Search Results - "Sterk, Damjan"

Co-crystals, Salts or Mixtures of Both? The Case of Tenofovir Alafenamide Fumarates by Lengauer, Hannes, Makuc, Damjan, Šterk, Damjan, Perdih, Franc, Pichler, Arthur, Trdan Lušin, Tina, Plavec, Janez, Časar, Zdenko

“…Tenofovir alafenamide fumarate (TAF) is the newest prodrug of tenofovir that constitutes several drug products used for the treatment of HIV/AIDS. Although the…”
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Efficient and highly stereoselective assembly of rosuvastatin by Šterk, Damjan, Zaugg, Werner, Beutler, Ulrich, Loeser, Eric M., Prasad, Kapa, Časar, Zdenko

“…[Display omitted] We report an asymmetric synthesis of rosuvastatin starting from an α,β-unsaturated aldehyde precursor containing the rosuvastatin…”
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Study of the Reaction of Bulky Aryllithium Reagents with 3,4-Dimethyl-2,5-diphenyl-1,3,2-oxazaphospholidine-2-borane Derived from Ephedrine by Stephan, Michel (Massoud S.), Šterk, Damjan, Modec, Barbara, Mohar, Barbara

“…The ring opening of enantiomerically pure 3,4-dimethyl-2,5-diphenyl-1,3,2-oxazaphospholidine-2-borane (1) with a variety of bulky aryllithium reagents was…”
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Enantioselective and diastereoselective synthesis of fluorinated dipeptides by late electrophilic fluorination by Mohar, Barbara, Sterk, Damjan, Ferron, Laurent, Cahard, Dominique

“…Asymmetric synthesis of fluorinated dipeptides by electrophilic fluorination occurs with up to 73:27 enantiomeric ratio and high >98:2 diastereomeric ratio…”
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Application of Flow Photochemical Bromination in the Synthesis of a 5‑Bromomethylpyrimidine Precursor of Rosuvastatin: Improvement of Productivity and Product Purity by Šterk, Damjan, Jukič, Marko, Časar, Zdenko

“…In this report we present a flow photochemical bromination of a 5-methyl-substituted pyrimidine precursor of rosuvastatin. The study demonstrated that the…”
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Highly Enantioselective Transfer Hydrogenation of Fluoroalkyl Ketones by Šterk, Damjan, Stephan, Michel, Mohar, Barbara

“…The asymmetric transfer hydrogenation of fluoroalkyl ketones mediated by [Ru(η 6-arene)((S,S)-R2NSO2DPEN)] catalysts using HCO2H−Et3N afforded the…”
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DiPAMP's Big Brother "i-Pr-SMS-Phos" Exhibits Exceptional Features Enhancing Rhodium(I)-Catalyzed Hydrogenation of Olefins by Stephan, Michel, Šterk, Damjan, Mohar, Barbara

“…Switching Knowles DiPAMP’s {DiPAMP=1,2‐bis[(o‐anisyl)(phenyl)phosphino]‐ ethane} MeO groups with i‐PrO ones led to the i‐Pr‐SMS‐Phos…”
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Concise and highly efficient approach to three key pyrimidine precursors for rosuvastatin synthesis by STERK, Damjan, CASAR, Zdenko, JUKIC, Marko, KOSMRLJ, Janez

“…We report the synthesis of 5-formyl-, 5-(hydroxymethyl)-, and 5-(bromomethyl) substituted…”
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Profiling the tuneable R-SMS-Phos structure in the rhodium(I)-catalyzed hydrogenation of olefins: the last stand? by Stephan, Michel, Šterk, Damjan, Zupančič, Borut, Mohar, Barbara

“…A diversified family of enantiopure P-stereogenic "R-SMS-Phos" {R-SMS-Phos = 1,2-bis[(o-RO-phenyl)(phenyl)phosphino]ethane} ligands wherein R = branched or…”
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3-Mercaptopropionic acid as a new reagent for the industrially applicable synthesis of highly pure O-desmethylvenlafaxine from venlafaxine by Furlan, Borut, Časar, Zdenko, Šterk, Damjan, Fabris, Jan

“…3-Mercaptopropionic acid was introduced as a cheap new O-demethylating agent as exemplified by its application in the synthesis of antidepressant…”
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Corrigendum to “Enantioselective and diastereoselective synthesis of fluorinated dipeptides by late electrophilic fluorination”: [Tetrahedron Lett. 46 (2005) 5029] by Mohar, Barbara, Sterk, Damjan, Ferron, Laurent, Cahard, Dominique

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Transfer hydrogenation of activated ketones using novel chiral Ru(II)- N-arenesulfonyl-1,2-diphenylethylenediamine complexes by Šterk, Damjan, Stephan, Massoud S., Mohar, Barbara

“…Graphic A series of α-keto esters and α,α,α-trifluoromethyl ketones were reduced in high yields and excellent enantioselectivities under Ru-catalysed transfer…”
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New chiral N-( N, N-dialkylamino)sulfamoyl-1,2-diamine ligands for highly enantioselective transfer hydrogenation of ketones by Šterk, Damjan, Stephan, Massoud S., Mohar, Barbara

“…Chiral Ru(II) and Rh(III) complexes of N-( N, N-dialkylamino)sulfamoyl-1,2-diamine catalyze the transfer hydrogenation of various classes of aromatic ketones…”
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