Search Results - "Vigorita, Maria Gabriella"

In vitro antiproliferative activity against human colon cancer cell lines of representative 4-thiazolidinones. Part I by Ottanà, Rosaria, Carotti, Stefania, Maccari, Rosanna, Landini, Ida, Chiricosta, Giuseppa, Caciagli, Barbara, Vigorita, Maria Gabriella, Mini, Enrico

“…The characterization of two cyclooxygenase isoforms (COX), the rate-limiting enzyme for the synthesis of prostaglandins (PGs) from arachidonic acid, has…”
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Evaluation of in vitro aldose redutase inhibitory activity of 5-arylidene-2,4-thiazolidinediones by Maccari, Rosanna, Ottanà, Rosaria, Ciurleo, Rosella, Vigorita, Maria Gabriella, Rakowitz, Dietmar, Steindl, Theodora, Langer, Thierry

“…A number of 5-arylidene-2,4-thiazolidinediones containing a hydroxy or a carboxymethoxy group in their 5-benzylidene moiety have been synthesised and evaluated…”
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In vitro advanced antimycobacterial screening of isoniazid-related hydrazones, hydrazides and cyanoboranes: Part 14 by Maccari, Rosanna, Ottanà, Rosaria, Vigorita, Maria Gabriella

“…The in vitro antimycobacterial activities of some isoniazid derivatives are reported. As a part of an ongoing search for new isoniazid-related…”
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5-Arylidene-2,4-thiazolidinediones as inhibitors of protein tyrosine phosphatases by Maccari, Rosanna, Paoli, Paolo, Ottanà, Rosaria, Jacomelli, Michela, Ciurleo, Rosella, Manao, Giampaolo, Steindl, Theodora, Langer, Thierry, Vigorita, Maria Gabriella, Camici, Guido

“…4-(5-Arylidene-2,4-dioxothiazolidin-3-yl)methylbenzoic acids ( 2) were synthesized and evaluated in vitro as inhibitors of PTP1B and LMW-PTP, two protein…”
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Synthesis and in vitro evaluation of 5-arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones with antidegenerative activity on human chondrocyte cultures by Ottanà, Rosaria, Maccari, Rosanna, Ciurleo, Rosella, Vigorita, Maria Gabriella, Panico, Anna Maria, Cardile, Venera, Garufi, Floriana, Ronsisvalle, Simone

“…5-Arylidene-3-hydroxyalkyl-2-phenylimino-4-thiazolidinones ( 7, 8) were synthesized and evaluated for their antidegenerative activity on human chondrocyte…”
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In vitro aldose reductase inhibitory activity of 5-benzyl-2,4-thiazolidinediones by Rakowitz, Dietmar, Maccari, Rosanna, Ottanà, Rosaria, Vigorita, Maria Gabriella

“…Several 5-benzyl-2,4-thiazolidinediones ( 5– 7) were synthesised and tested as in vitro aldose reductase (ALR2) inhibitors. Most of them, particularly…”
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In Vitro Antimycobacterial Activities of 2′-Monosubstituted Isonicotinohydrazides and Their Cyanoborane Adducts by MACCARI, Rosanna, OTTANA, Rosaria, MONFORTE, Francesca, VIGORITA, Maria Gabriella

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
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Modeling and biological evaluation of 3,3′-(1,2-ethanediyl)bis[2-(4-methoxyphenyl)-thiazolidin-4-one], a new synthetic cyclooxygenase-2 inhibitor by Ottaná, Rosaria, Mazzon, Emanuela, Dugo, Laura, Monforte, Francesca, Maccari, Rosanna, Sautebin, Lidia, De Luca, Grazia, Vigorita, Maria Gabriella, Alcaro, Stefano, Ortuso, Francesco, Caputi, Achille P, Cuzzocrea, Salvatore

“…Within the series of chiral 3,3′-(1,2-ethanediyl)bis[2-arylthiazolidin-4-ones], the 3,4-dimethoxyphenyl substituted derivative was found in the primary…”
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Facile Biocatalytic Access to 9-Fluorenylmethyl Polyglycosides: Evaluation of Antiviral Activity on Immunocompetent Cells by Tramice, Annabella, Arena, Adriana, De Gregorio, Ambra, Ottanà, Rosaria, Maccari, Rosanna, Pavone, Bernadette, Arena, Nicoletta, Iannello, Daniela, Vigorita, Maria Gabriella, Trincone, Antonio

“…The biological activities of a series of mono‐ and oligosaccharides (β‐xylosides and α‐glucosides) of 9‐fluorenylmethanol were investigated together with…”
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9-Fluorenon-4-carboxamides: synthesis, conformational analysis, anti-HSV-2, and immunomodulatory evaluation. Note II by Alcaro, Stefano, Arena, Adriana, Bella, Rosaria Di, Neri, Simonetta, Ottanà, Rosaria, Ortuso, Francesco, Pavone, Bernadette, Vigorita, Maria Gabriella

