Search Results - "Vasilevich, N I"

Design and development of macrocyclization methods for compounds with potential tuberculocidal activity to decrease CYP450 liver cytochrome inhibition by Vasilevich, N. I., Aksenova, E. A., Aksenova, A. A., Afanasyev, I. I.

“…A procedure for macrocyclization of compounds with potential tuberculocidal activity was developed in order to obtaining compounds with a lower degree of…”
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Synthesis and antiamnesic activity of a series of N-acylprolyl-containing dipeptides by Gudasheva, TA, Voronina, TA, Ostrovskaya, RU, Rozantsev, GG, Vasilevich, NI, Trofimov, SS, Kravchenko, EV, Skoldinov, AP, Seredenin, SB

“…Esters and amides of a series of N-acylprolyl-containing dipeptides were synthesized. It was established that these substances possess the ability to prevent…”
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Aminopyridine- and aminopyrimidine-based serine/threonine protein kinase inhibitors are drug candidates for treating drug-resistant tuberculosis by Maslov, D. A., Bekker, O. B., Alekseeva, A. G., Kniazeva, L. M., Mavletova, D. A., Afanasyev, I. I., Vasilevich, N. I., Danilenko, V. N.

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Examination of the 1,4-disubstituted azetidinone ring system as a template for combretastatin A-4 conformationally restricted analogue design by SUN, Lichun, VASILEVICH, Natalya I, FUSELIER, Joseph A, HOCART, Simon J, COY, David H

“…A series of novel 1,4-diaryl-2-azetidinones was prepared by stereospecific Staudinger reaction as conformationally restricted analogues of combretastatin A-4…”
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Conversion of O -succinimidyl carbamates to N -( O -carbamoyl)-succinmonoamides and ureas: effects of N -substituents and reaction conditions on the reaction pathway by Vasilevich, Natalya I., Coy, David H.

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Abilities of 3,4-Diarylfuran-2-one Analogs of Combretastatin A-4 to Inhibit Both Proliferation of Tumor Cell Lines and Growth of Relevant Tumors in Nude Mice by LICHUN SUN, VASILEVICH, Natalya I, FUSELIER, Joseph A, COY, David H

“…Background: Combretastatin A-4 (CA-4) and its analogs are potent inhibitors of tubulin polymerization and display strong inhibitory activity on both solid…”
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Selective conversion of O-succinimidyl carbamates to N-( O-carbamoyl)-succinmonoamides and ureas by Vasilevich, Natalya I., Sachinvala, Navzer D., Maskos, Karol, Coy, David H.

“…N-Monoalkyl- O-succinimidyl carbamates reacted with primary and secondary amines to produce ureas. However, N, N-dialkyl- O-succinimidyl carbamates reacted…”
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Synthesis and nootropic activity of pyrrolidino[1,2-a]diazacycloalkanes by Gudasheva, T. A., Vasilevich, N. I., Ostrovskaya, R. U., Trofimov, S. S., Voronina, T. A., Skoldinov, A. P., Rozantsev, G. G.

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The use of the HPLC method for the quantitative determination of a peptide analog of piracetam with nootropic activity and its main metabolites by Boĭko, S S, Zherdev, V P, Gudasheva, T A, Vasilevich, N I, Ostrovskaia, R U, Voronina, T A, Rozantsev, G G

“…HPLC method has been developed for pharmacokinetic study of nootropic peptide analog of pyracetam GVS-111 and its main metabolites. In the model experiments on…”
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Synthesis and antiamnesic activity of a series of N-acylprolyl-containing dipeptides by GUDASHEVA, T. A, VORONINA, T. A, OSTROVSKAYA, R. U, ROZANTSEV, G. G, VASILEVICH, N. I, TROFIMOV, S. S, KRAVCHENKO, E. V, SKOLDINOV, A. P, SEREDENIN, S. B

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Nootropic action of proline-based topological analogs of piracetam by Gudasheva, T. A., Vasilevich, N. I., Zolotov, N. N., Lezina, V. P., Rozenberg, S. G., Kravchenko, E. V., Ostrovskaya, R. U., Voronina, T. A., Rozantsev, G. G., Skoldinov, A. P.

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