Search Results - "Yakkala, Prasanna Anjaneyulu"

Rh(III)-Catalyzed [3 + 2] Annulation via C–H Activation: Direct Access to Trifluoromethyl-Substituted Indenamines and Aminoindanes by Chaudhary, Bharatkumar, Auti, Prashant, Shinde, Suchita Dattatray, Yakkala, Prasanna Anjaneyulu, Giri, Deepesh, Sharma, Satyasheel

“…The rhodium­(III)-catalyzed direct C–H addition and annulation of benzimidates and aldimines with β-(trifluoromethyl)-α,β-unsaturated ketones is described…”
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Prospects of Topoisomerase Inhibitors as Promising Anti-Cancer Agents by Yakkala, Prasanna Anjaneyulu, Penumallu, Naveen Reddy, Shafi, Syed, Kamal, Ahmed

“…Topoisomerases are very important enzymes that regulate DNA topology and are vital for biological actions like DNA replication, transcription, and repair. The…”
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Multicomponent Domino Reaction for Concise Access to 2‑Amino-Substituted 1,3,4 Oxadiazoles via Smiles Rearrangement by Yakkala, Prasanna Anjaneyulu, Khan, Imran A., Dannarm, Srinivas Reddy, Aboti, Jyoti, Sonti, Rajesh, Shafi, Syed, Kamal, Ahmed

“…A multicomponent domino reaction has been developed for the preparation of N-substituted 2-amino-1,3,4-oxadiazoles directly from various hydrazides (32…”
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Novel approaches for the development of direct KRAS inhibitors: structural insights and drug design by Haider, Kashif, Sharma, Anku, Yar, M Shahar, Yakkala, Prasanna Anjaneyulu, Shafi, Syed, Kamal, Ahmed

“…Hyperactivated RAS signaling is reported in 13% of all human cancers, in which ~80% resulted due to KRAS mutations alone. Direct inhibition of KRAS is an…”
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Development and Evaluation of Bis-benzothiazoles as a New Class of Benzothiazoles Targeting DprE1 as Antitubercular Agents by Samoon, Rabiya, Sau, Shashikanta, Roy, Arnab, Parida, Kishan Kumar, Sharma, Kalicharan, Yakkala, Prasanna Anjaneyulu, Dewangan, Rikeshwer Prasad, Abdin, Malik Zainul, Kalia, Nitin Pal, Shafi, Syed

“…Benzothiazole-bearing compounds have emerged as potential noncovalent DprE1 (decaprenylphosphoryl-β-d-ribose-2′-epimerase) inhibitors active against…”
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Design and Synthesis of Michael Acceptor‐Based Peptidyl β‐Nitrostyrenes as 3CLpro Inhibitors of SARS‐CoV‐2 by Sharma, Sweta, Yakkala, Prasanna Anjaneyulu, Aboti, Jyoti, Latief, Insha, Ansari, Mairaj Ahmed, Khan, Wajihul Hasan, Shafi, Syed

“…Severe Acute Respiratory Syndrome coronavirus 2 main protease was found to be one of the most attractive anti‐viral targets for the development of new chemical…”
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5‐Arylidene‐2,4‐thiazolidinediones as Cysteine Protease Inhibitors against Leishmania Donovani by Sharma, Sweta, Anjaneyulu Yakkala, Prasanna, Beg, Mirza A., Tanwar, Supriya, Latief, Insha, Khan, Arif, Sharma, Kalicharan, ur Rehman, Sayeed, Selvapandiyan, Angamuthu, Shafi, Syed

“…A series of 5‐arylidene‐2,4‐thiazolidinediones were synthesized using Knoevenagel condensation and evaluated for their anti‐leishmanial activity against L…”
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