Search Results - "Sayago, Francisco J."

Ru-catalyzed C H functionalization of phenylglycine derivatives: Synthesis of isoquinoline-1-carboxylates and isoindoline-1-carboxylates by Ruiz, Sara, Sayago, Francisco J., Cativiela, Carlos, Urriolabeitia, Esteban P.

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Nanoparticle-induced vascular blockade in human prostate cancer by Agemy, Lilach, Sugahara, Kazuki N., Kotamraju, Venkata Ramana, Gujraty, Kunal, Girard, Olivier M., Kono, Yuko, Mattrey, Robert F., Park, Ji-Ho, Sailor, Michael J., Jimenez, Ana I., Cativiela, Carlos, Zanuy, David, Sayago, Francisco J., Aleman, Carlos, Nussinov, Ruth, Ruoslahti, Erkki

“…The tumor-homing pentapeptide CREKA (Cys-Arg-Glu-Lys-Ala) specifically homes to tumors by binding to fibrin and fibrin-associated clotted plasma proteins in…”
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Stereoselective Synthesis of α-Amino-C-phosphinic Acids and Derivatives by Viveros-Ceballos, José Luis, Ordóñez, Mario, Sayago, Francisco J, Cativiela, Carlos

“…α-Amino-C-phosphinic acids and derivatives are an important group of compounds of synthetic and medicinal interest and particular attention has been dedicated…”
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Aldolase-Catalyzed Synthesis of Conformationally Constrained Iminocyclitols: Preparation of Polyhydroxylated Benzopyrrolizidines and Cyclohexapyrrolizidines by Laborda, Pedro, Sayago, Francisco J, Cativiela, Carlos, Parella, Teodor, Joglar, Jesús, Clapés, Pere

“…A straightforward chemo-enzymatic synthesis of new polyhydroxylated benzo­pyrrolizidines and cyclo­hexa­pyrrolizidines is developed. The two-step strategy…”
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Dynamic Kinetic Resolution of 1,3-Dihydro-2H-isoindole-1-carboxylic Acid Methyl Ester: Asymmetric Transformations toward Isoindoline Carbamates by Morán-Ramallal, Roberto, Gotor-Fernández, Vicente, Laborda, Pedro, Sayago, Francisco J, Cativiela, Carlos, Gotor, Vicente

“…Asymmetric syntheses of isoindoline carbamates have been successfully achieved through enzyme-mediated dynamic kinetic resolution processes and without…”
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Quantum-chemical predictions of redox potentials of carbamates in methanol by Haya, Luisa, Sayago, Francisco J, Mainar, Ana M, Cativiela, Carlos, Urieta, José S

“…Redox potentials for two stepwise anodic oxidations of a series of carbamates in methanolic solution have been calculated using ab initio and DFT quantum…”
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Synthesis of quaternary α-aminophosphonic acids by Ordóñez, Mario, Sayago, Francisco J., Cativiela, Carlos

“…[Display omitted]…”
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Synthesis of β‐Aryl‐α,β‐Dehydroaminophosphonates by Pd‐Catalyzed Fujiwara–Moritani C−C Coupling by Sáez, Javier, Dalmau, David, Sayago, Francisco J., Urriolabeitia, Esteban P.

“…The treatment of diethyl α,β‐dehydroaminophosphonate  1 with various arenes (ArH=toluene 2 a , benzene 2 b , anisole 2 c , bromobenzene 2 d , chlorobenzene 2 e…”
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Amide-triazole isosteric substitution for tuning self-assembly and incorporating new functions into soft supramolecular materials by Bachl, Jürgen, Mayr, Judith, Sayago, Francisco J, Cativiela, Carlos, Díaz Díaz, David

“…The proof-of-concept for the modular synthesis of new functional soft gel materials based on amide-triazole isosteric replacement has been demonstrated. A…”
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New approaches towards the synthesis of 1,2,3,4-tetrahydro isoquinoline-3-phosphonic acid (TicP) by Viveros-Ceballos, José Luis, Matías-Valdez, Lizeth A., Sayago, Francisco J., Cativiela, Carlos, Ordóñez, Mario

“…Two new strategies for the efficient synthesis of racemic 1,2,3,4-tetrahydroisoquinoline-3-phosphonic acid (Tic P ) (±)- 2 have been developed. The first…”
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An Improved Synthesis of the Antibiotic Dehydrophos by Jiménez‐Andreu, M. Mercedes, Sayago, Francisco J., Cativiela, Carlos

“…Within this work an efficient procedure for the synthesis of the vinyl phosphonate tripeptide dehydrophos is described. This procedure constitutes a…”
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Efficient access to (1H)-isoindolin-1-one-3-carboxylic acid derivatives by orthopalladation and carbonylation of methyl arylglycinate substrates by Nieto, Sonia, Sayago, Francisco J., Laborda, Pedro, Soler, Tatiana, Cativiela, Carlos, Urriolabeitia, Esteban P.

