Search Results - "Spampinato, Ambra"

FABP4 inhibitors 3D-QSAR model and isosteric replacement of BMS309403 datasets by Floresta, Giuseppe, Cilibrizzi, Agostino, Abbate, Vincenzo, Spampinato, Ambra, Zagni, Chiara, Rescifina, Antonio

“…The data have been obtained from FABP4 inhibitor molecules previously published. The 120 compounds were used to build a 3D-QSAR model. The development of the…”
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3D-QSAR assisted identification of FABP4 inhibitors: An effective scaffold hopping analysis/QSAR evaluation by Floresta, Giuseppe, Cilibrizzi, Agostino, Abbate, Vincenzo, Spampinato, Ambra, Zagni, Chiara, Rescifina, Antonio

“…[Display omitted] •A 3D-QSAR model was produced for the FABP4 inhibitors.•A scaffold hopping suggested 3000 potentially active FABP4 inhibitors.•Three…”
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trans-Cyclooctene- and Bicyclononyne-Linked Nucleotides for Click Modification of DNA with Fluorogenic Tetrazines and Live Cell Metabolic Labeling and Imaging by Spampinato, Ambra, Kužmová, Erika, Pohl, Radek, Sýkorová, Veronika, Vrábel, Milan, Kraus, Tomáš, Hocek, Michal

“…A series of 2′-deoxyribonucleoside triphosphates (dNTPs) bearing 2- or 4-linked trans-cyclooctene (TCO) or bicyclononyne (BCN) tethered through a shorter…”
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ABNOH‐Linked Nucleotides and DNA for Bioconjugation and Cross‐linking with Tryptophan‐Containing Peptides and Proteins by Spampinato, Ambra, Leone, Denise‐Liu', Pohl, Radek, Tarábek, Ján, Šoltysová, Markéta, Polák, Marek, Kádek, Alan, Sýkorová, Veronika, Řezáčová, Pavlína, Hocek, Michal

“…Reactive N‐hydroxy‐9‐azabicyclo[3.3.1]nonane (ABNOH) linked 2′‐deoxyuridine 5′‐O‐mono‐ and triphosphates were synthesized through a CuAAC reaction of…”
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