Search Results - "Shiga, Futoshi"

Asymmetric Total Synthesis of (+)- and ent-(−)-Yatakemycin and Duocarmycin SA:  Evaluation of Yatakemycin Key Partial Structures and Its Unnatural Enantiomer by Tichenor, Mark S, Trzupek, John D, Kastrinsky, David B, Shiga, Futoshi, Hwang, Inkyu, Boger, Dale L

“…Complementary to studies that provided the first yatakemycin total synthesis resulting in its structure revision and absolute stereochemistry assignment, a…”
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Synthesis and antitumor activity of novel cyclopropapyrroloindole(CPI) derivatives bearing methoxycarbonyl and trifluoromethyl groups by Fukuda, Yasumichi, Furuta, Hirosuke, Shiga, Futoshi, Oomori, Yasuo, Kusama, Yoshie, Ebisu, Hiroyuki, Terashima, Shiro

“…The title synthesis was achieved by employing oxidative cyclization of the enaminoester as a key step. Some of these novel…”
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Design and synthesis of novel 7-heterocycle-6-trifluoromethyl-3-oxoquinoxaline-2-carboxylic acids bearing a substituted phenyl group as superior AMPA receptor antagonists with good physicochemical properties by Takano, Yasuo, Shiga, Futoshi, Asano, Jun, Hori, Wataru, Fukuchi, Kazunori, Anraku, Tsuyoshi, Uno, Takashi

“…We describe the design, synthesis, and physicochemical properties and biological properties of a novel series of…”
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Design, synthesis, and AMPA receptor antagonistic activity of a novel 6-nitro-3-oxoquinoxaline-2-carboxylic acid with a substituted phenyl group at the 7 position by Takano, Yasuo, Shiga, Futoshi, Asano, Jun, Ando, Naoki, Uchiki, Hideharu, Fukuchi, Kazunori, Anraku, Tsuyosi

“…We describe the design, synthesis, and biological properties of a novel series of 6-nitro-3-oxoquinoxaline-2-carboxylic acids which bear a substituted phenyl…”
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Design and synthesis of novel 7-heterocycle-6-trifluoromethyl-3-oxoquinoxaline-2-carboxylic acids bearing a substituted phenyl group as superior AMPAreceptor antagonists with good physicochemical properties by TAKANO, Yasuo, SHIGA, Futoshi, ASANO, Jun, HORI, Wataru, FUKUCHI, Kazunori, ANRAKU, Tsuyoshi, UNO, Takashi

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Synthesis and AMPA receptor antagonistic activity of a novel class of quinoxalinecarboxylic acid with a substituted phenyl group at the C-7 position by TAKANO, Yasuo, SHIGA, Futoshi, ASANO, Jun, ANDO, Naoki, UCHIKI, Hideharu, ANRAKU, Tsuyosi

“…The synthesis and biological properties of a novel class of 7-heterocycle-substituted quinoxalinecarboxylic acids, which bear a substituted phenyl group…”
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Synthesis and AMPA receptor antagonistic activity of a novel 7-imidazolyl-6-trifluoromethyl quinoxalinecarboxylic acid with a substituted phenyl group and improved its good physicochemical properties by introduced CF3 group by TAKANO, Yasuo, SHIGA, Futoshi, ASANO, Jun, HORI, Wataru, ANRAKU, Tsuyosi, UNO, Takashi

“…We describe the synthesis, physicochemical, and biological properties of a novel series of 7-imidazolyl-6-trifluoromethyl quinoxalinecarboxylic acids with a…”
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Synthesis of 6-Alkylaminopyridazine-3-carboxylic Acid Derivatives as Dopamine β-Hydroxylase Inhibitors by KONNO, Shoetsu, SAGI, Mataichi, WADA, Kunio, SHIGA, Futoshi, YAMANAKA, Hiroshi

“…A series of 6-alkylaminopyridazine-3-carboxylic acid derivatives was tested for dopamine β-hydroxylase inhibitory activity in vitro according to the method of…”
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ドーパミンβ-水酸化酵素阻害活性を持つ6-アルキルアミノピリダジン-3-カルボン酸誘導体の合成 by 今野, 昌悦, 鷺, 又市, 和田, 邦雄, 志賀, 太, 山中, 宏

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Novel Syntheses of Optically Active CC-1065, U-73,975(Adozelesin), U-80,244(Carzelesin), U-77,779 (Bizelesin), KW-2189, and DU-86 by Fukuda, Yasumichi, Furuta, Hirosuke, Shiga, Futoshi, Asahina, Yoshikazu, Terashima, Shiro

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Synthesis and reaction of tributylstannylpyrazoles by SAKAMOTO, T, SHIGA, F, UCHIYAMA, D, KONDO, Y, YAMANAKA, H

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Synthesis of 6-Alkylaminopyridazine-3-carboxylic Acid Derivatives as Dopamine β-Hydroxylase Inhibitors by KONNO, Shoetsu, SAGI, Mataichi, WADA, Kunio, SHIGA, Futoshi, YAMANAKA, Hiroshi

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