Search Results - "Sadeque, M"

Flow around Cylinders in Open Channels by Sadeque, M. A, Rajaratnam, N, Loewen, M. R

“…This paper presents the results of an experimental study of flow around cylindrical objects in an open channel. Cylindrical objects of equal diameter and four…”
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Effects of Bed Roughness on Flow around Bed-Mounted Cylinders in Open Channels by Sadeque, M. A, Rajaratnam, N, Loewen, M. R

“…This paper presents the results of an experimental study of flow around cylindrical objects on a rough bed in an open channel. This is an extension of a…”
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Metopimazine is primarily metabolized by a liver amidase in humans by Busby, Robert W., Cai, Xiaokun, Yang, Sihyung, Ramos, Luis, Venkatarangan, Lata, Shen, Helen, Wax, Stephen, Sadeque, Abu J. M., De Colle, Cyril

“…Metopimazine (MPZ) is a peripherally restricted, dopamine D2 receptor antagonist used for four decades to treat acute nausea and vomiting. MPZ is currently…”
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Turbulent Flow near Vertical Angled Fish Screen by Rajaratnam, N, Katopodis, C, Sadeque, M. A. F, Pokharel, N

“…Mean and turbulent flow characteristics on the upstream and downstream sides of the screen in a flow diversion channel have important implications for…”
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Biopharmaceutics Permeability Classification of Lorcaserin, a Selective 5‑Hydroxytryptamine 2C Agonist: Method Suitability and Permeability Class Membership by Chen, Chuan, Ma, Michael G, Fullenwider, Cody L, Chen, Weichao G, Sadeque, Abu J. M

“…The objectives of the study were (1) to demonstrate that a Caco-2 cell-based permeability assay, developed in our laboratory, is suitable to identify the…”
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Identification of Human Sulfotransferases Involved in Lorcaserin N-Sulfamate Formation by Sadeque, Abu J M, Palamar, Safet, Usmani, Khawja A, Chen, Chuan, Cerny, Matthew A, Chen, Weichao G

“…Lorcaserin [(R)-8-chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine] hydrochloride hemihydrate, a selective serotonin 5-hydroxytryptamine (5-HT) 5-HT(2C)…”
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Comparative study of the effect of ethanolic extract of Swietenia mahagoni seeds with rosiglitazone on experimentally induced diabetes mellitus in rats by Hasan, S M M M A, Khan, M I, Umar, B U, Sadeque, M Z

“…The study was performed to compare the blood glucose lowering effect of Swietenia mahagoni seeds with an oral antidiabetic drug, rosiglitazone in…”
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Kinetics of 5-HT2B receptor signaling: profound agonist-dependent effects on signaling onset and duration by Unett, David J, Gatlin, Joel, Anthony, Todd L, Buzard, Daniel J, Chang, Steve, Chen, Chuan, Chen, Xiaohua, Dang, Huong T-M, Frazer, John, Le, Minh K, Sadeque, Abu J M, Xing, Charles, Gaidarov, Ibragim

“…The kinetics of drug-receptor interactions can profoundly influence in vivo and in vitro pharmacology. In vitro, the potencies of slowly associating agonists…”
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Identification of human cytochrome P450 and flavin-containing monooxygenase enzymes involved in the metabolism of lorcaserin, a novel selective human 5-hydroxytryptamine 2C agonist by Usmani, Khawja A, Chen, Weichao G, Sadeque, Abu J M

“…Lorcaserin, a selective serotonin 5-hydroxytryptamine 2C receptor agonist, is being developed for weight management. The oxidative metabolism of lorcaserin,…”
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Increased drug delivery to the brain by P-glycoprotein inhibition by Sadeque, Abu J. M., Wandel, Christoph, He, Hauibing, Shah, Selina, Wood, Alastair J. J.

