Search Results - "Sulur, G."

Polymorphs and Cocrystals of Nalidixic Acid by Gangavaram, Swarupa, Raghavender, S, Sanphui, Palash, Pal, Sharmistha, Manjunatha, Sulur G, Nambiar, Sudhir, Nangia, Ashwini

“…Only one X-ray crystal structure of the parent quinolone antibiotic nalidixic acid is known in the published and patent literature. A systematic search for new…”
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Thermal studies of furosemide–caffeine binary system that forms a cocrystal by Pal, Sharmistha, Roopa, B. N., Abu, Khalid, Manjunath, Sulur G., Nambiar, Sudhir

“…Thermal techniques, differential scanning calorimetry (DSC), and hot stage microscopy (HSM) have been used to study the interactions between furosemide and…”
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Novel furosemide cocrystals and selection of high solubility drug forms by Goud, N Rajesh, Gangavaram, Swarupa, Suresh, Kuthuru, Pal, Sharmistha, Manjunatha, Sulur G, Nambiar, Sudhir, Nangia, Ashwini

“…Furosemide was screened in cocrystallization experiments with pharmaceutically acceptable coformer molecules to discover cocrystals of improved physicochemical…”
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LATITUDE study: PSA response characteristics and correlation with overall survival (OS) and radiological progression-free survival (rPFS) in patients with metastatic hormone-sensitive prostate cancer (mHSPC) receiving ADT+abiraterone acetate and prednisone (AAP) or placebo (PBO) by Matsubara, N., Chi, K.N., Ozguroglu, M., Rodriguez Antolin, A., Feyerabend, S., Fein, L., Alekseev, B.Y., Sulur, G., Protheroe, A., Li, S., Mundle, S.D., De Porre, P., Tran, N., Fazazi, K.

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Semmler–Wolff aromatisation: a concise route for the synthesis of 5-amino-quinazolines and 4-amino-indoles by Manjunatha, Sulur G., Bachu, Sreekanth, Gautam, Vibha, Kumari, Mohana, Nambiar, Sudhir, Ramasubramanian, Sridharan, Puranik, Ramachandra

“…[Display omitted] A simple and efficient methodology for the synthesis of 5-amino-quinazolines and 4-amino-indoles via Semmler–Wolff aromatisation reaction has…”
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A novel synthetic approach to 4-acetamido-1-arylindazoles via Semmler–Wolff rearrangement of 1-aryl-6,7-dihydro-5H-indazol-4-one oxime by Manjunatha, Sulur G., Bachu, Sreekanth, Kadambar, Vasantha Krishna, Murugan, Andiappan, Ramasubramanian, Sridharan, Ramachandra, Puranik, Nambiar, Sudhir

“…A simple and efficient procedure for the syntheses of 4-acetamido-1-arylindazoles from corresponding 1-aryl-6,7-dihydro-5H-indazol-4-one oximes by…”
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Facile synthesis of 3-aryl/alkylamino 5-aryl/alkyl 1,2,4-oxadiazoles from acylthiourea by Chennakrishnareddy, Gundala, Debasis, Hazra, Jayan, Rapai, Manjunatha, Sulur G.

“…Facile and selective synthesis of 3-aryl/alkylamino 5-aryl/alkyl 1,2,4-oxadiazoles starting from N-acylthioureas has been demonstrated. The regio-selectivity…”
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Palladium on carbon–bromobenzene mediated esterification and transesterification by Aavula, Sanjeev Kumar, Chikkulapalli, Anil, Hanumanthappa, N., Jyothi, Indira, Vinod Kumar, C.H., Manjunatha, Sulur G.

“…A series of carboxylic acids were converted into their corresponding esters using the Pd/C catalyzed hydrogenation conditions in the presence of catalytic…”
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A mechanistic investigation of Biginelli reaction under base catalysis by Kamal Raj, M., Rao, H. Surya Prakash, Manjunatha, Sulur G, Sridharan, R., Nambiar, Sudhir, Keshwan, Jaikumar, Rappai, Jayan, Bhagat, Sagar, Shwetha, B.S., Hegde, Dinesh, Santhosh, U.

“…The mechanism of the three component base mediated Biginelli dihydropyrimidines synthesis was investigated using Accurate Mass TOF LC–MS-ESI and Tandem TOF…”
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Novel approach towards one pot stereospecific synthesis of carbohydrate derived substituted imidazolines by Gautam, Vibha, Kagita, Veera Babu, Nambiar, Sudhir, Phaneendra, Gutala, Manjunatha, Sulur G., Ramasubramanian, Sridharan, Suresh Babu, M., Keshwan, Jaikumar, Bhagat, Sagar, Prakash, Ravindran, Puranik, Ramachandra

“…A simple synthetic approach has been developed towards one pot synthesis of 2-imidazolines under mild acidic conditions from N-acetyl glucosamine via reductive…”
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Exploiting the Differential Reactivities of Halogen Atoms: Development of a Scalable Route to IKK2 Inhibitor AZD3264 by Murugan, Andiappan, Bachu, Sreekanth, Manjunatha, Sulur G, Ramakrishnan, Ravi, Kadambar, Vasantha Krishna, Reddy, Chandrasekhara, Torlikonda, Venkata Rao, George, Sajan, Ramasubramanian, Sridharan, Nambiar, Sudhir

