Search Results - "YAKAIAH, T"

Synthesis of novel 4,6-disubstituted quinazoline derivatives, their anti-inflammatory and anti-cancer activity (cytotoxic) against U937 leukemia cell lines by Chandrika, P. Mani, Yakaiah, T., Rao, A. Raghu Ram, Narsaiah, B., Reddy, N. Chakra, Sridhar, V., Rao, J. Venkateshwara

“…In view of the link between use of NSAIDs and altered cancer incidence and a growing evidence of COX-II implication in angiogenesis, a novel series of…”
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Synthesis and structure–activity relationships of novel pyrimido[1,2- b]indazoles as potential anticancer agents against A-549 cell lines by Yakaiah, T., Lingaiah, B.P.V., Narsaiah, B., Shireesha, B., Ashok Kumar, B., Gururaj, S., Parthasarathy, T., Sridhar, B.

“…A series of novel pyrimido[1,2- b]indazoles 5, 7 have been prepared from 3-trifluoromethyl-5-phenyl-2,6-dicyano anilines 1 via novel indazole regioisomers 3…”
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Click chemistry: Studies on the synthesis of novel fluorous tagged triazol-4-yl substituted quinazoline derivatives and their biological evaluation – Theoretical and experimental validation by Mani Chandrika, P., Yakaiah, T., Gayatri, G., Pranay Kumar, K., Narsaiah, B., Murthy, U.S.N., Raghu Ram Rao, A.

“…The formation of N- and O-propargylated quinazoline derivatives 2, 3 from quinazol-4-ones 1 was theoretically predicted by optimizations at B3LYP/6-31G* level,…”
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Synthesis and theoretical studies on energetics of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines – Their potential as adenosine receptor ligands by Sirisha, B., Narsaiah, B., Yakaiah, T., Gayatri, G., Sastry, G. Narahari, Prasad, M. Raghu, Rao, A. Raghuram

“…A series of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines 6a– c and 7a– d was synthesized in two steps from thienopyrimidin-4-ones 2 through…”
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GdCl3 catalysed Grieco condensation : A facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity by YAKAIAH, T, LINGAIAH, B. P. V, NARSAIAH, B, PRANAY KUMAR, K, MURTHY, U. S. N

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Perfluorinated resin-sulfonic acid (Nafion-H): an efficient, environment friendly and recyclable heterogeneous catalyst for the one-pot multicomponent synthesis of β-acetamido ketones by Yakaiah, T., Lingaiah, B. P. V., Reddy, G. Venkat, Narsaiah, B., Rao, P. Shanthan

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Efficient Strategy for the Synthesis of 4-Hydroxy-1H-pyrrole-2,3-dicarboxylic Ester Derivatives Using Transition-Metal-Oxide Catalysts by Paul, V. Luke, Yakaiah, T., Reddy, A. Raghuram, Shekhar, A. Chandra, Rao, P. Shanthan, Narsaiah, B.

“…A facile and an efficient strategy for the synthesis of multisubstituted pyrrole derivatives was developed using an unusual ring annulation of dialkyl…”
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Silica Sulphuric Acid: An Efficient and Recyclable Catalyst for the Synthesis of β-Acetamido Ketones in Single Pot by Yakaiah, T., Reddy, G. Venkat, Lingaiah, B. P. V., Narsaiah, B., Rao, P. Shanthan

“…An efficient method has been developed for the synthesis of β-acetamido ketones by a multicomponent condensation route using sulphuric acid on silica gel as an…”
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Regioselective addition of Grignard reagents to 2,6-dicyanoanilines and cyclization to new quinazoline derivatives under thermal/microwave irradiation conditions by Maitraie, D., Yakaiah, T., Srinivas, K., Venkat Reddy, G., Ravikanth, S., Narsaiah, B., Shanthan Rao, P., Ravikumar, K., Sridhar, B.

