Search Results - "Sestili, I"

LTB4 as marker of 5-LO inhibitory activity of two new N- ω-ethoxycarbonyl-4-quinolones by Bossù, E, Aglianò, A.M, Desideri, N, Sestili, I, Porrà, R, Grandilone, M, Quaglia, M.G

“…The supposed 5-LO inhibitory activity of two N- ω-ethoxycarbonyl-4-quinolones was tested determining leukotriene B4 (LTB 4) in RBL-1 cell cultures, pretreated…”
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Synthesis and Anti-Human Immunodeficiency Virus Type 1 Integrase Activity of Hydroxybenzoic and Hydroxycinnamic Acid Flavon-3-yl Esters by Desideri, N, Sestili, I, Stein, ML, Tramontano, E, Corrias, S, La Colla, P

“…A series of new hydroxybenzoic and hydroxycinnamic acid flavon-3-yl esters were synthesized in order to obtain compounds targeting the human immunodeficiency…”
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Synthesis and Pharmacological Evaluation of 1,2-Dihydrospiro[isoquinoline-4(3H),4′-piperidin]-3-ones as Nociceptin Receptor Agonists by Mustazza, Carlo, Borioni, Anna, Sestili, Isabella, Sbraccia, Maria, Rodomonte, Andrea, Del Giudice, Maria Rosaria

“…Some synthesized 1,2-dihydrospiro[isoquinoline-4(3H),4′-piperidin]-3-ones were evaluated as ligands for nociceptin receptor (NOP receptor). Their affinity was…”
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Synthesis of some guanylhydrazones and imidazolinylhydrazones as thromboxane-synthase and platelet aggregation inhibitors by Desideri, N, Sestili, I, Piccardoni, P, Rotondo, S, Cerletti, C, Stein, M L

“…The imidazolinylhydrazones of (3-pyridinyloxy)-acetaldehyde and of 6-[3-(2-formyl-pyridinyl)oxy]hexanoic acid were synthesized as cyclic analogues of the…”
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Synthesis and Evaluation as NOP Ligands of Some Spiro[piperidine-4,2′(1′H)-quinazolin]-4′(3′H)-ones and Spiro[piperidine-4,5′(6′H)-[1,2,4]triazolo[1,5-c]quinazolines] by Mustazza, Carlo, Borioni, Anna, Sestili, Isabella, Sbraccia, Maria, Rodomonte, Andrea, Ferretti, Rosella, Giudice, Maria Rosaria Del

“…Some spiro[piperidine-4,2′(1′H)-quinazolin]-4′(3′H)-ones 3 and spiro[piperidine-4,5′(6′H)-[1,2,4]triazolo[1,5-c]quinazolines] 4 were synthesized and evaluated…”
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A new synthetic approach of N-(4-amino-2-methylquinolin-6-yl)-2-(4-ethylphenoxymethyl)benzamide (JTC-801) and its analogues and their pharmacological evaluation as nociceptin receptor (NOP) antagonists by Sestili, Isabella, Borioni, Anna, Mustazza, Carlo, Rodomonte, Andrea, Turchetto, Luciana, Sbraccia, Maria, Riitano, Daniela, Del Giudice, Maria Rosaria

“…A series of 4-amino-2-methylquinoline and 4-aminoquinazoline derivatives, including the reference NOP antagonist JTC-801, were synthesized by an alternative…”
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Anti-picornavirus activity of new substituted flavons and flavanones by Tomao, P, Conti, C., Orsi, N., Desideri, N., Sestili, I., Stein, M.L.

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N-omega-carbethoxypentyl-4-quinolones: a new class of leukotriene biosynthesis inhibitors by Desideri, N, Sestili, I, Stein, M L, Manarini, S, Dell'Elba, G, Cerletti, C

“…6-[(4-Quinolinyl)oxy]hexanoic acids and the corresponding esters were designed and synthesized as inhibitors of the production of arachidonic acid metabolites…”
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Chiral discrimination and antipicornavirus activity of 6-oxazolinylisoflavan by Quaglia, M G, Desideri, N, Bossù, E, Sestili, I, Tomao, P, Conti, C, Orsi, N

“…Racemic 6-oxazolinylisoflavan, a highly effective inhibitor of rhinovirus serotype 1B in vitro, was resolved by high-performance liquid chromatography on a…”
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Synthesis and binding properties to GABA receptors of 3-hydroxypyridinyl- and 3-hydroxypiperidinyl-analogues of baclofen by Desideri, N, Galli, A, Sestili, I, Stein, M L

“…The synthesis of 3-(3-hydroxy-2-pyridinyl)propanoic acid, 3-(3-hydroxy-2-pyridinyl)-4-aminobutanoic acid, their corresponding piperidine compounds, and of some…”
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An improved determination ofG A(x) from single-π+ electroproduction by Paver, N., Verzegnassi, C., Pistilli, P., Sestili, I.

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Synthesis of guanylhydrazones derived from 3-pyridinol and evaluation of their effect on serum thromboxane B2 and prostaglandin E2 production by Desideri, N, Stein, M L, Conti, S, Sestili, I, Bucchi, F, Cerletti, C

“…3-Pyridyloxyacetaldehyde guanylhydrazone and the guanylhydrazones of pyridine-2- and -4-aldehydes substituted at the 3-position with the omega-carboxypentyloxy…”
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The expression analysis of mouse interleukin-6 splice variants argued against their biological relevance by Annibalini, Giosue, Guescini, Michele, Agostini, Deborah, De Matteis, Rita, Sestili, Piero, Tibollo, Pasquale, Mantuano, Michela, Martinelli, Chiara, Stocchi, Vilberto

“…Alternative splicing generates several interleukin-6 (IL-6) isoforms; for them an antagonistic activity to the wild-type IL-6 has been proposed. In this study…”
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