Search Results - "Somnath Halder"

Mutual prodrugs containing bio-cleavable and drug releasable disulfide linkers by Jain, Arun K., Gund, Machhindra G., Desai, Dattatraya C., Borhade, Namdev, Senthilkumar, Subrayan P., Dhiman, Mini, Mangu, Naveen K., Mali, Sunil V., Dubash, Nauzer P., Halder, Somnath, Satyam, Apparao

“…[Display omitted] •We have reported novel mutual prodrugs containing drug-releasable disulfide linkers.•Drug release in simulated gastric fluid and human…”
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Synthesis of highly functionalized phenylalanine derivatives via cross-enyne metathesis reactions by Kotha, Sambasivarao, Halder, Somnath, Brahmachary, Enugurthi

“…A new method for the synthesis of constrained phenylalanine derivatives is described. In this regard, the simple synthesis of acyclic diene building blocks…”
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Benzannulation by Kotha, Sambasivarao, Misra, Shilpi, Halder, Somnath

“…Various synthetic methodologies developed in recent years for benzannulation have been reviewed. These methodologies include cycloaddition approaches,…”
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Synthesis of macrocyclic cyclophane-based unusual α-amino acid derivatives by Kotha, Sambasivarao, Halder, Somnath

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Accidental discovery of a ‘longer-range’ vinylogous Pummerer-type lactonization: formation of sulindac sulfide lactone from sulindac by Halder, Somnath, Satyam, Apparao

“…Unexpected formation of sulindac sulfide lactone ( 4) from sulindac ( 1) in presence of oxalyl chloride and Et 3N has occurred probably via a thionium…”
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The therapeutic potential of GPR120: a patent review by Halder, Somnath, Kumar, Sanjay, Sharma, Rajiv

“…Type 2 diabetes (T2D) is a complex metabolic disorder characterized by persistent hyperglycemia and a wide range of underlying metabolic defects. The…”
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NO-NSAIDs. Part 3：Nitric Oxide-Releasing Prodrugs of Non-steroidal Anti-inflammatory Drugs by Namdev Borhade, Asif Rahimkhan Pathan, Somnath Halder, Manoj Karwa, Mini Dhiman, Venu Pamidiboina, Machhindra Gund, Jagannath Janardhan Deshattiwar, Sunil Vasantrao Mali, Nitin Janardanrao Deshmukh, Subrayan Palanisamy Senthilkumar, Parikshit Gaikwad, Santhosh Goud Tipparam, Jayesh Mudgal, Milan Chandra Dutta, Aslam Usmangani Burhan, Gajanan Thakre, Ankur Sharma, Shubhada Deshpande, Dattatraya Chandrakant Desai, Nauzer Pervez Dubash, Arun Kumar Jain, Somesh Sharma, Kumar Venkata Subrahmanya Nemmani, Apparao Satyam

“…In continuation of our efforts to discover novel nitric oxide-releasing non-steroidal anti-inflammatory drugs (NO-NSAIDs) as potentially "Safe NSAIDs," we…”
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Synthesis of dibenzocyclobutenylglycine derivatives by Kotha, Sambasivarao, Halder, Somnath, Sreenivasachary, Nampally

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Intelligent phase detection of signals on varying SNR using machine learning algorithms by Halder, Somnath, Sonar, Souvik

“…The phase detection as a part of phased-locked loop (PLL) circuit is a critical component in any telecommunication systems. With the advancement of modern-era…”
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Synthesis and Antimicrobial Evaluation of Amphiphilic Neamine Derivatives by Baussanne, Isabelle, Bussière, Antoine, Halder, Somnath, Ganem-Elbaz, Carine, Ouberai, Myriam, Riou, Mickael, Paris, Jean-Marc, Ennifar, Eric, Mingeot-Leclercq, Marie-Paule, Décout, Jean-Luc

“…The aminoglycoside antibiotics bind to the 16S bacterial rRNA and disturb the protein synthesis. One to four hydroxyl functions of the small aminoglycoside…”
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Synthesis and Transfection Properties of a Series of Lipidic Neamine Derivatives by Le Gall, Tony, Baussanne, Isabelle, Halder, Somnath, Carmoy, Nathalie, Montier, Tristan, Lehn, Pierre, Décout, Jean-Luc

“…With the view to develop novel bioinspired nonviral vectors for gene delivery, we synthesized a series of cationic lipids with a neamine headgroup, which…”
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Copper(II) complexes of lipophilic aminoglycoside derivatives for the amino acid enantiomeric separation by ligand-exchange liquid chromatography by Zaher, Mustapha, Baussanne, Isabelle, Ravelet, Corinne, Halder, Somnath, Haroun, Mohamed, Fize, Jennifer, Décout, Jean-Luc, Peyrin, Eric

“…In this paper, a new class of ligand-exchange chiral stationary phase (LE-CSP) based on the copper complexes of lipophilic aminoglycoside derivatives was…”
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NO-NSAIDs. Part 3 by Borhade, Namdev, Rahimkhan Pathan, Asif, Halder, Somnath, Karwa, Manoj, Dhiman, Mini, Pamidiboina, Venu, Gund, Machhindra, Janardhan Deshattiwar, Jagannath, Vasantrao Mali, Sunil, Janardanrao Deshmukh, Nitin, Palanisamy Senthilkumar, Subrayan, Gaikwad, Parikshit, Goud Tipparam, Santhosh, Mudgal, Jayesh, Chandra Dutta, Milan, Usmangani Burhan, Aslam, Thakre, Gajanan, Sharma, Ankur, Deshpande, Shubhada, Chandrakant Desai, Dattatraya, Pervez Dubash, Nauzer, Kumar Jain, Arun, Sharma, Somesh, Venkata Subrahmanya Nemmani, Kumar, Satyam, Apparao

“…In continuation of our efforts to discover novel nitric oxide-releasing non-steroidal anti-inflammatory drugs (NO-NSAIDs) as potentially "Safe NSAIDs," we…”
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First and unexpected synthesis of macrocyclic cyclophane-based unusual α-amino acid derivatives by phosphazene base without high dilution conditions by KOTHA, Sambasivarao, HALDER, Somnath, DAMODHARAN, Lakshminarasimhan, PATTABHI, Vasantha

“…First synthesis of a macrocylic cyclophane-based unusual alpha-amino acid derivative 11 by coupling of ethyl isocyanoacetate with…”
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First synthesis of optically active benzocyclobutene and biphenylene-based unusual α-amino acid derivatives by Kotha, Sambasivarao, Sreenivasachary, Nampally, Halder, Somnath

“…Various optically pure benzocyclobutene and biphenylene-based α-amino acid derivatives are prepared in a very high diastereoselective manner via a six step…”
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