Search Results - "Sim, Galina"

Molecular and crystal structure of 5,9-dimethyl-5H-pyrano[3,2-c:5,6-c′]bis[2,1-benzothiazin]-7(9H)-one 6,6,8,8-tetroxide dimethylformamide monosolvate by Andrii Rybalka, Svitlana Shishkina, Igor Ukrainets, Lyudmila Sidorenko, Galina Sim

“…The title molecule crystallizes as a dimethylformamide monosolvate, C19H14N2O6S2·C3H7NO. The molecule was expected to adopt mirror symmetry but slightly…”
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The Crystal Structure of N-(1-Arylethyl)-4-methyl- 2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamides as the Factor Determining Biological Activity Thereof by Ukrainets, Igor V., Hamza, Ganna M., Burian, Anna A., Voloshchuk, Natali I., Malchenko, Oxana V., Shishkina, Svitlana V., Danylova, Irina A., Sim, Galina

“…In order to detect new structural and biological patterns in a series of hetaryl-3-carboxylic acid derivatives, the optically pure (S)- and (R)-enantiomers of…”
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The Study of the Structure—Diuretic Activity Relationship in a Series of New N-(Arylalkyl)-6-hydroxy-2-methyl-4-oxo-2,4-dihydro-1H-pyrrolo-[3,2,1-ij]quinoline-5-carboxamides by Ukrainets, Igor, Golik, Mykola, Sidorenko, Lyudmila, Korniyenko, Valentina, Grinevich, Lina, Sim, Galina, Kryvanych, Olga

“…In accordance with the principles of “me-too” technique, the preparative method for obtaining has been proposed, and the synthesis of a large series of new…”
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Synthesis and Regularities of the Structure–Activity Relationship in a Series of N-Pyridyl-4-methyl-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamides by Ukrainets, Igor V., Burian, Anna A., Hamza, Ganna M., Voloshchuk, Natali I., Malchenko, Oxana V., Shishkina, Svitlana V., Sidorenko, Lyudmila V., Burian, Kateryna O., Sim, Galina

“…According to our quantum and chemical calculations 4-methyl-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxylic acid imidazolide is theoretically almost as reactive…”
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Molecular Conformations and Biological Activity of N-Hetaryl(aryl)alkyl-4-methyl-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamides by Ukrainets, Igor, Hamza, Ganna, Burian, Anna, Voloshchuk, Natali, Malchenko, Oxana, Shishkina, Svitlana, Grinevich, Lina, Grynenko, Vasyl, Sim, Galina

“…The analysis of our previous studies on the search for synthetic analgesics among N-R-amides of bicyclic hetaryl-3-carboxylic acids has been performed; on its…”
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Synthesis, Spatial Structure and Analgesic Activity of Sodium 3-Benzylaminocarbonyl-1-methyl-2,2-dioxo-1H-2λ⁶,1-benzothiazin-4-olate Solvates by Ukrainets, Igor V, Petrushova, Lidiya A, Shishkina, Svitlana V, Grinevich, Lina A, Sim, Galina

“…In order to obtain and then test pharmocologically any possible conformers of the new feasible analgesic benzyl-4-hydroxy-1-methyl-2,2-dioxo-1…”
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Design, Synthesis and Biological Evaluation of Novel N-Alkyl-4-Methyl-2,2- Dioxo-1H-2λ 6 ,1-Benzothiazine-3-Carboxamides as Promising Analgesics by Ukrainets, Igor, Burian, Anna, Voloshchuk, Natali, Taran, Illia, Shishkina, Svitlana, Severina, Hanna, Grinevich, Lina, Sim, Galina, Burian, Kateryna, Georgiyants, Victoriya

“…An analysis of the literature on the painkillers long used in traditional medicine, which are isolated from plant materials, has shown that many of them are…”
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Molecular and crystal structure of 5,9-dimethyl-5 H -pyrano[3,2- c :5,6- c ′]bis[2,1-benzothiazin]-7(9 H )-one 6,6,8,8-tetroxide dimethylformamide monosolvate by Rybalka, Andrii, Shishkina, Svitlana, Ukrainets, Igor, Sidorenko, Lyudmila, Sim, Galina

“…The title molecule crystallizes as a dimethylformamide monosolvate, C 19 H 14 N 2 O 6 S 2 ·C 3 H 7 NO. The molecule was expected to adopt mirror symmetry but…”
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Mol-ecular and crystal structure of 5,9-dimethyl-5H-pyrano3,2-c:5,6-c'bis-2,1-benzo-thia-zin-7(9H)-one 6,6,8,8-tetroxide di-methyl-formamide monosolvate by Rybalka, Andrii, Shishkina, Svitlana, Ukrainets, Igor, Sidorenko, Lyudmila, Sim, Galina

“…The title mol-ecule crystallizes as a di-methyl-formamide monosolvate, C19H14N2O6S2·C3H7NO. The mol-ecule was expected to adopt mirror symmetry but slightly…”
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Mol-ecular and crystal structure of 5,9-dimethyl-5 H -pyrano[3,2- c :5,6- c ']bis-[2,1-benzo-thia-zin]-7(9 H )-one 6,6,8,8-tetroxide di-methyl-formamide monosolvate by Rybalka, Andrii, Shishkina, Svitlana, Ukrainets, Igor, Sidorenko, Lyudmila, Sim, Galina

