a Designed PAR-1 Antagonist by Miao, Hua-Ming, Zhao, Gui-Long, Zhang, Lin-Shan, Shao, Hua, Wang, Jian-Wu

“…The synthesis of a designed, sterically congested geminal dimethyl‐bearing PAR‐1 antagonist was achieved by a route of ten steps, with the oxidation of an…”
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SrCl2 as an efficient cocatalyst for acidic hydrolysis of methyl glycosides by Shi, Yong-Heng, Xie, Ya-Fei, Liu, Yu-Qiang, Wei, Qun-Chao, Xu, Wei-Ren, Tang, Li-Da, Zhao, Gui-Long

“…SrCl2 was found to be the most efficient cocatalyst for the acidic hydrolysis of methyl glycosides after 26 kinds of most representative metal salts were…”
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Design,synthesis and biological activity of cyclohexane-bearing C-glucoside derivatives as SGLT2 inhibitors by Zhang, Shuo, Wang, Yu-Li, Wei, Qun-Chao, Xu, Wei-Ren, Tang, Li-Da, Zhao, Gui-Long, Wang, Jian-Wu

“…Seven cyclohexane-bearing C-glucoside derivatives（7,9,12,13 and 17-19） were designed and synthesized as SGLT2 inhibitors starting from a potent SGLT2 inhibitor…”
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Design,synthesis and in vivo anti-hyperglycemic activity of gem-dimethyl-bearing C-glucosides as SGLT2 inhibitors by Zhao, Wen Jing, Shi, Yong Heng, Zhao, Gui Long, Wang, Yu Li, Shao, Hua, Da Tang, Li, Wang, Jian Wu

“…A series of gem-dimethyl-bearing C-glucosides were designed and synthesized as SGLT2 inhibitors,with anhydrous aluminum chloride-mediated Friedel-Crafts…”
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A New Synthetic Approach to Elvucitabine by Zhang, Ling-yu, Lou, Yuan-yuan, Zhao, Gui-long, Zhang, Lin-shan, Chen, Yan

“…A new synthetic approach to elvucitabine started from L-xylose via the reactions of 10 steps in an overall yield of 20% was developed. The key steps included…”
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Synthesis, biological evaluation and 3D-QSAR studies of 1,2,4-triazole-5-substituted carboxylic acid bioisosteres as uric acid transporter 1 (URAT1) inhibitors for the treatment of hyperuricemia associated with gout by Wu, Jing-wei, Yin, Ling, Liu, Yu-qiang, Zhang, Huan, Xie, Ya-fei, Wang, Run-ling, Zhao, Gui-long

“…[Display omitted] As a part of our ongoing research to develop novel URAT1 inhibitors, 19 compounds (1a-1s) based on carboxylic acid bioisosteres were…”
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Total Synthesis of 4′′-O-Acetylmananthoside B Part II: Synthesis of the Disaccharide Fragment by ZHAO, Gui-Long, YU, Zhao-Yun, LI, Yan, PANG, Li-Na, WANG, Jian-Wu

“…A disaccharide compound, p‐methoxyphenyl 2,3,4‐tri‐O‐benzyl‐β‐L‐arabinopyranosyl‐(1→6)‐2‐O‐benzyl‐3,4‐di‐O‐acetyl‐β‐D‐galactopyranoside (17), was successfully…”
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(3-Phenyl-isoxazol-5-yl)methanol by Yin, Ling, Zhao, Gui-Long, Jia, Jiong, Meng, Qing-Yang, Wang, Jian-Wu

“…In the title compound, C(10)H(9)NO(2), the isoxazole and phenyl rings form a dihedral angle of 25.82 (3)°. In the crystal, inter-molecular O-H⋯O hydrogen bonds…”
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2-[(2,6-Dichloro-benz-yl)amino]-N-(4-methyl-thia-zol-2-yl)acetamide by Luo, Jie, Zhao, Gui-Long, Shao, Hua, Wang, Yu-Li, Qu, Bao-Han

