Search Results - "Telvekar, Vikas N."
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Efficient protocol for the synthesis of quinoxaline, benzoxazole and benzimidazole derivatives using glycerol as green solvent
Published in Tetrahedron letters (26-10-2011)“…A straightforward, efficient and more sustainable catalyst-free method has been developed for the synthesis of quinoxaline, benzoxazole, and benzimidazole ring…”
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2
Synthesis and evaluation of novel chloropyrrole molecules designed by molecular hybridization of common pharmacophores as potential antimicrobial agents
Published in Bioorganic & medicinal chemistry letters (01-10-2010)“…In an attempt to identify new potential lead as antimicrobial agent, 31 novel chloropyrrole derivatives of aroyl hydrazones and chalcones incorporating common…”
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3
Readily switchable one-pot 5-exo-dig cyclization using a palladium catalyst
Published in RSC advances (2017)“…A convenient, ligand-free, Pd(OAc) 2 -catalyzed one-pot reaction has been developed for the synthesis of oxazolines and oxazoles from easily available acid…”
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4
One pot synthesis of aromatic azide using sodium nitrite and hydrazine hydrate
Published in Tetrahedron letters (06-03-2013)“…A simple, rapid, and efficient protocol for the synthesis of aryl azide using sodium nitrite and hydrazine hydrate at room temperature is discussed. The short…”
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5
Novel 2-(2-benzylidenehydrazinyl)benzo[d]thiazole as potential antitubercular agents
Published in Combinatorial chemistry & high throughput screening (01-03-2013)“…Molecular hybridization approach was used to synthesize substituted 2-(2-(4-aryl oxy benzylidene) hydrazinyl)benzo thiazole derivatives with…”
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6
Simple and Efficient Method for the Preparation of Aryl Azides Using Sonication
Published in Synthetic communications (01-04-2012)“…An efficient procedure for the preparation of aryl azides using sonication is described. The convenient sonication-mediated azidation protocol is applicable to…”
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7
Simple and Facile Benzylic C-H Oxidation Using (Diacetoxyiodo)benzene and Catalytic Sodium Azide
Published in Synthetic communications (01-05-2012)“…A synthetic utility of hypervalent iodine reagent, (diacetoxyiodo)benzene, with a catalytic amount of sodium azide for oxidation of benzylic C-H to…”
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8
Efficient Synthesis of Bis(4-Dimethaminophenyl)arylmethanes and Bis(4-Diamethaminophenyl)alkanes Using Iodine Reagent
Published in Synthetic communications (18-07-2013)“…A novel synthetic utility of NaICl 2 for the preparation of bis(4-dimethaminophenyl)arylmethanes and bis(4-dimethaminophenyl)alkanes is described. In the…”
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9
Selective Oxidation of Hydrazides Using o-Iodoxybenzoic Acid to Carboxylic Acids, Esters, and Aldehydes
Published in Chemistry letters (05-06-2010)“…A selective method for conversion of hydrazide to corresponding aldehydes, acids, and esters by using hypervalent iodine reagent o-iodoxybenzoic acid (IBX) has…”
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10
Oxidation of Dihydrazones of Diaryl α-Diketones to Diarylacetylenes Using Sodium Periodate
Published in Chemistry letters (05-12-2010)“…Oxidation of dihydrazones of α-diketones to acetylene was investigated by using sodium periodate. Further, the described method is also found to be suitable…”
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11
Synthesis and biological evaluation of novel N' (4-aryloxybenzylidene)- 1H-benzimidazole-2 carbohydrazide derivatives as anti-tubercular agents
Published in Combinatorial chemistry & high throughput screening (01-01-2014)“…A series of structurally novel, (E)-N'-(4-aryloxybenzylidene)-1H-benzimidazole-2-carbohydrazide derivatives were synthesized by molecular hybridization…”
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12
Novel 2-(2-(4-aryloxybenzylidene) hydrazinyl)benzothiazole derivatives as anti-tubercular agents
Published in Bioorganic & medicinal chemistry letters (01-01-2012)“…A series of structurally novel, substituted 2-(2-(4-aryloxybenzylidene) hydrazinyl)benzothiazole derivatives incorporating 2-hydrazinyl benzothiazole and…”
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13
One-Pot Multicomponent Synthesis of 3-Methyl-4-(Hetero)Arylmethylene Isoxazole-5(4H)-Ones Using Guanidine Hydrochloride as the Catalyst under Aqueous Conditions
Published in Polycyclic aromatic compounds (21-10-2022)“…Here, we have developed an expeditious and efficient protocol for the synthesis of isoxazole-5(4H)-ones derivatives using guanidine hydrochloride as a catalyst…”
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14
Concentrated solar radiation-assisted one-pot/multicomponent synthesis of pyranopyrazole derivatives under neat condition
Published in Research on chemical intermediates (01-10-2021)“…Concentrated solar radiation (CSR)-assisted synthesis of pyranopyrazole derivatives under solvent and catalyst-free condition has been reported in the present…”
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15
Silica chloride (SiO2-Cl) catalyzed one pot synthesis of 2,3-disubstituted-thiazolidin-4-one
Published in Synthetic communications (02-05-2020)“…In this paper, we report one-pot, three-component cyclo condensation of an aldehyde, an amine and thioglycolic acid to form 2,3-disubstituted-thiazolidin-4-one…”
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16
Transferrin conjugates of antitubercular drug isoniazid: Synthesis and in vitro efficacy
Published in European journal of medicinal chemistry (01-12-2019)“…Tuberculosis (TB) caused by Mycobacterium tuberculosis (Mtb) has become the world's leading killer disease due to a single infectious agent which survives in…”
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17
Novel peptidomimetic peptide deformylase (PDF) inhibitors of Mycobacterium tuberculosis
Published in Chemical biology & drug design (01-01-2021)“…Emergence of MDR‐TB and XDR‐TB led to the failure of available anti‐tubercular drugs. In order to explore, identify and develop new anti‐tubercular drugs,…”
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18
ZSM-5 catalyzed one pot three-component synthesis of 5-substituted-1H-tetrazoles from aldehyde
Published in Synthetic communications (17-12-2019)“…In this paper, we report one-pot three-component synthesis of 5-substituted-1H-tetrazoles from aldehyde using zeolite-based heterogeneous catalyst (ZSM-5)…”
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One pot synthesis of α‐N‐heteroaryl ketone derivatives from aryl ketones using aqueous NaICl2
Published in Journal of heterocyclic chemistry (01-04-2022)“…A simple and efficient method for the synthesis of α‐heteroaryl ketones from aryl ketones and amine using aqueous sodium dichloroiodate is established. This…”
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20
Novel N′-benzylidene benzofuran-3-carbohydrazide derivatives as antitubercular and antifungal agents
Published in Bioorganic & medicinal chemistry letters (15-03-2012)“…Tuberculosis constitutes today a serious threat to human health worldwide, aggravated by the increasing number of identified multi-drug resistant strains of…”
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