Search Results - "Stoltefuss, J."

Inhibition of human hepatitis B virus (HBV) by a novel non-nucleosidic compound in a transgenic mouse model by Weber, O., Schlemmer, K.-H., Hartmann, E., Hagelschuer, Ina, Paessens, A., Graef, E., Deres, K., Goldmann, S., Niewoehner, U., Stoltefuss, J., Haebich, D., Ruebsamen-Waigmann, H., Wohlfeil, Stefan

“…BAY 41-4109 is a member of a class of heteroaryl-pyrimidines that was recently identified as potent inhibitors of human hepatitis B virus (HBV) replication. We…”
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Stereoselective Mukaiyama-Michael/Michael/Aldol Domino Cyclization as the Key Step in the Synthesis of Pentasubstituted Arenes: An Efficient Access to Highly Active Inhibitors of Cholesteryl Ester Transfer Protein (CETP) by Paulsen, Holger, Antons, Stefan, Brandes, Arndt, Lögers, Michael, Müller, Stephan Nicholas, Naab, Paul, Schmeck, Carsten, Schneider, Stephan, Stoltefuß, Jürgen

“…Seemingly heartbreaking for a stereochemist, the one‐step selective construction of a stereopentad and its prompt destruction by aromatization has been proven…”
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A new type of Ca-channel modulation by a novel class of 1,4-dihydropyridines by Bechem, M., Goldmann, S., Gross, R., Hallermann, St, Hebisch, S., Hütter, J., Rounding, H.-P., Schramm, M., Stoltefuss, J., Straub, A.

“…Both Ca-antagonistic as well as Ca-agonistic 1,4-dihydropyridines (DHPs) have become extremely important tools to investigate the role of Ca-channels under…”
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Pharmacologic and radioligand binding studies of 1,4-dihydropyridines in rat cardiac and vascular preparations: stereoselectivity and voltage dependence of antagonist and activator interactions by Zheng, W, Stoltefuss, J, Goldmann, S, Triggle, D J

“…The pharmacologic and radioligand-binding properties of 1,4-dihydropyridines in an activator (Bay K 8644) and an antagonist (nifedipine) series were studied in…”
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Novel Antibiotics for the Treatment of Gram-Positive Bacterial Infections by Brands, Michael, Endermann, Rainer, Gahlmann, Reinhold, Krüger, Jochen, Raddatz, Siegfried, Stoltefuβ, Jürgen, Belov, Vladimir N, Nizamov, Shamil, Sokolov, Viktor V, de Meijere, Armin

“…The natural dipeptide antibiotic TAN 1057 A,B displays excellent antibacterial activity against staphylococci including methicillin resistant Staphylococcus…”
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Determination of the absolute configuration of the active amlodipine enantiomer as (-)-S: a correction by Goldmann, Siegfried, Stoltefuss, Juergen, Born, Liborius

“…The active (-) enantiomer of amlodipine was originally reported to have R configuration. This does not concur with other 1,4-dihydropyridines with known…”
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Fluorine-Substitution in Cholesteryl Ester Transfer Protein Inhibitors (CETPInhibitors) – Biology, Chemistry, SAR, and Properties by Holger Paulsena, Siegfried Zaiss, Delf Schmidt, Hilmar Bischoff, Klaus-Dieter Bremm, Paul Naab, Michael Lögers, Stephan N. Wirtz, Jürgen Stoltefuss, Gunter Schmidt, Arndt Brandes, Carsten Schmeck, Stefan Antons

“…The inhibition of the cholesteryl ester transfer protein (CETP) provides a method for the elevation of the high density lipoprotein cholesterol (HDL-C) level,…”
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Deterination of the absolute configuration of the active amlodipine enantiomer as (-)-S : a correction by GOLDMANN, S, STOLTEFUSS, J, BORN, L

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A new type of Ca-channel modulation by a novel class of 1,4-dihydropyridines by Bechem, M, Goldmann, S, Gross, R, Hallermann, S, Hebisch, S, Hütter, J, Rounding, H P, Schramm, M, Stoltefuss, J, Straub, A

“…Both Ca-antagonistic as well as Ca-agonistic 1,4-dihydropyridines (DHPs) have become extremely important tools to investigate the role of Ca-channels under…”
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