Search Results - "Tastenoy, M"

Molecular cloning and functional characterization of a human VIP receptor from SUP-T1 lymphoblasts by Svoboda, M, Tastenoy, M, Van Rampelbergh, J, Goossens, J F, De Neef, P, Waelbroeck, M, Robberecht, P

“…We have cloned and sequenced a cDNA isolated from a human SUP-T1 lymphoblast cell line library. It encoded a 457 amino acids protein having 87% identity with…”
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Relative quantitative analysis of glucagon receptor mRNA in rat tissues by Svoboda, M, Tastenoy, M, Vertongen, P, Robberecht, P

“…Total RNA prepared from nine rat tissues were analyzed for their content in glucagon receptor mRNA by two independent hybridization approaches: (1) simple dot…”
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Binding of selective antagonists to four muscarinic receptors (M1 to M4) in rat forebrain by Waelbroeck, M, Tastenoy, M, Camus, J, Christophe, J

“…To compare the proportions of four muscarinic receptors in different rat brain regions, we used competition curves with four selective antagonists, at…”
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Cloning of a splice variant of the pituitary adenylate cyclase-activating polypeptide (PACAP) type I receptor by Svoboda, M, Tastenoy, M, Ciccarelli, E, Stiévenart, M, Christophe, J

“…The rat pancreatic acinar cell line AR 4-2J is endowed with numerous PACAP type I receptors (PACAPR1). The cDNA of this receptor was PCR amplified at low…”
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Mutational Analysis of the Glucose Regulatory Element in the Promoter of the Glucagon Receptor Gene by PORTOIS, LAURENCE, TASTENOY, MICHÈLE, SVOBODA, MICHAL

“…: Recently, we identified a glucose regulatory element in the promoter of the rat glucagon receptor gene. The effect of glucose is centered on a highly…”
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Stereoselective recognition of the enantiomers of phenglutarimide and of six related compounds by four muscarinic receptor subtypes by Waelbroeck, M., Lazareno, S., Pfaff, O., Friebe, T., Tastenoy, M., Mutschler, E., Lambrecht, G.

“…1 We have compared the binding properties of the enantiomers of phenglutarimide (1) and of six related compounds to M1 receptors in NB‐OK‐1 cells, M2 receptors…”
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Functional analysis of the glucose response element of the rat glucagon receptor gene in insulin-producing INS-1 cells by Portois, L., Tastenoy, M., Viollet, B., Svoboda, M.

“…Glucose stimulates the transcription of the glucagon receptor gene in hepatocytes and in pancreatic β cells. We recently identified a glucose response element…”
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Binding properties of nine 4‐diphenyl‐acetoxy‐N‐methyl‐piperidine (4‐DAMP) analogues to M1, M2, M3 and putative M4 muscarinic receptor subtypes by Waelbroeck, M., Camus, J., Tastenoy, M., Christophe, J.

“…1 We compared the binding properties of 4‐diphenyl‐acetoxy‐N‐methyl‐piperidine methiodide (4‐DAMP) and nine analogues of this compound on muscarinic receptors…”
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A cDNA construct allowing the expression of rat hepatic glucagon receptors by Svoboda, M, Ciccarelli, E, Tastenoy, M, Robberecht, P, Christophe, J

“…We constructed a full open reading frame (ORF) for the rat hepatic glucagon receptor using two non functional pCDM8 clones of a putative glucagon receptor…”
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Small introns in a hepatic cDNA encoding a new glucagon-like peptide 1-type receptor by Svoboda, M, Ciccarelli, E, Tastenoy, M, Cauvin, A, Stiévenart, M, Christophe, J

“…A cDNA fragment was PCR amplified at low-stringency from rat DNA, using two degenerated primers corresponding to consensus sequences in the second and third…”
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Binding kinetics of quinuclidinyl benzilate and methyl-quinuclidinyl benzilate enantiomers at neuronal (M1), cardiac (M2), and pancreatic (M3) muscarinic receptors by Waelbroeck, M, Tastenoy, M, Camus, J, Christophe, J

“…We analyzed the competition kinetics of quinuclidinyl benzilate (QNB) and QNB methiodide enantiomers on human NB-OK1 neuroblastoma (M1), rat cardiac (M2), and…”
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Thermodynamics of antagonist binding to rat muscarinic M2 receptors: antimuscarinics of the pridinol, sila‐pridinol, diphenidol and sila‐diphenidol type by Waelbroeck, M., Camus, J., Tastenoy, M., Lambrecht, G., Mutschler, E., Kropfgans, M., Sperlich, J., Wiesenberger, F., Tacke, R., Christophe, J.