“…The orthopalladation of methyl arylglycinate derivatives has been studied. The reaction proceeds efficiently for different electron-withdrawing and…”
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Cyclopalladation and Reactivity of Amino Esters through CH Bond Activation: Experimental, Kinetic, and Density Functional Theory Mechanistic Studies by Laga, Eduardo, García-Montero, Angel, Sayago, Francisco J., Soler, Tatiana, Moncho, Salvador, Cativiela, Carlos, Martínez, Manuel, Urriolabeitia, Esteban P.

“…The orthopalladation, through CH bond activation, of a large number of amino esters and amino phosphonates derived from phenylglycine, and having different…”
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Synthesis of [c]-Fused Bicyclic Proline Analogues by Calaza, M. Isabel, Sayago, Francisco J., Laborda, Pedro, Cativiela, Carlos

“…An overview of synthetic methods developed to build [c]‐fused bicyclic proline analogues is presented. The focus is on the preparation of azabicycles that bear…”
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First Synthesis of (R)- and (S)-1,2,3,4-Tetrahydroisoquinoline-3-phosphonic Acid (TicP) Using a Pictet-Spengler Reaction by Viveros-Ceballos, José Luis, Ordóñez, Mario, Sayago, Francisco J., Jiménez, Ana I., Cativiela, Carlos

“…We report here a practical and efficient synthesis of diethyl 1,2,3,4‐tetrahydroisoquinoline‐3‐phosphonate derivatives. The target compounds were prepared in…”
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1‐Aminovinylphosphonate Esters as Substrates for the Diels‐Alder Reaction: First Synthetic and Theoretical Study by Jiménez‐Andreu, M. Mercedes, Bueno‐Morón, Jorge, Sayago, Francisco J., Cativiela, Carlos, Tejero, Tomás, Merino, Pedro

“…The Diels‐Alder reaction of 1‐aminovinylphosphonate esters has been studied for the first time as a suitable procedure leading to quaternary carbocyclic…”
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Stereodivergent Synthesis of Two Novel α-Aminophosphonic Acids Characterised by a cis-Fused Octahydroindole System by Arizpe, Alicia, Sayago, Francisco J., Jiménez, Ana I., Ordóñez, Mario, Cativiela, Carlos

“…The synthesis of two new α‐aminophosphonic acids, namely (2S*,3aS*,7aS*)‐ and (2R*,3aS*,7aS*)‐octahydroindole‐2‐phosphonic acids, is described. They are…”
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Access to the cis-Fused Stereoisomers of Proline Analogues Containing an Octahydroindole Core by Sayago, Francisco J., Laborda, Pedro, Calaza, M. Isabel, Jiménez, Ana I., Cativiela, Carlos

“…An overview of the synthetic methods developed to build all the cis‐fused stereoisomers of octahydroindole‐2‐carboxylic acid and its α‐methylated derivative in…”
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Synthesis of Phosphoproline Derivatives with an Octahydroisoindole Structure by Arizpe, Alicia, Sayago, Francisco J., Jiménez, Ana I., Ordóñez, Mario, Cativiela, Carlos

“…The synthesis of two phosphoproline analogues possessing an octahydroisoindole structure is described for the first time. The new α‐aminophosphonic acids can…”
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Remote Substituent Effects on the Stereoselectivity and Organocatalytic Activity of Densely Substituted Unnatural Proline Esters in Aldol Reactions by de Gracia Retamosa, María, de Cózar, Abel, Sánchez, Mirian, Miranda, José I., Sansano, José M., Castelló, Luis M., Nájera, Carmen, Jiménez, Ana I., Sayago, Francisco J., Cativiela, Carlos, Cossío, Fernando P.

“…The organocatalytic activities of highly substituted proline esters obtained through asymmetric [3+2] cycloadditions of azomethine ylides derived from glycine…”
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