“…Background Although the antidiarrheal loperamide is a potent opiate, it does not produce opioid central nervous system effects at usual doses in patients. On…”
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Identification of human UDP-glucuronosyltransferases involved in N-carbamoyl glucuronidation of lorcaserin by Sadeque, Abu J M, Usmani, Khawja A, Palamar, Safet, Cerny, Matthew A, Chen, Weichao G

“…Lorcaserin, a selective serotonin 5-HT(2C) receptor agonist, is a weight management agent in clinical development. Lorcaserin N-carbamoyl glucuronidation…”
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Solid lipid nanoparticles: An effective lipid-based technology for cancer treatment by Akanda, Mushfiq, Mithu, MD Sadeque Hossain, Douroumis, Dennis

“…Solid lipid nanoparticles (SLN) are considered at the forefront of nanotechnology's rapidly developing field, with several potential applications in drug…”
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Ligand binding studies of engineered cytochrome P-450d wild type, proximal mutants, and distal mutants by Shimizu, Toru, Sadeque, Abu Jafar M, Sadeque, Gul Nahar, Hatano, Masahiro, Fujii-Kuriyama, Yoshiaki

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Effect of mechanochemical grinding conditions on the formation of pharmaceutical cocrystals and co-amorphous solid forms of ketoconazole – Dicarboxylic acid by Hossain Mithu, MD Sadeque, Ross, Steven A., Hurt, Andrew P., Douroumis, Dennis

“…Mechanochemical grinding is one of the commonly used solvent-free methods for the successful preparation of pharmaceutical cocrystals, which is marked as green…”
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Transverse myelitis in a 26-year-old male with tuberculosis by Harizi, Edlira, Shemsi, Kledisa, Kola, Erisa, Hyseni, Fjolla, Kola, Ina, Siddique, Mohammad Abubaker, Sadeque, Jafor, Decka, Arlind, Dervishi, Migena, Nasir, Fareeha, Capi, Livia, Ayala, Ivan, Ghosh, Ammy Shankar, Swarna, Sanzida Sharmin, Musa, Juna, Ahmetgjekaj, Ilir

“…Acute transverse myelitis is an inflammatory condition covering the entire cross section of the spinal cord, spreading on two or more vertebral segments,…”
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BACULOVIRUS-MEDIATED EXPRESSION AND PURIFICATION OF HUMAN FMO3 by R. L. Haining, A. P. Hunter, A. J. M. Sadeque, R. M. Philpot, A. E. Rettie

“…The baculovirus expression vector system was used to overexpress human FMO3 in insect cells for catalytic, structural, and immunochemical studies. Membranes…”
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Diagnostic Accuracy of Refractory Shadowing from Uterine Leiomyomas: Sonographic-Pathologic Correlation by Khan, T R, Afroze, N, Islam, M R, Rahman, M M, Sadeque, A M, Khan, E R

“…This cross sectional study was carried out in the Department of Radiology & Imaging, Bangladesh Institute of Research and Rehabilitation in Diabetes, Endocrine…”
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Incidence of helminthic infections and comparative study of pyrantel pamoate with levamisole and mebendazole in hospital patients at Barisal, Bangladesh by Islam, A F, Sadeque, M, Biswas, K, Ahmed, N, Mahmood, G

“…A study was carried out to find out the incidence of helminthic infections in hospitalized patients at Sher-e-Bangla Medical College, Barisal and to determine…”
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Comparative Efficacy of Dried Fruits of Carica Papaya Linn. and Vitamin-E on Preventing Hepatotoxicity in Rats by Sadeque, MZ, Begum, ZA, Umar, BU, Ferdous, AH, Sultana, S, Uddin, MK

“…In the absence of an effective treatment in modern medicine, efforts are being made to find suitable herbal remedies for hepatitis. This prospective…”
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Evaluation of culture, histological examination, serology and the rapid urease test for diagnosis of Helicobacter pylori in patients with dyspepsia in Bangladesh by Morshed, M G, Jinnah, F, Islam, M S, Rumi, M A, Ahmed, S, Ahmed, M M, Sadeque, M, Chowdhury, M F

“…Helicobacter pylori, a gram-negative, microaerophilic bacterium, has been established to have a causal association with chronic gastritis, peptic ulcer,…”
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