“…1 We studied the effect of temperature on the binding to rat heart M2 muscarinic receptors of antagonists related to the carbon/silicon pairs…”
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Binding and functional properties of antimuscarinics of the hexocyclium/sila‐hexocyclium and hexahydro‐diphenidol/hexahydro‐sila‐diphenidol type to muscarinic receptor subtypes by Waelbroeck, M., Tastenoy, M., Camus, J., Christophe, J., Strohmann, C., Linoh, H., Zilch, H., Tacke, R., Mutschier, E., Lambrecht, G.

“…1 In an attempt to assess the structural requirements for the muscarinic receptor selectivity of hexahydro‐diphenidol (hexahydro‐difenidol) and…”
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Binding and functional properties of hexocyclium and sila‐hexocyclium derivatives to muscarinic receptor subtypes by Waelbroeck, M., Camus, J., Tastenoy, M., Feifel, R., Mutschler, E., Tacke, R., Strohmann, C., Rafeiner, K., Miranda, J.F. Rodrigues, Lambrecht, G.

“…1 We have compared the binding properties of several hexocyclium and sila‐hexocyclium derivatives to muscarinic M1 receptors (in rat brain, human neuroblastoma…”
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VIP and related peptides induce rapid homologous desensitization in the human lymphoma SUP T1 cell line by Robberecht, P, De Neef, P, Waelbroeck, M, Tastenoy, M, Christophe, J

“…Incubation of human SUP T1 lymphoblasts with VIP, helodermin and related peptides induced homologous desensitization within 5 min as indicated by: 1) a…”
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Stereoselectivity of (R)- and (S)-hexahydro-difenidol binding to neuroblastoma M1, cardiac M2, pancreatic M3, and striatum M4 muscarinic receptors by Waelbroeck, M, Camus, J, Tastenoy, M, Mutschler, E, Strohmann, C, Tacke, R, Lambrecht, G, Christophe, J

“…(R)-Hexahydro-difenidol has a higher affinity for M1 receptors in NB-OK 1 cells, pancreas M3 and striatum M4 receptors (pKi 7.9 to 8.3) than for cardiac M2…”
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Identification of a Glucose Response Element in the Promoter of the Rat Glucagon Receptor Gene by Portois, L, Maget, B, Tastenoy, M, Perret, J, Svoboda, M

“…We cloned the 5′ upstream region of the rat glucagon receptor gene, demonstrating that the 5′ noncoding domain of the glucagon receptor mRNA contained two…”
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Sequencing of eleven introns in genomic DNA encoding rat glucagon receptor and multiple alternative splicing of its mRNA by Maget, Barbara, Tastenoy, Michèle, Svoboda, Michal

“…We used the PCR (polymerase chain reaction) to amplify fragments of glucagon receptor DNA from genomic DNA. Sequencing of the subcloned fragments demonstrated…”
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Molecular cloning and in vitro properties of the recombinant rabbit secretin receptor by Svoboda, Michal, Tastenoy, Michele, De Neef, Philippe, Delporte, Christine, Waelbroeck, Magali, Robberecht, Patrick

“…The rabbit secretin receptor cDNA was cloned from rabbit pancreas using combined polymerase chain reaction (PCR)/rapid amplification of cDNA ends (PCR/RACE)…”
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Pharmacology of hexahydro-difenidol, hexahydro-sila-difenidol and related selective muscarinic antagonists by Lambrecht, G, Feifel, R, Moser, U, Wagner-Röder, M, Choo, L K, Camus, J, Tastenoy, M, Waelbroeck, M, Strohmann, C, Tacke, R

“…A series of hexahydro-difenidol (HHD) and hexahydro-sila-difenidol (HHSiD) analogues modified in the amino group, the phenyl ring and in the alkylene chain…”
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