Search Results - "Vitous, J."

Synthesis of nevirapine and its major metabolite by Grozinger, K. G., Fuchs, V., Hargrave, K. D., Mauldin, S., Vitous, J., Campbell, S., Adams, J.

“…Several synthetic methods were developed during the process optimization for the large scale synthesis of nevirapine (1), a non‐nucleoside inhibitor of HIV‐1…”
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Electronic Control of Chiral Quaternary Center Creation in the Intramolecular Asymmetric Heck Reaction by Busacca, Carl A, Grossbach, Danja, Campbell, Scot J, Dong, Yong, Eriksson, Magnus C, Harris, Robert E, Jones, Paul-James, Kim, Ji-Young, Lorenz, Jon C, McKellop, Keith B, O'Brien, Erin M, Qiu, Fenghe, Simpson, Robert D, Smith, Lana, So, Regina C, Spinelli, Earl M, Vitous, Jana, Zavattaro, Chiara

“…The Boehringer-Ingelheim phosphinoimidazoline (BIPI) ligands were applied to the formation of chiral quaternary centers in the asymmetric Heck reaction…”
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Beta-blocking drug metipranolol: plasma levels and pharmacodynamic action in man by Mayer, O, Cepelák, V, Vitous, J, Potmĕsil, J

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The observation of the influence of the unretarded form of xanthinol-niacinate (Complamine) in ulcus cruris venosum on the skin temperature of the lower extremities with the biochemical determination of the levels of the preparation (author's transl) by Resl, Jr, V, Götzová, Vitous, J

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Novel non-nucleoside inhibitors of HIV-1 reverse transcriptase. 1. Tricyclic pyridobenzo- and dipyridodiazepinones by Hargrave, Karl D, Proudfoot, John R, Grozinger, Karl G, Cullen, Ernest, Kapadia, Suresh R, Patel, Usha R, Fuchs, Victor U, Mauldin, Scott C, Vitous, Jana

“…Novel pyrido[2,3-b][1,4]benzodiazepinones (I), pyrido[2,3-b][1,5]benzodiazepinones (II), and dipyrido[3,2-b:2',3'-e][1,4]diazepinones (III) were found to…”
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Inhibition of human leukocyte elastase (HLE) by N-substituted peptidyl trifluoromethyl ketones by Skiles, Jerry W, Fuchs, Victor, Miao, Clara, Sorcek, Ronald, Grozinger, Karl G, Mauldin, Scott C, Vitous, Jana, Mui, Philip W, Jacober, Stephen

“…A series of tripeptides possessing trifluoromethyl or aryl ketone residues at P1 were prepared and evaluated both in vitro and in vivo as potential inhibitors…”
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Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 (HIV-1) reverse transcriptase. IV: 2-substituted dipyridodiazepinones as potent inhibitors of both wild-type and cysteine-181 HIV-1 reverse transcriptase enzymes by PROUDFOOT, J. R, HARGRAVE, K. D, ROSE, J, DAVID, E, MAULDIN, S. C, FUCHS, V. U, VITOUS, J, HOERMANN, M, KLUNDER, J. M, PALAYAKOTAI RAGHAVAN, SKILES, J. W, MUI, P, KAPADIA, S. R, RICHMAN, D. D, SULLIVAN, J. L, CHENG-KON SHIH, GROB, P. M, ADAMS, J, PATEL, U. R, GROZINGER, K. G, MCNEIL, D. W, CULLEN, E, CARDOZO, M, LIANG TONG, KELLY, T. A

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Clinical pharmacology of Metipranolol (trimepranol injection VUFB, Spofa tablets). The importance of clinical dosages by Mayer, O, Cepelák, V, Vitous, J

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Novel non-nucleoside inhibitors of HIV-1 reverse transcriptase. I, Tricyclic pyridobenzo- and dipyridodiazepinones by HARGRAVE, K. D, PROUDFOOT, J. R, KLUNDER, J. M, PAL, K, SKILES, J. W, MCNEIL, D. W, ROSE, J. M, CHOW, G. C, SKOOG, M. T, WU, J. C, SCHMIDT, G, ENGEL, W. W, GROZINGER, K. G, CULLEN, E, KAPADIA, S. R, PATEL, U. R, FUCHS, V. U, MAULDIN, S. C, VITOUS, J, BEHNKE, M. L

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Clinical pharmacology of trimepranol (pharmacokinetic informations and effects on heart rate in healthy individuals) by Mayer, O, Petrlík, M, Vitous, J, Cepelák, V

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Utilization of injected choline by the brain and ileum of albino rats

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Activity of heart pacemaker and thyroid hormone level in the blood of guinea pigs of different age by Vitous, J, Vlk, J

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Evaluation of the biologic availability of drugs under clinical conditions by Cepelák, V, Mayer, O, Cepeláková, H, Vitous, J, Petrlík, M

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