Search Results - "Zebardast, Tannaz"
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Design and synthesis of new 1,3-benzthiazinan-4-one derivatives as selective cyclooxygenase (COX-2) inhibitors
Published in Bioorganic & medicinal chemistry (01-08-2009)“…A new group of 1,3-benthiazinan-4-ones, possessing a methyl sulfonyl pharmacophore, were synthesized and their biological activities were evaluated for…”
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Molecular Docking and QSAR Study of 2-Benzoxazolinone, Quinazoline and Diazocoumarin Derivatives as Anti-HIV-1 Agents
Published in Iranian journal of pharmaceutical research : IJPR (01-06-2019)“…A series of 2-benzoxazolinone, diazocoumarin and quinazoline derivatives have been shown to inhibit HIV replication in cell culture. To understand the…”
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Design and synthesis of 3-alkyl-2-aryl-1,3-thiazinan-4-one derivatives as selective cyclooxygenase (COX-2) inhibitors
Published in Bioorganic & medicinal chemistry letters (15-06-2009)“…The design, synthesis and evaluation of a series of 3-alkyl-2-aryl-1,3-thiazinan-4-ones, possessing a methylsulfonyl pharmacophore, as potent and selective…”
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QSAR Modeling of COX -2 Inhibitory Activity of Some Dihydropyridine and Hydroquinoline Derivatives Using Multiple Linear Regression (MLR) Method
Published in Iranian journal of pharmaceutical research : IJPR (01-01-2017)“…COX-2 inhibitory activities of some 1,4-dihydropyridine and 5-oxo-1,4,5,6,7,8-hexahydroquinoline derivatives were modeled by quantitative structure-activity…”
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Design and Synthesis of New 1,3-Benzdiazinan-4-one Derivatives as Selective Cyclooxygenase (COX-2) Inhibitors
Published in Archiv der Pharmazie (Weinheim) (01-04-2012)“…A new group of regioisomeric 2,3‐diaryl‐1,3‐benzdiazinan‐4‐ones, possessing a methyl sulfonyl pharmacophore, were synthesized and their biological activities…”
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Synthesis and biological evaluation of 1,3-diphenylprop-2-en-1-ones possessing a methanesulfonamido or an azido pharmacophore as cyclooxygenase-1/-2 inhibitors
Published in Bioorganic & medicinal chemistry (15-10-2006)“…A group of ( E)-1,3-diphenylprop-2-en-1-one derivatives (chalcones) possessing a MeSO 2NH, or N 3, COX-2 pharmacophore at the para-position of the C-1 phenyl…”
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