Search Results - "Telser, Joachim"

Structure and Total Synthesis of Lysobactin (Katanosin B) by von Nussbaum, Franz, Anlauf, Sonja, Benet-Buchholz, Jordi, Häbich, Dieter, Köbberling, Johannes, Musza, László, Telser, Joachim, Rübsamen-Waigmann, Helga, Brunner, Nina A.

“…Tackle‐resistant bacteria: Determination of the 3D structure of the antibiotic lysobactin has led to its total synthesis and resulted in a high‐yielding…”
Get full text

A Stereoselective Synthesis of Nonracemic (+)-Desoxoprosophylline by a Tandem Wittig [2+3]-Cycloaddition Reaction by Herdeis, Claus, Telser, Joachim

“…L‐Ascorbic acid serves as chiral starting material for the synthesis of (+)‐desoxoprosophylline. The synthetic pathway includes the formation of an O‐protected…”
Get full text

Identification of novel GLUT inhibitors by Siebeneicher, Holger, Bauser, Marcus, Buchmann, Bernd, Heisler, Iring, Müller, Thomas, Neuhaus, Roland, Rehwinkel, Hartmut, Telser, Joachim, Zorn, Ludwig

“…[Display omitted] The compound class of 1H-pyrazolo[3,4-d]pyrimidines was identified using HTS as very potent inhibitors of facilitated glucose transporter 1…”
Get full text

Effects of allylic and homoallylic substituents on the ring closing metathesis reaction used to synthesise simplified eleuthesides by Caggiano, Lorenzo, Castoldi, Damiano, Beumer, Raphael, Bayón, Pau, Telser, Joachim, Gennari, Cesare

“…During the course of our synthetic studies towards simplified eleuthesides, we have found that p-methoxyphenyl (PMP) protected allylic alcohols are compatible…”
Get full text

Dibenzodioxocinones—A new class of CETP inhibitors by Brückner, David, Hafner, Frank-Thorsten, Li, Volkhart, Schmeck, Carsten, Telser, Joachim, Vakalopoulos, Alexandros, Wirtz, Gabriele

“…Dibenzodioxocinones with high inhibitory potential for CETP and good plasma stability were prepared by semisynthesis from a natural product precursor…”
Get full text

Synthesis of novel simplified sarcodictyin/eleutherobin analogs with potent microtubule-stabilizing activity, using ring closing metathesis as the key-step by Beumer, Raphael, Bayón, Pau, Bugada, Piergiuliano, Ducki, Sylvie, Mongelli, Nicola, Sirtori, Federico Riccardi, Telser, Joachim, Gennari, Cesare

“…The synthesis of a number of novel simplified eleutheside analogs with potent tubulin-assembling and microtubule-stabilizing properties is described, using…”
Get full text

A carbonylative cross-coupling strategy to the total synthesis of the sarcodictyins: preliminary studies and synthesis of a cyclization precursor by Ceccarelli, Simona M, Piarulli, Umberto, Telser, Joachim, Gennari, Cesare

“…Preliminary studies were conducted on the implementation of a new strategy to the total synthesis of the common diterpenoid tricyclic skeleton of sarcodictyins…”
Get full text

Synthesis of novel simplified eleutheside analogues with potent microtubule-stabilizing activity, using ring-closing metathesis as the key-step by Beumer, Raphael, Bayón, Pau, Bugada, Piergiuliano, Ducki, Sylvie, Mongelli, Nicola, Sirtori, Federico Riccardi, Telser, Joachim, Gennari, Cesare

“…The synthesis of a number of novel simplified eleutheside analogues with potent tubulin-assembling and microtubule-stabilizing properties is described, using…”
Get full text

Synthesis of a simplified sarcodictyin analogue which retains microtubule stabilising properties by Telser, Joachim, Beumer, Raphael, Bell, Andrew A, Ceccarelli, Simona M, Monti, Diego, Gennari, Cesare

“…A strategy featuring ring-closing metathesis as key reaction is applied to the synthesis of the sarcodictyin analogue 15 . The precursor diene is accessed via…”
Get full text

Studies on the synthesis of chiral nonracemic 3,4-disubstituted azepanes, a formal synthesis of (+)- and (−)-balanol by Herdeis, Claus, Mohareb, Rafat M, Neder, Reinhard B, Schwabenländer, Franz, Telser, Joachim

“…Sugar lactones were converted to 3,4-disubstituted azepanes and caprolactam derivatives by selective deoxygenation, functionalization and reductive…”
Get full text

Structure and Total Synthesis of Lysobactin (Katanosin B) by von Nussbaum, Franz, Anlauf, Sonja, Benet-Buchholz, Jordi, Häbich, Dieter, Köbberling, Johannes, Musza, László, Telser, Joachim, Rübsamen-Waigmann, Helga, Brunner, Nina A.

“…Gegen resistente Bakterien: Die Bestimmung der Kristallstruktur ermöglichte die Totalsynthese des Antibiotikums Lysobactin. Der minimale Einsatz von…”
Get full text

Structure and Total Synthesis of Lysobactin (Katanosin B) by von Nussbaum, Franz, Anlauf, Sonja, Benet‐Buchholz, Jordi, Häbich, Dieter, Köbberling, Johannes, Musza, László, Telser, Joachim, Rübsamen‐Waigmann, Helga, Brunner, Nina A.

Get full text