Search Results - "Shetnev, A. A."

Room Temperature Synthesis of Bioactive 1,2,4-Oxadiazoles by Baykov, Sergey V, Shetnev, Anton A, Semenov, Artem V, Baykova, Svetlana O, Boyarskiy, Vadim P

“…1,2,4-Oxadiazole is an essential motif in drug discovery represented in many experimental, investigational, and marketed drugs. This review covers synthetic…”
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Synthesis, Antibacterial, and Antimonooxidase Activity of 4-(2-Methyl-1,3-oxazol-5-yl)benzenesulfonamide by Gasilina, O. A., Romanycheva, A. A., Shetnev, A. A., Korsakov, M. K.

“…A new method for obtaining 4-(2-methyl-1,3-oxazol-5-yl)benzenesulfonamide, an antiglaucomatous drug candidate oxazopt, was developed using a diazotization…”
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Hybrid 2D Supramolecular Organic Frameworks (SOFs) Assembled by the Cooperative Action of Hydrogen and Halogen Bonding and π⋯π Stacking Interactions by Baykov, Sergey V, Semenov, Artem V, Presnukhina, Sofia I, Tarasenko, Marina V, Shetnev, Anton A, Frontera, Antonio, Boyarskiy, Vadim P, Kukushkin, Vadim Yu

“…The - and -isomers of 6-(3-(3,4-dichlorophenyl)-1,2,4-oxadiazol-5-yl)cyclohex-3-ene-1-carboxylic acid ( - and - ) were obtained by the reaction of…”
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Synthesis and Monoamine Oxidase Inhibition Properties of (Sulfamoylphenyl)quinoline-4-carboxylic Acids by Efimova, J., Shetnev, A., Korsakov, M., Petersen, E., Petzer, A., Petzer, J. P.

“…By reaction between acetylbenzenesulfonamides with several substituted isatins, we have synthesized a series of 22 primary sulfonamides, 16 of which were…”
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N-Arylation of 1,2,4- and 1,3,4-Oxadiazolones under Activated Aromatic Nucleophilic Substitution Conditions by Konstantinova, A. S., Shetnev, A. A., Volobueva, A. S., Korsakov, M. K.

“…The possibilities of N -arylation of 1,2,4-oxadiazol-5(4 H )-ones and 1,3,4-oxadiazol-2(3 H )-ones with various electron-deficient chloro- and…”
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Unusual Formation of 1,2,4-Oxadiazine Core in Reaction of Amidoximes with Maleic or Fumaric Esters by Presnukhina, Sofia I, Tarasenko, Marina V, Geyl, Kirill K, Baykova, Svetlana O, Baykov, Sergey V, Shetnev, Anton A, Boyarskiy, Vadim P

“…We have developed a simple and convenient method for the synthesis of 3-aryl- and 3-hetaryl-1,2,4-oxadiazin-5-ones bearing an easily functionalizable…”
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Synthesis and Evaluation of Antibacterial Activity of 1,2,4-Oxadiazole-Containing Biphenylcarboxylic Acids by Tarasenko, M. V., Presnukhina, S. I., Baikov, S. V., Shetnev, A. A.

“…A one-pot method for the synthesis of biphenylcarboxylic acids containing 1,2,4-oxadiazole ring in the NaOH–DMSO system was developed. The results of in vitro…”
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Synthesis and Antimicrobial Activity of Hexahydrochromeno[4,3-d]pyrimidine-2-thiones Thiouronium Salts by Makarova, E. S., Romanycheva, A. A., Blyumina, M. V., Shetnev, A. A., Filimonov, S. I.

“…The thiouronium salts of chromeno[4,3- d ]pyrimidine-2-thiones were isolated as individual diastereomers and characterized by 1 H, 13 C NMR spectroscopy and…”
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2-(1,2,4-Oxadiazol-5-yl)anilines Based on Amidoximes and Isatoic Anhydrides: Synthesis and Structure Features by Tarasenko, M. V., Kotlyarova, V. D., Baykov, S. V., Shetnev, A. A.

“…An efficient one-pot method was developed for the synthesis of 2-(1,2,4-oxadiazol-5-yl)anilines via the reaction of amidoximes with isatoic anhydrides in a…”
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Synthesis of 3,5-Disubstituted-1,2,4-oxadiazole Sulfonamides in the Superbasic t-BuONa/DMAA System by Efimova, J. A., Shetnev, A. A., Gasilina, O. A., Tarasenko, M. V., Korsakov, M. K.

“…An improved synthesis of 3,5-disubstituted-1,2,4-oxadiazoles with a sulfonamide fragment is proposed. Our previously developed synthesis of the target…”
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Pharmacological Properties of Sulfonamide Derivatives, New Inhibitors of Carbonic Anhydrase by Khokhlov, A. L., Shetnev, A. A., Korsakov, M. K., Fedorov, V. N., Tyushina, A. N., Volkhin, N. N., Vdovichenko, V. P.