“…An efficient and scalable synthesis of AZD3264 is described in which the differential reactivities of various halogen atoms have been employed. The process…”
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Regio-selective synthesis of 1,2-aminoalcohols from epoxides and chlorohydrins by Murugan, Andiappan, Kadambar, Vasantha Krishna, Bachu, Sreekanth, Rajashekher Reddy, M., Torlikonda, Venkatarao, Manjunatha, Sulur G., Ramasubramanian, Sridharan, Nambiar, Sudhir, Howell, Gareth P., Withnall, Jane

“…A simple and efficient procedure for the regio-selective synthesis of 1,2-aminoalcohols from terminal epoxides and chlorohydrins by using NaHMDS as the source…”
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Convenient N-acetylation of amines in N,N-dimethylacetamide with N,N-carbonyldiimidazole by Chikkulapalli, Anil, Aavula, Sanjeev Kumar, Mona NP, Rifahath, C., Karthikeyan, C.H., Vinodh Kumar, Sulur G., Manjunatha, Sumathi, Shanmugam

“…[Display omitted] Dimethylacetamide (DMAc) acts as an efficient source of acetyl and dimethylamine gas in the presence of N,N-carbonyldiimidazole (CDI)…”
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A Greener Approach for the Large-Scale Synthesis of 1,4,5-Trisubstituted Pyrazole, AZD8329 by Rangappa, Paramashivappa, Ghosh, Avipsa, Chitrapadi, Smitha, Kantikar, Gajanan, CH, Vinod Kumar, Sythana, Sureshkumar, Manjunath, Sulur G, Nambiar, Sudhir, R, Sridhran

“…The development of a convenient, safe and scalable process for AZD8329 manufacturing is reported here. Synthesis was achieved in a two-step telescopic process…”
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Development of a Safe, Scalable Process for the Preparation of an Oxaisoxazolidinone by Santhosh, U, Kshirsagar, Yogesh M, Venkatesan, K, Hazra, Debasis, Kindel, Jnaneshwara, Sridharan, R, Ennis, David, Howells, Garnet E, Stefinovic, Marijan, Manjunatha, Sulur G, Nambiar, Sudhir

“…This report describes the development and scale up of the synthesis of oxaisoxazolidinone 1, a significant synthon in the synthesis of the MRSA development…”
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Development of an Efficient, Scalable Route for the Preparation of a Novel Insulin-Like Growth Factor‑1 Receptor Modulator by Kumar, CH Vinod, Kavitake, Santosh, Kumar, Sythana Suresh, Cornwall, Philip, Ashok, Mithun, Bhagat, Sagar, Manjunatha, Sulur G, Nambiar, Sudhir

“…A chromatography-free and efficient synthesis of insulin-like growth factor-1 receptor (IGF-1R) modulator is reported. Herein we describe an improved synthesis…”
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Understanding of the mass spectrometric fragmentation pathways of a few potentially genotoxic haloaniline isomers in their protonated form by collision-induced dissociation by Patrick, Rex, Nagarajan, N.S., Pan, Hefeng, Saha, Subhra Kanti, Rapai, Jayan, Torlikonda, Venkatarao, Panda, Manoranjan, Manjunatha, Sulur G., Nambiar, Sudhir

“…Collision-induced dissociation (CID) mass spectra of a few haloaniline isomers, (chloroanilines, dichloroanilines, difluoroanilines, chloro-fluoroanilines and…”
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A simple way of recycling of homogeneous catalyst in Suzuki reaction by Manjunatha, Sulur G., Rangappa, Paramashivappa, Sythana, Sureshkumar, Babu, Sureshbabu M., Tadiparthi, Krishnaji, Gundala, Chennakrishnareddy

“…A simple and practical method of recycling homogeneous catalysts in the Suzuki reaction using appropriate work up conditions is reported here. The commonly…”
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TCL1 Oncogene Expression in AIDS-Related Lymphomas and Lymphoid Tissues by Teitell, Michael, Damore, Michael A., Sulur, Girija G., Turner, Devin E., Stern, Marc-Henri, Said, Jonathan W., Denny, Christopher T., Wall, Randolph

“…AIDS-related non-Hodgkin's lymphoma (AIDS NHL) comprises a diverse and heterogeneous group of high-grade B cell tumors. Certain classes of AIDS NHL are…”
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TCL1 oncogene expression in B cell subsets from lymphoid hyperplasia and distinct classes of B cell lymphoma by SAID, Jonathan W, HOYER, Katrina K, RAWLINGS, David J, WALL, Randolph, TEITELL, Michael A, FRENCH, Samuel W, ROSENFELT, Lisa, GARCIA-LLORET, Maria, KOH, Patricia J, CHENG, Tse-Chang, SULUR, Girija G, PINKUS, Geraldine S, KUEHL, W. Michael

“…Activation of the TCL1 oncogene has been implicated in T cell leukemias/lymphomas and recently was associated with AIDS diffuse large B cell lymphomas…”
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