“…In the title compound, C(13)H(13)Cl(2)N(3)OS, the thia-zole and benzene rings are roughly parallel to one another in two layers [dihedral angle = 5.08 (2)°]…”
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tert-Butyl N-(5-bromo-1H-imidazo[4,5-b]pyridin-2-ylmeth-yl)carbamate by Yin, Ling, Jia, Jiong, Zhao, Gui-Long, Wang, Jian-Wu

“…In the mol-ecule of the title compound, C(12)H(15)BrN(4)O(2), the imidazole and pyridine rings are strictly coplanar [maximum deviation 0.006 (3) Å]. In the…”
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A Facile Approach to Indolizines via Tandem Reaction by Wang, Jianwu, Ge, Yan-Qing, Jia, Jiong, Yang, He, Zhao, Gui-Long, Zhan, Fu-Xu

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A New Method for the Synthesis of [1,2,4]Triazolo[1,5-a]pyridine Derivatives by Wang, Jian-Wu, Ge, Yan-Qing, Zhao, Wei-Ming, Xu, Wei-Ren, Zhao, Gui-Long, Jia, Jiong

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Synthesis of Nitrogen Bridgehead Heterocycles with Phosphonates via a Novel Tandem Process by Wang, Jian-Wu, Jia, Jiong, Xie, Ya-Fei, Feng, Lei, Xu, Hua-Qiang, Meng, Song, Zhao, Gui-Long, Xu, Wei-Ren, Ge, Yan-Qing

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Bioremediation of Oil Sludge in Shengli Oilfield by De-qing, Shi, Jian, Zhang, Zhao-long, Gui, Jian, Dong, Tian-li, Wang, Murygina, Valentina, Kalyuzhnyi, Sergey

“…Large quantity of dehydrated oil sludge, generated in the disposal process of oil-containing sewage in Shengli oilfield, needs to be rendered harmless to human…”
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Ethyl 6-methylsulfanyl-2-phenyl-1H-imidazo[1,2-b]pyrazole-7-carboxylate monohydrate by Teng-fei Shao, Gui-long Zhao, Jian-wu Wang

“…The title compound, C15H15N3O2S·H2O, has been obtained in a search for new imidazo[1,2-b]pyrazole derivatives with better biological activity. The…”
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(5-Bromo-2-methyl-phen-yl)(4-eth-oxy-phen-yl)methanone by Shi, Yong-Heng, Zhao, Gui-Long, Shao, Hua, Liu, Wei, Xu, Wei-Ren

“…In the title compound, C(16)H(15)BrO(2), the dihedral angle between the benzene rings is 68.5 (2)°. In the crystal structure, mol-ecules are linked by weak…”
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1-(3-tert-Butyl-4-hy-droxy-phen-yl)ethanone by Miao, Hua-Ming, Zhao, Gui-Long, Shao, Hua, Wang, Jian-Wu

“…The title compound, C(12)H(16)O(2), is approximately planar (r.m.s. deviation = 0.030 Å), apart from two methyl groups of the tert-butyl unit [deviations of…”
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Ethyl 6-methyl-2- p -tolylpyrazolo[1,5- a ]pyridine-5-carboxylate by Jia, Jiong, Ge, Yan-qing, Zhao, Gui-long, Wang, Jian-wu

“…In the title molecule, C18H18N2O2, the bicyclic ring system and the benzene ring form a dihedral angle of 13.45 (3)°. In the crystal structure, weak…”
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5-(4-Ethoxybenzyl)-1H-tetrazole by Yun-Long Gao, Gui-Long Zhao, Hua Shao, Wei Liu, Jian-wu Wang

“…In the title molecule, C10H12N4O, the tetrazole and benzene rings form a dihedral angle of 67.52 (2)°. In the crystal, intermolecular N—H...N…”
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Ethyl 6-methyl-2-p-tolyl-pyrazolo[1,5-a]pyridine-5-carboxyl-ate by Jia, Jiong, Ge, Yan-Qing, Zhao, Gui-Long, Wang, Jian-Wu

“…In the title mol-ecule, C(18)H(18)N(2)O(2), the bicyclic ring system and the benzene ring form a dihedral angle of 13.45 (3)°. In the crystal structure, weak…”
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