Search Results - "T. Iminov, Rustam"

C−C Coupling through Nitrogen Deletion: Application to Library Synthesis by Holovach, Serhii, Melnykov, Kostiantyn P., Poroshyn, Illia, Iminov, Rustam T., Dudenko, Dmytro, Kondratov, Ivan, Levin, Mark, Grygorenko, Oleksandr O.

“…A protocol for parallel C(sp3)−C(sp3) coupling of (hetero)aromatic aldehydes and (hetero)arylmethyl amines based on a reductive amination – “nitrogen deletion”…”
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C−C Coupling through Nitrogen Deletion: Application to Library Synthesis by Holovach, Serhii, Melnykov, Kostiantyn P., Poroshyn, Illia, Iminov, Rustam T., Dudenko, Dmytro, Kondratov, Ivan, Levin, Mark, Grygorenko, Oleksandr O.

“…Invited for the cover of this issue are Oleksandr Grygorenko and his Ukrainian colleagues at Enamine Ltd., Taras Shevchenko National University of Kyiv,…”
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Building the Housane: Diastereoselective Synthesis and Characterization of Bicyclo[2.1.0]pentane Carboxylic Acids by Semeno, Volodymyr V, Vasylchenko, Vadym O, Vashchenko, Bohdan V, Lutsenko, Dmytro O, Iminov, Rustam T, Volovenko, Olesia B, Grygorenko, Oleksandr O

“…An approach to 1,3-disubstitued bicyclo[2.1.0]­pentane (housane) derivatives was developed. The method relied on lithium bis­(trimethylsilyl)­amide-mediated…”
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Simple and Convenient Synthesis of 2,3,4,5-Tetrahydro-1,5-dioxopyrrolo[1,2-a]quinazoline- 3a(1H)-carboxylic Acids in Multi-Gram Scale by V. Tverdokhlebov, Anton, T. Iminov, Rustam, A. Tolmachev, Andrey, M. Volovenko, Yulian, N. Kostyuk, Alexander, N. Chernega, Alexander, B. Rusanov, Eduard

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Preparation of 5-Amino-1,2-dihydro-4-(1-methyl-4-piperidinyl)pyrrol-3-ones by V. Tverdokhlebov, Anton, A. Chalyk, Bohdan, T. Iminov, Rustam, A. Tolmachev, Andrey

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Multigram Synthesis of Fluoroalkyl-Substituted Pyrazole-4-carboxylic Acids by Iminov, Rustam T., Mashkov, Alexander V., Vyzir, Ivan I., Chalyk, Bohdan A., Tverdokhlebov, Anton V., Mykhailiuk, Pavel K., Babichenko, Ludmila N., Tolmachev, Andrey A., Volovenko, Yulian M., Biitseva, Angelina, Shishkin, Oleg V., Shishkina, Svetlana V.

“…Acylation of tert‐butyl 3‐(methylamino)but‐2‐enoate with fluorinated acetic acid anhydrides occurred at the enamine carbon atom. The reaction of the resulting…”
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Synthesis of fluorinated oxazoles by oxidative cyclization of fluorinated enamides by Shishlyk, Oleg S., Shcherbatiuk, Andrey V., Iminov, Rustam T., Tverdokhlebov, Anton V., Tolmachev, Andrey A., Mykhailiuk, Pavel K., Biitseva, Angelina V.

“…[Display omitted] •Fluorinated isoxazoles were obtained by oxidation of the corresponding enamides.•These fluorinated building blocks are useful for Drug…”
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A Convenient Route to 1-Alkyl-5-trifluoromethyl-1,2,3-triazole-4-carboxylic Acids Employing a Diazo Transfer Reaction by Iminov, Rustam T., Mashkov, Alexander V., Chalyk, Bohdan A., Mykhailiuk, Pavel K., Tverdokhlebov, Anton V., Tolmachev, Andrey A., Volovenko, Yulian M., Shishkin, Oleg V., Shishkina, Svetlana V.

“…The reaction of ethyl 3‐(alkylamino)‐4,4,4‐trifluoro‐but‐2‐enoates with mesyl azide in the presence of 1,8‐diazabicyclo[5.4.0]undec‐7‐ene (DBU) gave ethyl…”
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Synthesis of condensed tetrahydroimidazo[1,2-a]quinazoline-1,5-dione derivatives by Iminov, Rustam T., Tverdokhlebov, Anton V., Tolmachev, Andrey A., Volovenko, Yulian M., Shishkina, Svetlana V., Shishkin, Oleg. V.

“…Heating of N-{2-[(R-amino)carbonyl]phenyl}prolinamides in triethyl orthoformate solution was found to give…”
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Synthesis of structurally constrained 4-quinazolinone derivatives with a tetrahedral C-2 atom present in three rings by Iminov, Rustam T., Tverdokhlebov, Anton V., Tolmachev, Andrey A., Volovenko, Yulian M., Shishkina, Svetlana V., Shishkin, Oleg V.

“…The reaction of 2-aminobenzamides with 2-oxocyclopentane-, 2-oxocyclohexane-, and 2-oxocycloheptaneacetic acids esters was found to give…”
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Front Cover: C−C Coupling through Nitrogen Deletion: Application to Library Synthesis (Chem. Eur. J. 4/2023) by Holovach, Serhii, Melnykov, Kostiantyn P., Poroshyn, Illia, Iminov, Rustam T., Dudenko, Dmytro, Kondratov, Ivan, Levin, Mark, Grygorenko, Oleksandr O.

“…Good chemistry, like great music, sometimes needs a good collaboration. The Cover Picture shows a combination of nitrogen‐deleting anomeric amide power…”
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