Search Results - "Shedage, Sandeep A"

Identification and preclinical characterization of a novel and potent poly (ADP-ribose) polymerase (PARP) inhibitor ZYTP1 by Jain, Mukul R., Mohapatra, Jogeswar, Bandhyopadhyay, Debdutta, Chatterjee, Abhijit, Ghoshdastidar, Krishnarup, Patel, Dinesh, Patel, Ankit, Bhayani, Hitesh, Srivastava, Brijesh Kumar, Shedage, Sandeep A., Kadam, Pravin, Sundar, Rajesh, Patel, Harilal, Giri, Poonam, Patel, Prakash, Gupta, Laxmikant, Srinivas, Nuggehally R., Patel, Pankaj R., Desai, Ranjit C.

“…Purpose Poly(ADP-ribose) polymerase-1 (PARP-1) is a nuclear enzyme involved in the detection and repair of DNA damage. Studies have shown that inhibition of…”
Get full text

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist by Kumar Srivastava, Brijesh, Soni, Rina, Patel, Jayendra Z, Jha, Satadru, Shedage, Sandeep A, Gandhi, Neha, Sairam, Kalapatapu V V M, Pawar, Vishwanath, Sadhwani, Nisha, Mitra, Prasenjit, Jain, Mukul R, Patel, Pankaj R

“…Facile synthesis of biaryl pyrazole sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxylic acid…”
Get full text

Bioisosteric replacement of dihydropyrazole of 4S-(-)-3-(4-chlorophenyl)-N-methyl-N'-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole by Srivastava, Brijesh Kumar, Soni, Rina, Joharapurkar, Amit, Sairam, Kalapatapu V V M, Patel, Jayendra Z, Goswami, Amitgiri, Shedage, Sandeep A, Kar, Sidhartha S, Salunke, Rahul P, Gugale, Shivaji B, Dhawas, Amol, Kadam, Pravin, Mishra, Bhupendra, Sadhwani, Nisha, Unadkat, Vishal B, Mitra, Prasenjit, Jain, Mukul R, Patel, Pankaj R

“…Design, synthesis and conformational analysis of few imidazole and oxazole as bioisosters of…”
Get full text

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1 H-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist by Kumar Srivastava, Brijesh, Soni, Rina, Patel, Jayendra Z., Jha, Satadru, Shedage, Sandeep A., Gandhi, Neha, Sairam, Kalapatapu V.V.M., Pawar, Vishwanath, Sadhwani, Nisha, Mitra, Prasenjit, Jain, Mukul R., Patel, Pankaj R.

“…Facile synthesis of biaryl pyrazole sulfonamide derivative of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1 H-pyrazole-3-carboxylic acid…”
Get full text

Facile synthesis, ex-vivo and in vitro screening of 3-sulfonamide derivative of 5-(4-chlorophenyl)-l-(2.4-dichlorophenyl)-4-methyl-lH-pyrazole-3-carboxylic acid piperidin-1-ylamide (SR141716) a potent CB1 receptor antagonist by BRIJESH KUMAR SRIVASTAVA, SONI, Rina, JAIN, Mukul R, PATEL, Pankaj R, PATEL, Jayendra Z, JHA, Satadru, SHEDAGE, Sandeep A, GANDHI, Neha, SAIRAM, Kalapatapu V. V. M, PAWAR, Vishwanath, SADHWANI, Nisha, MITRA, Prasenjit

Get full text

Bioisosteric replacement of dihydropyrazole of 4 S-(−)-3-(4-chlorophenyl)- N-methyl- N′-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-1H-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole by Srivastava, Brijesh Kumar, Soni, Rina, Joharapurkar, Amit, Sairam, Kalapatapu V.V.M., Patel, Jayendra Z., Goswami, Amitgiri, Shedage, Sandeep A., Kar, Sidhartha S., Salunke, Rahul P., Gugale, Shivaji B., Dhawas, Amol, Kadam, Pravin, Mishra, Bhupendra, Sadhwani, Nisha, Unadkat, Vishal B., Mitra, Prasenjit, Jain, Mukul R., Patel, Pankaj R.

“…Design, synthesis and conformational analysis of few imidazole and oxazole as bioisosters of 4 S-(−)-3-(4-chlorophenyl)- N-methyl-…”
Get full text

Bioisosteric replacement of dihydropyrazole of 4S-(-)-3-(4-chlorophenyl)-N-methyl-N'-[(4-chlorophenyl)-sulfonyl]-4-phenyl-4,5-dihydro-lH-pyrazole-1-caboxamidine (SLV-319) a potent CB1 receptor antagonist by imidazole and oxazole by BRIJESH KUMAR SRIVASTAVA, SONI, Rina, DHAWAS, Amol, KADAM, Pravin, MISHRA, Bhupendra, SADHWANI, Nisha, UNADKAT, Vishal B, MITRA, Prasenjit, JAIN, Mukul R, PATEL, Pankaj R, JOHARAPURKAR, Amit, SAIRAM, Kalapatapu V. V. M, PATEL, Jayendra Z, GOSWAMI, Amitgiri, SHEDAGE, Sandeep A, KAR, Sidhartha S, SALUNKE, Rahul P, GUGALE, Shivaji B

Get full text