Search Results - "Thimmalapura, Vishwanatha M"

Thioacids - synthons for amide bond formation and ligation reactions: assembly of peptides and peptidomimetics by N, Narendra, Thimmalapura, Vishwanatha M, Hosamani, Basavaprabhu, Prabhu, Girish, Kumar, L Roopesh, Sureshbabu, Vommina V

“…The synthesis of α-amino thioacids and peptide thioacids and their applications in chemoselective amide bond formation, ligation of…”
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Synthesis of Nβ‑Protected Amino Sulfenyl Methyl Formamides and Sulfonyl Methyl Formamides: A Simple Protocol by Srinivasulu, Chinthaginjala, Sagar, Nagamangala R, Vishwanatha, Thimmalapura M, Durgamma, Suram, Sureshbabu, Vommina V

“…Chiral amino acid-derived formamides represent one of the most versatile components in multicomponent reactions. Herein, we describe a facile synthesis of…”
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Tubulysin Synthesis Featuring Stereoselective Catalysis and Highly Convergent Multicomponent Assembly by Vishwanatha, Thimmalapura M, Giepmans, Ben, Goda, Sayed K, Dömling, Alexander

“…A concise and modular total synthesis of the highly potent N14-desacetoxytubulysin H (1) has been accomplished in 18 steps in an overall yield of up to 30%…”
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Sulfur-Switch Ugi Reaction for Macrocyclic Disulfide-Bridged Peptidomimetics by Vishwanatha, Thimmalapura M, Bergamaschi, Enrico, Dömling, Alexander

“…A general strategy is introduced for the efficient synthetic access of disulfide linked artificial macrocycles via a Ugi four-component reaction (U4CR)…”
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A Pro‐Fluorescent Ubiquitin‐Based Probe to Monitor Cysteine‐Based E3 Ligase Activity by Pérez Berrocal, David A., Vishwanatha, Thimmalapura M., Horn‐Ghetko, Daniel, Botsch, J. Josephine, Hehl, Laura A., Kostrhon, Sebastian, Misra, Mohit, Ðikić, Ivan, Geurink, Paul P., Dam, Hans, Schulman, Brenda A., Mulder, Monique P. C.

“…Protein post‐translational modification with ubiquitin (Ub) is a versatile signal regulating almost all aspects of cell biology, and an increasing range of…”
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Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles by Vishwanatha, Thimmalapura M, Kurpiewska, Katarzyna, Kalinowska-Tłuścik, Justyna, Dömling, Alexander

“…An alternative approach toward the simple and robust synthesis of highly substituted peptidic thiazole derivatives using Ugi-multicomponent reaction (U-MCR) is…”
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A Pro‐Fluorescent Ubiquitin‐Based Probe to Monitor Cysteine‐Based E3 Ligase Activity by Pérez Berrocal, David A., Vishwanatha, Thimmalapura M., Horn‐Ghetko, Daniel, Botsch, J. Josephine, Hehl, Laura A., Kostrhon, Sebastian, Misra, Mohit, Ðikić, Ivan, Geurink, Paul P., Dam, Hans, Schulman, Brenda A., Mulder, Monique P. C.

“…Protein post‐translational modification with ubiquitin (Ub) is a versatile signal regulating almost all aspects of cell biology, and an increasing range of…”
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Synthesis of 1, 5‐ Disubstituted Tetrazole via Ugi Azide Reaction: An Asymmetric Induction Approach by Santhosh, L., Nagamangala, Sagar R., Thimmalapura, Vishwanatha M., Vommina, Sureshbabu V.

“…The Ugi‐azide reaction of an enantiopure amino acid derived isocyanides, amino acid esters, aldehydes and TMS‐N3 in MeOH:THF solvent system at 50 °C yielded…”
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