“…Two strategies have been developed for the synthesis of novel quinazoline derivatives. 2,6-Dicyanoanilines were reacted with Grignard reagents followed by…”
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Efficient and Convenient Method for the Synthesis of Poly Functionalised 4H-Pyrans by Lingaiah, B. P. V., Reddy, G. Venkat, Yakaiah, T., Narsaiah, B., Reddy, S. N., Yadla, R., Rao, P. Shanthan

“…An efficient single-pot method for the synthesis of polyfunctionalized 4H-pyrans using alkaline metal fluoride as a catalyst is described. # IICT Communication…”
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Novel Bu4N+Br− catalyzed one-pot multi-component synthesis of 2-amino nicotinonitriles in aqueous medium by Kurumurthy, C., Naresh Kumar, R., Yakaiah, T., Shanthan Rao, P., Narsaiah, B.

“…An efficient single-pot strategy for 2-amino nicotinonitrile derivatives 5 has been developed by multi-component reaction of arylaldehydes 1 , methylketones 2…”
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GdCl3 promoted synthesis of novel pyrimidine fused indazole derivatives and their anticancer activity by Yakaiah, T., Kurumurthy, C., Lingaiah, B. P. V., Narsaiah, B., Pamanji, R., Velatooru, L. R., Venkateswara Rao, J., Gururaj, S., Parthasarathy, T., Sridhar, B.

“…The three component Grieco condensation of indazoles, aliphatic/aromatic aldehydes, and electron rich olefins in the presence of GdCl 3 resulted in a novel…”
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Synthesis of novel optically pure α-amino acid functionalised-7-trifluoromethyl substituted quinolone derivatives and their antibacterial activity by Venkat Lingaiah, B. P., Yakaiah, T., Ravi Kumar, A., Sathaiah, G., Chandra Shekhar, A., Raju, K., Shanthan Rao, P., Narsaiah, B., Murthy, U. S. N.

“…7-Trifluoromethyl-4-hydroxy quinoline-3-carboxylic acid ethyl ester was prepared from 3-amino benzotrifluoride and EMME. The hydroxyquinoline was reacted with…”
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GdCl(3) catalysed Grieco condensation: a facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity by Yakaiah, T, Lingaiah, B P V, Narsaiah, B, Kumar, K Pranay, Murthy, U S N

“…Indazole regioisomers such as 3-amino-4-(trifluoromethyl)-6-phenyl-1H-indazole-7-carbonitrile 1 and…”
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GdCl 3 catalysed Grieco condensation: A facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity by Yakaiah, T., Lingaiah, B.P.V., Narsaiah, B., Kumar, K. Pranay, Murthy, U.S.N.

“…Indazole regioisomers such as 3-amino-4-(trifluoromethyl)-6-phenyl-1 H-indazole-7-carbonitrile 1 and 3-amino-6-(trifluoromethyl)-4-phenyl-1…”
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Synthesis of novel 4,6-disubstituted quinazoline derivatives, their anti-inflammatory and anti-cancer activity (cytotoxic) against U937 leukemia cell line by MANI CHANDRIKA, P, YAKAIAH, T, RAGHU RAM RAO, A, NARSAIAH, B, CHAKRA REDDY, N, SRIDHAR, V, VENKATESHWARA RAO, J

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ZnBr2-Catalyzed Efficient Oxidative Homo Coupling of Aryl Magnesium Bromides by Kanth, S. Ravi, Reddy, G. Venkat, Yakaiah, T., Narsaiah, B., Rao, P. Shanthan

“…Oxidative homo coupling of various arylmagnesium bromides in the presence of ZnBr 2 gave the corresponding symmetrical biaryls in moderate to good yields at…”
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Gadolinium(III) chloride: a novel and an efficient reagent for the synthesis of homoallylic alcohols by Lingaiah, B. Venkat, Ezikiel, G., Yakaiah, T., Reddy, G. Venkat, Rao, P. Shanthan

“…Carbonyl compounds efficiently undergo nucleophilic addition reactions with allylstannanes in the presence of GdCl 3·6H 2O in acetonitrile under extremely mild…”
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ZnBr 2 ‐Catalyzed Efficient Oxidative Homo Coupling of Aryl Magnesium Bromides by Kanth, S. Ravi, Reddy, G. Venkat, Yakaiah, T., Narsaiah, B., Rao, P. Shanthan

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Synthesis of New Trifluoromethyl Substituted 11H-Isoindolo[2,1-a]benzimidazol-11-one Derivatives by Narsaiah, Banda, P. V. Lingaiah, Boddupally, Yakaiah, Tallapally, S. Rao, Pamulaparthy

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