Search Results - "Winiski, Anthony P."
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1
Pharmacological Inhibition of Stearoyl CoA Desaturase in the Skin Induces Atrophy of the Sebaceous Glands
Published in Journal of investigative dermatology (01-08-2013)Get full text
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2
Structure–activity relationship studies on a novel class of antiproliferative agents derived from Lavendustin A. Part I: Ring A modifications
Published in Bioorganic & medicinal chemistry (15-08-2008)“…The SAR of A-ring modified analogues of a novel class of antiproliferative agents and studies on the mode of action of compound 1 are described and discussed…”
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3
Determination of the transbilayer distribution of fluorescent lipid analogs by nonradiative fluorescence resonance energy transfer
Published in Biochemistry (Easton) (01-03-1992)“…We measured the nonradiative fluorescence resonance energy transfer between 7-nitro-2,1,3-benzoxadiazol-4-yl (NBD) labeled lipids (amine labeled…”
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4
Estrogenic Potential of 2-Alkyl-4-(thio)chromenone 6-O-Sulfamates: Potent Inhibitors of Human Steroid Sulfatase
Published in Journal of medicinal chemistry (06-11-2003)“…2-Alkylchromen-4-one 6-O-sulfamates, a new class of potent steroid sulfatase (STS) inhibitors, were evaluated for their estrogenic potential…”
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5
6-(2-Adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate: A potent non-steroidal irreversible inhibitor of human steroid sulfatase
Published in Bioorganic & medicinal chemistry letters (15-12-2003)“…We report the synthesis and results from the in vitro evaluation of 6-(adamantan-2-ylidene-hydroxybenzoxazole)-O-sulfamate 1 as an irreversible inhibitor of…”
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6
ICAM-1 Expression in a Spontaneously Transformed Human Keratinocyte Cell Line: Characterization by a Simple Cell-ELISA Assay
Published in Journal of investigative dermatology (01-07-1992)“…Interferon gamma (IFN-γ) is known to induce ICAM-1 on keratinocytes (KC) in vitro, and its expression in vivo is correlated with epidermal T-cell infiltration…”
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7
Novel Antiproliferative Agents Derived from Lavendustin A
Published in Journal of medicinal chemistry (01-11-1994)“…The active partial structure of the potent tyrosine kinase inhibitor lavendustin A was derivatized in the search for novel agents against cellular…”
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8
An experimental test of the discreteness-of-charge effect in positive and negative lipid bilayers
Published in Biochemistry (Easton) (16-12-1986)“…The electrostatic properties of charged bilayers and the bilayer component of biological membranes are often described theoretically by assuming the charge is…”
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9
Fluorescent probes of electrostatic potential 1 nm from the membrane surface
Published in Biochemistry (Easton) (01-01-1988)“…We measured the electrostatic potential 1 nm from the surface of charged phospholipid bilayer membranes to test the predictions of the Gouy-Chapman theory…”
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10
Bilayer membranes containing the ganglioside GM1: models for electrostatic potentials adjacent to biological membranes
Published in Biochemistry (Easton) (25-09-1984)“…Although the Gouy-Chapman-Stern theory of the aqueous diffuse double layer describes well the electrostatic potential adjacent to negatively charged…”
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