Search Results - "Sproull, Steven J"

3-Oxa-15-cyclohexyl prostaglandin DP receptor agonists as topical antiglaucoma agents by Hellberg, Mark R., Conrow, Raymond E., Sharif, Najam A., McLaughlin, Marsha A., Bishop, John E., Crider, Julie Y., Dean, W.Dennis, DeWolf, Kevin A., Pierce, David R., Sallee, Verney L., Selliah, Robert D., Severns, Bryon S., Sproull, Steven J., Williams, Gary W., Zinke, Paul W., Klimko, Peter G.

“…A series of prostaglandin DP agonists containing a 3-oxa-15-cyclohexyl motif was synthesized and evaluated in several in vitro and in vivo biological assays…”
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Enantioselective Synthesis of Brinzolamide (AL-4862), a New Topical Carbonic Anhydrase Inhibitor. The “DCAT Route” to Thiophenesulfonamides by Conrow, Raymond E, Dean, W. Dennis, Zinke, Paul W, Deason, Michael E, Sproull, Steven J, Dantanarayana, Anura P, DuPriest, Mark T

“…A large scale synthesis of the topical carbonic anhydrase inhibitors AL-4623A (13a·HCl) and AL-4862 (13b) from 3-acetyl-2,5-dichlorothiophene (“DCAT”, 1) is…”
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Enantioselective Synthesis of AL-4414A, a Topically Active Carbonic Anhydrase Inhibitor by DuPriest, Mark T, Zinke, Paul W, Conrow, Raymond E, Kuzmich, Daniel, Dantanarayana, Anura P, Sproull, Steven J

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