Search Results - "Stimac, Vlado"
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Synthesis and biological properties of 4″-O-acyl derivatives of 8a-Aza-8a-homoerythromycin
Published in Journal of antibiotics (01-03-2009)“…A series of 4″- O- acyl derivatives of 8a-aza-8a-homoerythromycins A were synthesized and tested against Gram-positive and Gram-negative bacteria. Derivatives…”
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2
Synthesis and Antibacterial Activity of Isomeric 15-Membered Azalides
Published in Journal of antibiotics (01-12-2006)“…A series of 3-keto and 3-O-acyl derivatives of both 6-O-alkyl-8a-aza-8a-homoerythromycin A and 6-O-alkyl-9a-aza-9a-homo-erythromycin A were synthesised and…”
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3
Synthesis of macrolones with central piperazine ring in the linker and its influence on antibacterial activity
Published in Bioorganic & medicinal chemistry (01-12-2011)“…Three macrolides, clarithromycin, azithromycin and 11-O-Me-azithromycin have been selected for the construction of a series of new macrolone derivatives…”
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4
Initial Scale-Up and Process Improvements for the Preparation of a Lead Antibacterial Macrolone Compound
Published in Organic process research & development (19-11-2010)“…Macrolones are a novel class of potent antimicrobial agents that consist of a macrolide scaffold to which a quinolone unit is tethered by various linkers to…”
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Synthesis and biological activity of 4″- O-acyl derivatives of 14- and 15-membered macrolides linked to ω-quinolone-carboxylic unit
Published in Bioorganic & medicinal chemistry (01-09-2010)“…The synthesis and antimicrobial activity of a new class of macrolide antibiotics which consist of a macrolide scaffold and a quinolone unit covalently…”
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6
Novel desosamine-modified 14- and 15-membered macrolides without antibacterial activity
Published in Bioorganic & medicinal chemistry letters (15-05-2012)“…Novel modifications of the desosamine sugar of 14- and 15-membered antibacterial macrolides, in which the desosamine was fused with…”
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Synthesis and properties of macrolones characterized by two ether bonds in the linker
Published in Bioorganic & medicinal chemistry (01-09-2010)“…In this paper synthesis of macrolones 1– 18 starting from azithromycin is reported. Two key steps in the construction of the linker between macrolide and…”
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Erratum: Synthesis and biological properties of 4″-O-acyl derivatives of 8a-Aza-8a-homoerythromycin
Published in Journal of antibiotics (28-06-2010)“…Correction to: The Journal of Antibiotics (2009) 62, 133–144; doi:10.1038/ja.2009.1 The authors of the above article noted an error in the publication of this…”
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Synthesis and biological properties of 4''-O-acyl derivatives of 8a-Aza-8a-homoerythromycin
Published in Journal of antibiotics (01-06-2010)Get full text
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10
3-O-Acilni derivati premoštenih 15-članih azalida: priprava, određivanje strukture i antibakterijska aktivnost
Published in Croatica Chemica Acta (15-06-2005)“…Opisani su priprava, odre|ivanje strukture i biološka ispitivanja 15-članih azalida aciliranih na položaju C-3. Kiselom hidrolizom pripadajućih 3-kladinozil…”
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