“…The title mol-ecule crystallizes as a di-methyl-formamide monosolvate, C H N O S ·C H NO. The mol-ecule was expected to adopt mirror symmetry but slightly…”
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Mol­ecular and crystal structure of 5,9-dimethyl-5H-pyrano[3,2-c:5,6-c′]bis­[2,1-benzo­thia­zin]-7(9H)-one 6,6,8,8-tetroxide di­methyl­formamide monosolvate by Rybalka, Andrii, Shishkina, Svitlana, Ukrainets, Igor, Sidorenko, Lyudmila, Sim, Galina

“…The benzo­thia­zine skeleton is not planar, with a maximum deviation of 0.3154 (11) Å from the least-squares plane. The mol­ecule was expected to adopt mirror…”
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Biological properties of two enantiomorphic forms of N -(2,6-dimethylphenyl)-4-hydroxy-2,2-dioxo-1 H -2λ 6 ,1-benzothiazine-3-carboxamide, a structural analogue of piroxicam by Shishkina, Svitlana V., Ukrainets, Igor V., Vashchenko, Olga V., Voloshchuk, Natali I., Bondarenko, Pavlo S., Petrushova, Lidiya A., Sim, Galina

“…The title benzothiazine-3-carboxamide, C 17 H 16 N 2 O 4 S, crystallized in two enantiomorphic crystal forms with the space groups P 3 2 and P 3 1 despite the…”
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Biological properties of two enantiomorphic forms of N‐(2,6‐dimethylphenyl)‐4‐hydroxy‐2,2‐dioxo‐1H‐2λ6,1‐benzothiazine‐3‐carboxamide, a structural analogue of piroxicam by Shishkina, Svitlana V., Ukrainets, Igor V., Vashchenko, Olga V., Voloshchuk, Natali I., Bondarenko, Pavlo S., Petrushova, Lidiya A., Sim, Galina

“…The title benzothiazine‐3‐carboxamide, C17H16N2O4S, crystallized in two enantiomorphic crystal forms with the space groups P32 and P31 despite the absence of a…”
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Biological properties of two enantiomorphic forms of N-(2,6-dimethylphenyl)-4-hydroxy-2,2-dioxo-1H-2λ 6 ,1-benzothiazine-3-carboxamide, a structural analogue of piroxicam by Shishkina, Svitlana V, Ukrainets, Igor V, Vashchenko, Olga V, Voloshchuk, Natali I, Bondarenko, Pavlo S, Petrushova, Lidiya A, Sim, Galina

“…The title benzothiazine-3-carboxamide, C H N O S, crystallized in two enantiomorphic crystal forms with the space groups P3 and P3 despite the absence of a…”
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Molecular Conformations and Biological Activity of N-Hetaryl(aryl)alkyl-4-methyl-2,2-dioxo-1H-2λ^sup 6^, 1-benzothiazine-3-carboxamides by Ukrainets, Igor V, Hamza, Ganna M, Burian, Anna A, Voloshchuk, Natali I, Malchenko, Oxana V, Shishkina, Svitlana V, Grinevich, Lina A, Grynenko, Vasyl V, Sim, Galina

“…According to the results of the pharmacological tests carried out on the model of carrageenan inflammation it has been found that all without exception…”
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Synthesis, Spatial Structure and Analgesic Activity of Sodium 3-Benzylaminocarbonyl-1-methyl-2,2-dioxo-1H-2[lamda]^sup 6^,1-benzothiazin-4-olate Solvates by Ukrainets, Igor V, Petrushova, Lidiya A, Shishkina, Svitlana V, Grinevich, Lina A, Sim, Galina

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Crystal Habits and Biological Properties of N-(4-Trifluoromethylphenyl)-4-Hydroxy-2,2-Dioxo-1H-2λ6,1-Benzothiazine-3-Carboxamide by Ukrainets, Igor V., Petrushova, Lidiya A., Fedosov, Andrii I., Voloshchuk, Natali I., Bondarenko, Pavlo S., Shishkina, Svitlana V., Sidorenko, Lyudmila V., Sim, Galina

“…In order to study polymorphic modifications of N-(4-trifluoromethylphenyl)-4-hydroxy-2,2-dioxo-1H-2λ6,1-benzothiazine-3-carboxamide, which is of interest as a…”
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The Study of the Structure-Diuretic Activity Relationship in a Series of New N -(Arylalkyl)-6-hydroxy-2-methyl-4-oxo-2,4-dihydro-1 H -pyrrolo-[3,2,1- ij ]quinoline-5-carboxamides by Ukrainets, Igor V, Golik, Mykola Y, Sidorenko, Lyudmila V, Korniyenko, Valentina I, Grinevich, Lina A, Sim, Galina, Kryvanych, Olga V

“…In accordance with the principles of "me-too" technique, the preparative method for obtaining has been proposed, and the synthesis of a large series of new…”
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The Effective Synthesis of N-(Arylalkyl)-1-R-4-hydroxy-2,2-dioxo- 1H-2[lamda]^sup 6^,1-benzothiazine-3-carboxamides as Promising Analgesics of a New Chemical Class by Ukrainets, Igor V, Petrushova, Lidiya A, Dzyubenko, Sergiy P, Sim, Galina, Grinevich, Lina A

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Synthesis, Structure, and Analgesic Properties of Halogen-Substituted 4-Hydroxy-2,2-dioxo-1H-2[lamda]^sup 6^, 1-benzothiazine-3-carboxanilides by Ukrainets, Igor V, Petrushova, Lidiya A, Shishkina, Svitlana V, Sidorenko, Lyudmila V, Sim, Galina, Kryvanych, Olga V

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