Search Results - "Srikanth, Danaboina"

Coumarin‐Thiourea Hybrids Show Potent Carbonic Anhydrase IX and XIII Inhibitory Action by Thacker, Pavitra S., Srikanth, Danaboina, Angeli, Andrea, Singh, Priti, Chinchilli, Krishna Kartheek, Arifuddin, Mohammed, Supuran, Claudiu T.

“…A series of coumarin‐thiourea hybrids (4 a–o) has been synthesized, and the compounds have been evaluated against the tumour associated transmembrane isoform,…”
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Synthesis and Biological Evaluation of Coumarin-Linked 4-Anilinomethyl-1,2,3-Triazoles as Potent Inhibitors of Carbonic Anhydrases IX and XIII Involved in Tumorigenesis by Thacker, Pavitra S, Tiwari, Prerna L, Angeli, Andrea, Srikanth, Danaboina, Swain, Baijayantimala, Arifuddin, Mohammed, Supuran, Claudiu T

“…A series of coumarin-linked 4-anilinomethyl-1,2,3-triazoles ( - ) was synthesized via a molecular hybridization approach, through carbon C-6 of the coumarin…”
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Exploration of 1,3,5-trisubstituted pyrazoline derivatives as human carbonic anhydrase inhibitors: Synthesis, biological evaluation and in silico studies by Srikanth, Danaboina, Shanthi, Kollu, Paoletti, Niccolò, Joshi, Swanand Vinayak, Shaik, Mahammad Ghouse, Rana, Preeti, Vadakattu, Manasa, Yaddanapudi, Venkata Madhavi, Supuran, Claudiu T., Nanduri, Srinivas

“…The human carbonic anhydrase (hCA) IX and XII isoforms are overexpressed in hypoxic conditions, contributing to cancer. Lack of isoform selectivity has been…”
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6-Aminocoumarin oxime-ether/sulfonamides as selective hCA IX and XII inhibitors: Synthesis, evaluation, and molecular dynamics studies by Ghouse, Shaik Mahammad, Sinha, Kareena, Bonardi, Alessandro, Pawar, Gaurav, Malasala, Satyaveni, Danaboina, Srikanth, Mohammed, Arifuddin, Yaddanapudi, Venkata M, Supuran, Claudiu T, Nanduri, Srinivas

“…Carbonic anhydrase isoforms IX and XII are overexpressed in hypoxic tumor cells regulating various physiological processes such as cell proliferation,…”
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A comprehensive review on potential therapeutic inhibitors of nosocomial Acinetobacter baumannii superbugs by Srikanth, Danaboina, Joshi, Swanand Vinayak, Ghouse Shaik, Mahammad, Pawar, Gaurav, Bujji, Sushmitha, Kanchupalli, Vinaykumar, Chopra, Sidharth, Nanduri, Srinivas

“…[Display omitted] •An overview of different mechanisms of resistance and virulence factors of A. baumannii is presented.•Diverse structural classes of A…”
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Design, synthesis, SAR, and biological evaluation of saccharin‐based hybrids as carbonic anhydrase inhibitors by Chinchilli, Krishna K., Royyala, Venkata N., Thacker, Pavitra S., Angeli, Andrea, Danaboina, Srikanth, Singh, Priti, Nanduri, Srinivas, Supuran, Claudiu T., Arifuddin, Mohammed

“…Saccharin is a cyclic secondary sulfonamide, which is a selective inhibitor of the tumor‐associated carbonic anhydrase (CA; EC 4.2.1.1) enzymes CA IX and CA…”
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