“…Selective blocking of individual isoforms of carbonic anhydrase (CA) is now one of the main directions in the development of its inhibitors. The new…”
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Comparative Structural Study of Three Tetrahalophthalic Anhydrides: Recognition of X···O(anhydride) Halogen Bond and πh···O(anhydride) Interaction by Baykov, Sergey V, Semenov, Artem V, Katlenok, Eugene A, Shetnev, Anton A, Bokach, Nadezhda A

“…Structures of three tetrahalophthalic anhydrides (TXPA: halogen = Cl (TCPA), Br (TBPA), I (TIPA)) were studied by X-ray diffraction, and several types of…”
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Study of biotransformation of new selective carbonic anhydrase II inhibitor 4-(2-methyl-1,3-oxazole-5-yl)-benzenesulfonamide by Khokhlov, A. L., Yaichkov, I. I., Shetnev, A. A., Ivanovskiy, S. A., Korsakov, M. K., Gasilina, O. A., Volkhin, N. N., Petukhov, S. S.

“…The aim of the study was to determine biotransformation products of a new selective carbonic anhydrase II inhibitor –…”
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Synthesis of substituted hexahydro-2H-chromeno[4,3-d]pyrimidine-2,5-diones and their modification at the hydroxy group by Makarova, E. S., Kabanova, M. V., Filimonov, S. I., Shetnev, A. A., Suponitsky, K. Yu

“…We proposed an approach for the preparation of substituted hexahydro-2 H -chromeno-[4,3- d ]pyrimidine-2,5-diones and studied their selective acylation and…”
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Design of 4-Substituted Sulfonamidobenzoic Acid Derivatives Targeting Coxsackievirus B3 by Shetnev, Anton A, Volobueva, Alexandrina S, Panova, Valeria A, Zarubaev, Vladimir V, Baykov, Sergey V

“…A series of novel 4-substituted sulfonamidobenzoic acid derivatives was synthesized as the structural evolution of…”
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Regioselective synthesis of substituted tetrahydrochromeno[2,3-d]pyrimidin-2-ones and -pyrimidine-2-thiones by Makarova, E. S., Kabanova, M. V., Filimonov, S. I., Chirkova, Zh. V., Ivanovsky, S. A., Shetnev, A. A., Suponitsky, K. Yu

“…The regioselective synthesis of the substituted (4 R *,10a R *)-4-aryltetrahydro-2 H -chromeno[2,3- d ]pyrimidin-2-ones, -pyrimidine-2-thiones and (4 R *,5 R…”
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Synthesis and Photoluminescent Properties of 2-(3-Carboxymethylindazol-1-yl)anilines by Shetnev, A. A., Panova, V. A., Kutuzova, P. M., Tarasenko, M. V., Zhmykhova, M. V., Baykov, S. V., Filimonov, S. I.

“…A two-stage method for the preparation of 2-(3-carboxymethylindazol-1-yl)anilines using the N -arylation reaction of 3-carboxymethylindazoles with o…”
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Synthesis and properties of substituted 2-thioxohexahydropyrimidine-5-carbohydrazides by Makarova, E. S., Kabanova, M. V., Danilova, A. S., Filimonov, S. I., Smirnova, E. A., Shetnev, A. A.

“…A regioselective method for the synthesis of substituted (4 R* ,5 S* ,6 R* )-2-thioxohexahydro-pyrimidine-5-carbohydrazides from the corresponding…”
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Synthesis and Monoamine Oxidase Inhibition Properties of 4-(2-Methyloxazol-4-yl)benzenesulfonamide by Shetnev, Anton A, Efimova, Julia A, Korsakov, Mikhail K, Petzer, Anél, Petzer, Jacobus P

“…4-(2-Methyloxazol-4-yl)benzenesulfonamide was synthesized by the reaction of 4-(2-bromoacetyl)benzenesulfonamide with an excess of acetamide. The compound was…”
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N-Arylamino-1,2,4-oxadiazol-5(4H)-ones: Synthesis, Luminescent, Antibacterial, and Antienteroviral Properties by Konstantinova, A. S., Shetnev, A. A., Semenov, A. V., Presnukhina, S. I., Romanycheva, A. A., Volobueva, A. S., Zarubaev, V. V., Baykov, S. V., Korsakov, M. K.

“…Method for the preparation of N -arylamino-1,2,4-oxadiazol-5(4 H )-ones via reduction of N -nitrophenyl-1,2,4-oxadiazol-5(4 H )-ones with tin(II) chloride has…”
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