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5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel anti-inflammatory agents by Ottanà, Rosaria, Maccari, Rosanna, Barreca, Maria Letizia, Bruno, Giuseppe, Rotondo, Archimede, Rossi, Antonietta, Chiricosta, Giuseppa, Di Paola, Rosanna, Sautebin, Lidia, Cuzzocrea, Salvatore, Vigorita, Maria Gabriella

“…[Display omitted] The synthesis and pharmacological activity of 5-arylidene-2-imino-4-thiazolidinones ( 3a– 8a) are described. All derivatives exhibited…”
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Structure–activity relationships and molecular modelling of 5-arylidene-2,4-thiazolidinediones active as aldose reductase inhibitors by Maccari, Rosanna, Ottanà, Rosaria, Curinga, Carmela, Vigorita, Maria Gabriella, Rakowitz, Dietmar, Steindl, Theodora, Langer, Thierry

“…[Display omitted] The structure–activity relationships (SARs) of 5-arylidene-2,4-thiazolidinediones active as aldose reductase inhibitors (ARIs) were extended…”
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Rational Design, Synthesis, Biophysical and Antiproliferative Evaluation of Fluorenone Derivatives with DNA G-Quadruplex Binding Properties by Alcaro, Stefano, Artese, Anna, Iley, James N., Missailidis, Sotiris, Ortuso, Francesco, Parrotta, Lucia, Pasceri, Raffaele, Paduano, Francesco, Sissi, Claudia, Trapasso, Francesco, Vigorita, Maria Gabriella

“…Molecular modeling studies carried out with experimental DNA models with the sequence d[AG3(T2AG3)3] suggest that the introduction of a net positive charge…”
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In vitro advanced antimycobacterial screening of cobalt(II) and copper(II) complexes of fluorinated isonicotinoylhydrazones by Maccari, Rosanna, Ottanà, Rosaria, Bottari, Bruno, Rotondo, Enrico, Vigorita, Maria Gabriella

“…The in vitro antimycobacterial activities of metalcomplexes 1, 2 are reported. The in vitro antimycobacterial activity of cobalt(II) and copper(II) complexes…”
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2/4-Substituted-9-fluorenones and their O-glucosides as potential immunomodulators and anti-herpes simplex virus-2 agents. Part 5 by Arena, Adriana, Arena, Nicoletta, Ciurleo, Rosella, de Gregorio, Ambra, Maccari, Rosanna, Ottana', Rosaria, Pavone, Bernadette, Tramice, Annabella, Trincone, Antonio, Vigorita, Maria Gabriella

“…In pursuing a research on the antiviral and immunomodulatory activity of tilorone congeners, two new series of compounds were prepared and pharmacologically…”
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Tetraplex DNA specific ligands based on the fluorenone-carboxamide scaffold by Alcaro, Stefano, Artese, Anna, Iley, James N., Maccari, Rosanna, Missailidis, Sotiris, Ortuso, Francesco, Ottanà, Rosaria, Ragazzon, Patricia, Vigorita, Maria Gabriella

“…A series of fluorenone-carboxamide compounds was analyzed with regard to DNA binding properties by UV spectroscopy and competition dialysis methods. The…”
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2/4-Substituted-9-fluorenones and their 0-glucosides as potential immunomodulators and anti-herpes simplex virus-2 agents. Part 5 by ARENA, Adriana, ARENA, Nicoletta, CIURLEO, Rosella, DE GREGORIO, Ambra, MACCARI, Rosanna, OTTANA', Rosaria, PAVONE, Bernadette, TRAMICE, Annabella, TRINCONE, Antonio, GABRIELLA VIGORITA, Maria

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Biocatalysed synthesis of β- O-glucosides from 9-fluorenon-2-carbohydroxyesters. Part 3: IFN-inducing and anti-HSV-2 properties by Alcaro, Stefano, Arena, Adriana, Di Bella, Rosaria, Neri, Simonetta, Ottanà, Rosaria, Ortuso, Francesco, Pavone, Bernadette, Trincone, Antonio, Vigorita, Maria Gabriella

“…[Display omitted] In pursuing research on the antiviral, interferon (IFN)-inducing tilorone congeners, a new series of fluoren-carboxyhydroxyesters has been…”
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Configurational assignments of the diastereomers of 3,3′-(1,2-ethanediyl)bis[2-(3-fluorophenyl)-5-methyl-4-thiazolidinone] derivative with four stereogenic centers by Vigorita, Maria Gabriella, Ottaná, Rosaria, Monforte, Francesca, Previtera, Tindara, Maccari, Rosanna

“…Diastereomers of antiinflammatory/analgesic and antihistaminic 3,3′[(1,2‐ethanediyl)bis(2‐aryl‐4‐thiazo‐lidinone)] derivatives possessing two stereogenic…”
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2'-[1-(4-Fluorophenyl)ethyl]isonicotino-κN-hydrazide-Cyanoborane by Bruno, G., Maccari, R., Nicoló, F., Ottaná, R., Panzalorto, M., Scopelliti, R., Vigorita, M. G.

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