Search Results - "Vinodini, Arun"

Development and Execution of an Ni(II)-Catalyzed Reductive Cross-Coupling of Substituted 2-Chloropyridine and Ethyl 3-Chloropropanoate by Nimmagadda, Sri Krishna, Korapati, Satish, Dasgupta, Debottam, Malik, Noormohamed Abdul, Vinodini, Arun, Gangu, Aravind S., Kalidindi, Srinivas, Maity, Prantik, Bondigela, Siva Sankar, Venu, Alla, Gallagher, William P., Aytar, Selin, González-Bobes, Francisco, Vaidyanathan, Rajappa

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Development of a Safer Continuous Flow Process for B2(OH)4‑Mediated Chemoselective Reduction of Nitroarenes to Anilines by Revu, Omkar, Vasilev, Maksim, Gajula, Praveen, Kalikinidi, Nageswara Rao, Gadi, Madhusudhan Reddy, Zhao, Huiping, Gamage, Shanika M. P., Hibbert, Graham, Ravikumar, Ongolu, Gummidi, Lalitha, Nasipireddy, Venkatarathnam, Vinodini, Arun, Bietsch, Jonathan, Wang, Zhirui, Brown, Jack D., Sirasani, Gopal, Armstrong, Joseph D., Gangu, Aravind S., Qu, Bo, Senanayake, Chris H.

“…Tetrahydroxydiboron [B2(OH)4] is a chemoselective reducing reagent for nitro reductions in the presence of other labile functional groups. However, there are…”
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Development of a Safer Continuous Flow Process for B 2 (OH) 4 -Mediated Chemoselective Reduction of Nitroarenes to Anilines by Revu, Omkar, Vasilev, Maksim, Gajula, Praveen, Kalikinidi, Nageswara Rao, Gadi, Madhusudhan Reddy, Zhao, Huiping, Gamage, Shanika M. P., Hibbert, Graham, Ravikumar, Ongolu, Gummidi, Lalitha, Nasipireddy, Venkatarathnam, Vinodini, Arun, Bietsch, Jonathan, Wang, Zhirui, Brown, Jack D., Sirasani, Gopal, Armstrong, Joseph D., Gangu, Aravind S., Qu, Bo, Senanayake, Chris H.

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Development of a Scalable Synthetic Route to BMS-986251. Part 1: Synthesis of the Cyclohexane Dicarboxylate Fragment by Kuppusamy, Sankar, Gangu, Aravind S, Kalidindi, Srinivas, Ponnusamy, Muthukrishnan, Tendulkar, Shankar, Venu, Alla, Palani, Senthil, Nagappan, Vedhachalam, Vinodini, Arun, Mudryk, Boguslaw, Rupasinghe, Sanjeewa, Joe, Candice L, Coombs, John R, Gallagher, William P, Kopp, Nathaniel, Gonzalez-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa

“…The cyclohexane dicarboxylate unit of BMS-986251 (1), a potent and efficacious RORγt inverse agonist, was synthesized starting from Hagemann’s ester in seven…”
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Development of a Scalable Synthetic Route to BMS-986251, Part 2: Synthesis of the Tricyclic Core and the API by Kalidindi, Srinivas, Gangu, Aravind S, Kuppusamy, Sankar, Sathasivam, Shunmugaraj, Shekarappa, Vijaykumar, Murugan, Saravanan, Bondigela, Sivasankar, Kandasamy, Moorthy, Ghanta, Kishore, Vinodini, Arun, Shrikant, Abhishek, Ramachandran, Ravikumar, Gallagher, William P, Kopp, Nathaniel, González-Bobes, Francisco, Eastgate, Martin D, Vaidyanathan, Rajappa

“…BMS-986251, a potent and efficacious RORγt inverse agonist, was synthesized starting from 6-iodotetralone using 13 chemical transformations with only eight…”
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