Search Results - "STUP, T. L"

Structure-activity and cross-resistance evaluations of a series of human immunodeficiency virus type-1-specific compounds related to oxathiin carboxanilide by BUCKHEIT, R. W, KINJERSKI, T. L, BADER, J. P, YANG, S. S, FLIAKAS-BOLTZ, V, RUSSELL, J. D, STUP, T. L, PALLANSCH, L. A, BROUWER, W. G, DAO, D. C, HARRISON, W. A, SCHULTZ, R. J

“…Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit StumbleUpon…”
Get full text

Novel Modifications in the Alkenyldiarylmethane (ADAM) Series of Non-Nucleoside Reverse Transcriptase Inhibitors by Casimiro-Garcia, Agustin, Micklatcher, Mark, Turpin, Jim A, Stup, Tracy L, Watson, Karen, Buckheit, Robert W, Cushman, Mark

“…In an effort to obtain more insight into the interaction between HIV-1 reverse transcriptase and the alkenyldiarylmethanes (ADAMs), a new series of compounds…”
Get full text

Unique Anti-Human Immunodeficiency Virus Activities of the Nonnucleoside Reverse Transcriptase Inhibitors Calanolide A, Costatolide, and Dihydrocostatolide by BUCKHEIT, R. W, WHITE, E. L, FLIAKAS-BOLTZ, V, RUSSELL, J, STUP, T. L, KINJERSKI, T. L, OSTERLING, M. C, WEIGAND, A, BADER, J. P

“…Classifications Services AAC Citing Articles Google Scholar PubMed Related Content Social Bookmarking CiteULike Delicious Digg Facebook Google+ Mendeley Reddit…”
Get full text

Structural Analogues of the Calanolide Anti-HIV Agents. Modification of the trans-10,11-Dimethyldihydropyran-12-ol Ring (Ring C) by Zembower, David E, Liao, Shuyuan, Flavin, Michael T, Xu, Ze-Qi, Stup, Tracy L, Buckheit, Robert W, Khilevich, Albert, Mar, Aye Aye, Sheinkman, Abram K

“…(+)-Calanolide A is a potent inhibitor of reverse transcriptase from human immunodeficiency virus type 1 (HIV-1), which was isolated from an extract of…”
Get full text

In vitro anti-human immunodeficiency virus (HIV) activity of the chromanone derivative, 12-oxocalanolide A, a novel NNRTI by Ze-Qi Xu, Buckheit, Robert W., Stup, Tracy L., Flavin, Michael T., Khilevich, Albert, Rizzo, John D., Lin, Lin, Zembower, David E.

“…The three chromanone derivatives, (+)-, (−)-, and (±)-12-oxocalanolide A ( 2), were evaluated for in vitro antiviral activities against HIV and simian…”
Get full text

Synthesis and anti-HIV activity of cosalane analogues incorporating nitrogen in the linker chain by CASIMIRO-GARCIA, A, DE CLERCQ, E, PANNECOUQUE, C, WITVROUW, M, STUP, T. L, TURPIN, J. A, BUCKHEIT, R. W, CUSHMAN, M

“…Introduction of an amido group or an amino moiety into the alkenyl linker chain of cosalane (1) provided a new series of analogues 3-8. The new compounds were…”
Get full text

Comparative anti-HIV evaluation of diverse HIV-1-specific reverse transcriptase inhibitor-resistant virus isolates demonstrates the existence of distinct phenotypic subgroups by Buckheit, Robert W., Fliakas-Boltz, Valerie, Decker, William Don, Roberson, Joseph L., Stup, Tracy L., Pyle, Cathi A., White, E.Lucile, McMahon, James B., Currens, Michael J., Boyd, Michael R., Bader, John P.

“…We have biologically and biochemically evaluated a structurally diverse group of HIV-1-specific reverse transcriptase (RT) inhibitors and determined that the…”
Get full text

Synthesis and Anti-HIV Activity of Cosalane Analogues with Substituted Benzoic Acid Rings Attached to the Pharmacophore through Methylene and Amide Linkers by Ruell, Jeffrey A, De Clercq, Erik, Pannecouque, Christophe, Witvrouw, Myriam, Stup, Tracy L, Turpin, Jim A, Buckheit, Robert W, Cushman, Mark

“…The cosalane pharmacophore has been extended by the attachment of two additional substituted benzoic acid rings through amide and methylene linkers. The…”
Get full text