Search Results - "TSUBAKI, Atsushi"

A practical synthesis of the [(2R)-3-(morpholinocarbonyl)-2-(1-naphthylmethyl)propionyl]-L-histidine moiety (P4-P2) in renin inhibitors by Harada, Hiromu, Yamaguchi, Toshiaki, Iyobe, Akira, Tsubaki, Atsushi, Kamijo, Tetsuhide, Iizuka, Kinji, Ogura, Katsuyuki, Kiso, Yoshiaki

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Epoxidation of cholesterol by hepatic microsomal lipid hydroperoxides by Watabe, T, Isobe, M, Tsubaki, A

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A SIMPLE DIASTEREOSELECTIVE SYNTHESIS OF CYCLOHEXYLNORSTATINE AND ALLOCYCLOHEXYLNORSTATINE by HARADA, Hiromu, TSUBAKI, Atsushi, KAMIJO, Tetsuhide, IIZUKA, Kinji, KISO, Yoshiaki

“…Cyclohexylnorstatine [(2R, 3S)-3-amino-4-cyclohexyl-2-hydroxybutyric acid] (1) and allocyclohexylnorstatine [(2S, 3S)-3-amino-4-cyclohexyl-2-hydroxybutyric…”
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Behavioral studies of KSG-504, a new CCK-A receptor antagonist by Yamazaki, Y, Takeda, H, Akahane, M, Tsubaki, A, Ajisawa, Y

“…The effects of KSG-504 after intravenous administration on behavior and other central functions were studied. KSG-504 did not affect the general behavior of…”
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Synthesis and Structure-Activity Relationships of Human Renin Inhibitors Designed from Angiotensinogen Transition State by IIZUKA, Kinji, KAMIJO, Tetsuhide, HARADA, Hiromu, AKAHANE, Kenji, KUBOTA, Tetsuhiro, ETOH, Yasuo, SHIMAOKA, Iwao, TSUBAKI, Atsushi, MURAKAMI, Makoto, YAMAGUCHI, Toshiaki, IYOBE, Akira, UMEYAMA, Hideaki, KISO, Yoshiaki

“…The synthesis and the structure-activity relationships of renin inhibitors designed from the angiotensinogen transition state are described. These inhibitors…”
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Synthesis of Human Renin Inhibitory Peptides, Angiotensinogen Transition-State Analogs Containing a Retro-Inverso Amide Bond by HARADA, Hiromu, IIZUKA, Kinji, KAMIJO, Tetsuhide, AKAHANE, Kenji, YAMAMOTO, Ryoji, NAKANO, Yasushi, TSUBAKI, Atsushi, KUBOTA, Tetsuhiro, SHIMAOKA, Iwao, UMEYAMA, Hideaki, KISO, Yoshiaki

“…The experimental details for the synthesis of human renin inhibitors are described. In order to aviod metabolic degradation of the Phe-His (P3-P2) amide bond…”
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コレシストキニンA受容体拮抗剤の合成研究(第2報)含硫アミドカルボン酸誘導体の合成とコレシストキニンA受容体阻害作用 by 味澤, 幸義, 北澤, 牧雄, 中野, 泰志, 椿, 敦, 阪, 正昭, 佐藤, 和明, 岡崎, 浩輔, 小林, 通洋

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コレシストキニンA受容体拮抗剤の合成研究(第3報)ナフチルスルホン誘導体の合成とコレシストキニンA受容体阻害作用 by 味澤, 幸義, 北澤, 牧雄, 中野, 泰志, 椿, 敦, 阪, 正昭, 佐藤, 和明, 岡崎, 浩輔, 内田, 雅彦, 小林, 通洋

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Studies on the Synthesis of Cholecystokinin A Receptor Antagonists. III. Synthesis and Cholecystokinin A Receptor Inhibitory Activities of Naphthyl Sulfone Derivatives by AJISAWA, Yukiyoshi, KITAZAWA, Makio, NAKANO, Yasushi, TSUBAKI, Atsushi, BAN, Masaaki, SATO, Kazuaki, OKAZAKI, Kosuke, UCHIDA, Masahiko, KOBAYASHI, Michihiro

“…A number of naphthyl sulfone derivatives were synthesized and tested for cholecystokinin A (CCK-A) receptor inhibitory activity in order to study…”
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Studies on the Synthesis of Cholecystokinin A Receptor Antagonists. II. Synthesis and Cholecystokinin A Receptor Inhibitory Activities of Sulfur-Containing Amide-Carboxylic Acid Derivatives by AJISAWA, Yukiyoshi, KITAZAWA, Makio, NAKANO, Yasushi, TSUBAKI, Atsushi, BAN, Masaaki, SATO, Kazuaki, OKAZAKI, Kosuke, KOBAYASHI, Michihiro

“…A number of sulfur-containing amide-carboxylic acid derivatives were synthesized and tested for cholecystokinin A (CCK-A) receptor inhibitory activity in order…”
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