Search Results - "Willim, K"

941 REGULATION OF THE HEPATOCELLULAR RESPONSE TO ENDOPLASMIC RETICULUM STRESS BY THE TRANSCRIPTION FACTOR C-JUN/AP-1 by Fuest, M, Willim, K, Blum, H.E, Hasselblatt, P

Get full text

The first highly potent and selective non-peptide neuropeptide Y Y1 receptor antagonist: BIBP3226 by Rudolf, K, Eberlein, W, Engel, W, Wieland, H A, Willim, K D, Entzeroth, M, Wienen, W, Beck-Sickinger, A G, Doods, H N

“…The design and subsequent in vitro and in vivo biological characterisation of the first potent and selective non-peptide neuropeptide Y Y1 receptor antagonist,…”
Get more information

Subtype selectivity and antagonistic profile of the nonpeptide Y1 receptor antagonist BIBP 3226 by Wieland, H A, Willim, K D, Entzeroth, M, Wienen, W, Rudolf, K, Eberlein, W, Engel, W, Doods, H N

“…In the present study, the subtype specificity and species selectivity of the nonpeptide BIBP 3226, as well as its in vitro antagonism of neuropeptide Y…”
Get more information

BIBP 3226, the first selective neuropeptide Y1 receptor antagonist: A review of its pharmacological properties by Doods, Henri N., Wieland, Heike A., Engel, Wolfhard, Eberlein, Wolfgang, Willim, Klaus-Dieter, Entzeroth, Michael, Wienen, Wolfgang, Rudolf, Klaus

“…Based on the assumption that the pharmacophoric groups interacting with the Y1 receptor are located in the C-terminal part of neuropeptide Y, low molecular…”
Get full text

Characterization of muscarinic receptors in guinea-pig uterus by Doods, H N, Willim, K D, Boddeke, H W, Entzeroth, M

“…To characterize the muscarinic receptor present in guinea-pig uterus smooth muscle the affinities of a series of 27 muscarinic receptor antagonists for M1 (rat…”
Get more information

Receptor binding profiles of NPY analogues and fragments in different tissues and cell lines by Wieland, H.A., Willim, K., Doods, H.N.

“…To investigate receptor selectivity and possible species selectivity of a number of NPY analogues and fragments, receptor binding studies were performed using…”
Get full text

Labeling of neuropeptide Y receptors in SK-N-MC cells using the novel, nonpeptide Y1 receptor-selective antagonist [3H]BIBP3226 by ENTZEROTH, M, BRAUNGER, H, EBERLEIN, W, ENGEL, W, RUDOLF, K, WIENEN, W, WIELAND, H. A, WILLIM, K.-D, DOODS, H. N

“…The binding of tritium-labelled BIBP3226, N2-(diphenylacetyl)-N-[(4-hydroxy-phenyl)methyl]-D-arginine amide, to human neuroblastoma SK-N-MC cells was…”
Get full text

Divalent cations influencing neuropeptide Y receptor subtype binding in rat hippocampus and cortex membranes as well as in recombinant cells by Wieland, Heike A, Willim, K, Doods, Henri N

“…At least six types of neuropeptide Y (NPY) receptors (Y1–Y6) have been pharmacologically distinguished of which only the Y1, Y2, Y4 and Y5 subtypes have been…”
Get full text

High-affinity analogues of neuropeptide Y containing conformationally restricted non-proteinogenic amino acids by Beck-Sickinger, A G, Hoffmann, E, Paulini, K, Reissig, H U, Willim, K D, Wieland, H A, Jung, G

Get more information

Complete L‐Alanine Scan of Neuropeptide Y Reveals Ligands Binding to Y1 and Y2 Receptors with Distinguished Conformations by Beck‐Sickinger, Annette G., Weland, Heike A., Wittneben, Helmut, Willim, Klaus‐Dieter, Rudolf, Klaus, Jung, Günther

“…The synthesis of more than fifty 36‐residue oligopeptide analogs of neuropeptide Y (NPY) and their affinity to human Y1, and Y2, receptors is described. Each…”
Get full text

