Search Results - "Thopate, Yogesh"
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Synthesis and in vitro SAR evaluation of natural vanillin-based chalcones tethered quinolines as antiplasmodial agents
Published in Medicinal chemistry research (01-12-2022)“…A series of novel chalcone derivatives were synthesized and investigated against the chloroquine-sensitive P. falciparum 3D7 ( Pf 3D7) strain and…”
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2
Chemical Protein Synthesis by Native Chemical Ligation and Variations Thereof
Published in Chinese journal of chemistry (01-11-2019)“…For a long time, the total synthesis of proteins was considered as a “mission impossible” because of the tedious and complex synthetic steps and demanding…”
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Synergistic Cooperative Effect of L‐Arginine‐[bmim]Br in Cascade Decarboxylative Knoevenagel‐Thia‐Michael Addition Reactions: Green Approach Towards C−S Bond Formation with In Situ Generated Unactivated α,β‐Unsaturated Ester
Published in Advanced synthesis & catalysis (16-11-2018)“…In this report, a synergistic combination of L‐arginine and [bmim]Br has been realized for the first time towards step‐economical synthesis of…”
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Cascade Multicomponent Reaction Involving Unprecedented Gould Jacobs‐Heck/Suzuki Coupling‐Hydrolysis‐Decarboxylation Reactions in One Pot: Rapid Synthesis of Hybrid Heterocyclic Molecules
Published in Asian journal of organic chemistry (01-08-2022)“…Multicomponent reaction (MCR) has been one of the strong pillars of green chemistry. In this respect we herein report a multicomponent 5 step reaction in one…”
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A facile tandem double-dehydrative-double-Heck olefination strategy for pot-economic synthesis of (E)-distyrylbenzenes as multi-target-directed ligands against Alzheimer's disease employing C. elegans model
Published in Tetrahedron (05-04-2018)“…A concise, one pot and regioselective access to (E)-distyrylbenzenes (DSBs) from arylhalide and secondary phenylenediethanol, a stable precursor for in situ…”
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Palladium-Catalyzed Dehydrative Heck Olefination of Secondary Aryl Alcohols in Ionic Liquids: Towards a Waste-Free Strategy for Tandem Synthesis of Stilbenoids
Published in Angewandte Chemie International Edition (12-03-2012)“…All in one: A tandem strategy has been developed wherein secondary aryl alcohols are directly coupled with aryl halides to provide stilbenoids through a…”
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NMR and DFT Insight into the Synergistic Role of Bovine Serum Albumin-Ionic Liquid for Multicomponent Cascade Aldol/Knoevenagel-thia-Michael/Michael Reactions in One Pot
Published in ChemCatChem (06-10-2016)“…The synergistic combination of two catalysts is an emerging strategy towards the formation of unprecedented complex molecules, and herein bovine serum albumin…”
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A Highly Regioselective and Practical Synthesis of α‐Aryl Ketones under a Cooperative Cascade Effect of an Ionic Liquid and Tetrabutylammonium Fluoride
Published in Asian journal of organic chemistry (01-11-2019)“…A metal‐free regioselective synthesis of α‐aryl ketone from corresponding bromohydrin via cooperative cascade effect of [hmim]Br and tetrabutylammonium…”
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Towards a Step‐Economical and Waste‐Free [hmim]Br‐Catalyzed Deprotection of β‐Sulfido Carbonyl Groups into (E)‐Enones and Mechanistic Insights
Published in Asian journal of organic chemistry (01-12-2017)“…A neutral ionic liquid, [hmim]Br, catalyzed the direct dehydrosulfenylation of β‐sulfido carbonyl compounds under microwave irradiation into the corresponding…”
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Towards a Step-Economical and Waste-Free [hmim]Br-Catalyzed Deprotection of [beta]-Sulfido Carbonyl Groups into (E)-Enones and Mechanistic Insights
Published in Asian journal of organic chemistry (01-12-2017)“…A neutral ionic liquid, [hmim]Br, catalyzed the direct dehydrosulfenylation of [beta]-sulfido carbonyl compounds under microwave irradiation into the…”
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11
Palladium-Catalyzed Dehydrative Heck Olefination of Secondary Aryl Alcohols in Ionic Liquids: Towards a Waste-Free Strategy for Tandem Synthesis of Stilbenoids
Published in Angewandte Chemie (12-03-2012)“…Alles in einem: Eine Tandemstrategie wurde entwickelt, mit der sekundäre Arylalkohole direkt mit Arylhalogeniden gekuppelt wurden. Die Reaktion liefert…”
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