Search Results - "Temnyakova, Nadezhda S."

5-Nitroisoxazoles in SNAr Reactions: A Novel Chemo- and Regioselective Approach to Isoxazole-Based Bivalent Ligands of AMPA Receptors by Vasilenko, Dmitry A., Temnyakova, Nadezhda S., Dronov, Sevastian E., Radchenko, Eugene V., Grishin, Yuri K., Gabrel’yan, Alexey V., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Averina, Elena B., Palyulin, Vladimir A.

“…An efficient regioselective approach to novel functionalized bis(isoxazoles) with a variety of aromatic and aliphatic linkers was elaborated, based on the…”
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Biphenyl scaffold for the design of NMDA-receptor negative modulators: molecular modeling, synthesis, and biological activity by Karlov, Dmitry S, Temnyakova, Nadezhda S, Vasilenko, Dmitry A, Barygin, Oleg I, Dron, Mikhail Y, Zhigulin, Arseniy S, Averina, Elena B, Grishin, Yuri K, Grigoriev, Vladimir V, Gabrel'yan, Alexey V, Aniol, Viktor A, Gulyaeva, Natalia V, Osipenko, Sergey V, Kostyukevich, Yury I, Palyulin, Vladimir A, Popov, Petr A, Fedorov, Maxim V

“…NMDA ( N -methyl- d -aspartate) receptor antagonists are promising tools for the treatment of a wide variety of central nervous system impairments including…”
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5-Nitroisoxazoles in ISNAr/I Reactions: A Novel Chemo- and Regioselective Approach to Isoxazole-Based Bivalent Ligands of AMPA Receptors by Vasilenko, Dmitry A, Temnyakova, Nadezhda S, Dronov, Sevastian E, Radchenko, Eugene V, Grishin, Yuri K, Gabrel’yan, Alexey V, Zamoyski, Vladimir L, Grigoriev, Vladimir V, Averina, Elena B, Palyulin, Vladimir A

“…An efficient regioselective approach to novel functionalized bis(isoxazoles) with a variety of aromatic and aliphatic linkers was elaborated, based on the…”
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Novel bivalent positive allosteric AMPA receptor modulator of bis-amide series by Temnyakova, Nadezhda S., Vasilenko, Dmitry A., Lavrov, Mstislav I., Karlov, Dmitry S., Grishin, Yuri K., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Averina, Elena B., Palyulin, Vladimir A.

“…[Display omitted] A series of bis-amides of bis(aminoalkyl)benzenes and diaminoalkanes were synthesized. Positive modulation of kainate-induced transmembrane…”
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New nanomolar negative modulators of AMPA receptors by Temnyakova, Nadezhda S., Vasilenko, Dmitry A., Lavrov, Mstislav I., Karlov, Dmitry S., Grishin, Yuri K., Zamoyski, Vladimir L., Grigoriev, Vladimir V., Averina, Elena B., Palyulin, Vladimir A.

“…[Display omitted] Bisamides of 1,4-bis(aminomethyl)benzene with cyclopropane-, cyclobutane- and cyclopentanecarboxylic acids reveal the negative modulation of…”
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Ifenprodil-like NMDA receptor modulator based on the biphenyl scaffold by Temnyakova, Nadezhda S., Vasilenko, Dmitry A., Barygin, Oleg I., Dron, Mikhail Y., Averina, Elena B., Grishin, Yuri K., Grigoriev, Vladimir V., Palyulin, Vladimir A., Fedorov, Maxim V., Karlov, Dmitry S.

“…[Display omitted] Ifenprodil-like NMDA receptor negative allosteric modulator based on the biphenyl scaffold has been identified using virtual screening…”
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