Search Results - "Srinivas, Gujjary"
-
1
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists
Published in Bioorganic & medicinal chemistry letters (01-05-2012)“…The receptor model-supported design, synthesis and multi-parameter optimization of novel quinazoline derivatives as MCHR1 antagonists are described. The in…”
Get full text
Journal Article -
2
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: Part 2
Published in Bioorganic & medicinal chemistry letters (01-05-2012)“…The synthesis and design guided by SAR and SPR studies of novel quinazoline derivatives as MCHR1 antagonists are described. Compound 8 (DRL-21816) has emerged…”
Get full text
Journal Article -
3
Enantiospecific synthesis of (−)- d-noviose from (−)-pantolactone
Published in Tetrahedron letters (04-09-2006)“…Noviose, the rare sugar moiety present in novobiocin, is an important antimicrobial and antitumor agent that has been shown to inhibit DNA gyrase and HSP90. An…”
Get full text
Journal Article -
4
Synthesis of Novel Oxime Functionalized Aldol Products via Michael Addition of Oximes Onto Baylis–Hillman Adducts
Published in Synthetic communications (01-02-2006)Get full text
Journal Article