Divalent cations influencing neuropeptide Y receptor subtype binding in rat hippocampus and cortex membranes as well as in recombinant cells: Neuropeptide Y by WIELAND, H. A, WILLIM, K, DOODS, H. N

Get full text

A rational approach for the development of reduced-size analogues of neuropeptide Y with high affinity to the Y1 receptor by Rist, B, Wieland, H A, Willim, K D, Beck-Sickinger, A G

“…Four sets of centrally truncated analogues of neuropeptide Y have been synthesized. In each series the N-terminal part was constant, while the C-terminal…”
Get more information

Labeling of neuropeptide Y receptors in SK-N-MC cells using the novel, nonpeptide Y sub(1) receptor-selective antagonist [ super(3)H]BIBP3226 by Entzeroth, M, Braunger, H, Eberlein, W, Engel, W, Rudolf, K, Wienen, W, Wieland, HA, Willim, K D, Doods, H N

“…The binding of tritium-labelled BIBP3226, N super(2)-(diphenylacetyl)-N-[(4-hydroxy-phenyl) methyl]-D-arginine amide, to human neuroblastoma SK-N-MC cells was…”
Get full text

Complete L-alanine scan of neuropeptide Y reveals ligands binding to Y sub(1) and Y sub(2) receptors with distinguished conformations by Beck-Sickinger, A G, Wieland, HA, Wittneben, H, Willim, K-D, Rudolf, K, Jung, G

“…The synthesis of more than fifty 36-residue oligopeptide analogs of neuropeptide Y (NPY) and their affinity to human Y sub(1) and Y sub(2) receptors is…”
Get full text

Propagation Measurements in the Extremely Low Frequency (ELF) Band by White, D., Willim, D.

“…An experimental measurement program has been conducted to determine propagation parameters in the 40-50 and 70-80 Hz ranges. These measurements have utilized a…”
Get full text

Long-range communications at extremely low frequencies by Bernstein, S.L., Burrows, M.L., Evans, J.E., Griffiths, A.S., McNeill, D.A., Niessen, C.W., Richer, I., White, D.P., Willim, D.K.

“…Extremely low frequencies (ELF) are ideal for communicating with deeply submerged submarines because, below 100 Hz, electromagnetic waves penetrate deeply into…”
Get full text

Complete L‐Alanine Scan of Neuropeptide Y Reveals Ligands Binding to Y 1 and Y 2 Receptors with Distinguished Conformations by Beck‐Sickinger, Annette G., Weland, Heike A., Wittneben, Helmut, Willim, Klaus‐Dieter, Rudolf, Klaus, Jung, Günther

“…The synthesis of more than fifty 36‐residue oligopeptide analogs of neuropeptide Y (NPY) and their affinity to human Y 1 , and Y 2 , receptors is described…”
Get full text

Adaptive Equalizer for Pulse Transmission by Niessen, C., Willim, D.

“…Results are reported which are of interest in the automatic adaptive equalization of telephone lines or other narrowbandwidth channels where data transmission…”
Get full text

Labeling of neuropeptide Y receptors in SK-N-MC cells using the novel, nonpeptide Y 1 receptor-selective antagonist [ 3H]BIBP3226 by Entzeroth, Michael, Braunger, Hans, Eberlein, Wolfgang, Engel, Wolfhard, Rudolf, Klaus, Wienen, Wolfgang, Wieland, Heike A., Willim, Klaus-Dieter, Doods, Henri N.

“…The binding of tritium-labelled BIBP3226, N 2-(diphenylacetyl)- N-[(4-hydroxy-phenyl)methyl]- d-arginine amide, to human neuroblastoma SK-N-MC cells was…”
Get full text

Derivative-Discontinuous Electroheat Control by Roots, Willim K., Shridhar, Malayappan

“…In electroheat processes such as induction furnaces, arc furnaces, radiant furnaces, plasma torches, fluidized beds, etc., that are usually discontinuously…”
Get full text