Search Results - "Søby, Karina K"

Lu 35-138 ( (+ ) -(S ) -3-{1 -[2 -(1 -acetyl -2,3 -dihydro -1H -indol -3 -yl )ethyl] -3, 6 -dihydro -2H -pyridin -4 -yl} -6 -chloro -1H -indole ), a dopamine D4 receptor antagonist and serotonin reuptake inhibitor : Characterisation of its in vitro profile and pre-clinical antipsychotic potential by HERTEL, Peter, DIDRIKSEN, Michael, DI MAFLEO, Vincenzo, ESPOSITO, Ennio, BANG-ANDERSEN, Benny, ARMT, Jøm, POUZET, Bruno, BRENNUM, Lise T, SØBY, Karina K, LARSEN, Anna Kirstine, CHRISTOFFERSEN, Claus T, RAMIREZ, Teresa, MARCUS, Monica M, SVENSSON, Torgny H

“…The present study describes the pharmacological profile of the putative antipsychotic drug Lu 35-138…”
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Heteroaryl Analogues of AMPA. Synthesis and Quantitative Structure−Activity Relationships by Bang-Andersen, Benny, Lenz, Sibylle M, Søby, Karina K, Hansen, Hans O, Ebert, Bjarke, Bøgesø, Klaus P, Krogsgaard-Larsen, Povl

“…A number of 3-isoxazolol bioisosteres, 7a−i, of (S)-glutamic acid (Glu), in which the methyl group of (RS)-2-amino-3-(3-hydroxy-5-methylisoxazol-4-yl)propionic…”
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Excitatory Amino Acid Receptor Ligands:  Resolution, Absolute Stereochemistry, and Enantiopharmacology of 2-Amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic Acid by Johansen, Tommy N, Ebert, Bjarke, Bräuner-Osborne, Hans, Didriksen, Michael, Christensen, Inge T, Søby, Karina K, Madsen, Ulf, Krogsgaard-Larsen, Povl, Brehm, Lotte

“…(RS)-2-Amino-3-(4-butyl-3-hydroxyisoxazol-5-yl)propionic acid (Bu-HIBO, 6) has previously been shown to be an agonist at…”
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Lu 35-138 ((+)-(S)-3-{1-[2-(1-acetyl-2,3-dihydro-1H-indol-3-yl)ethyl]-3,6-dihydro-2H-pyridin-4-yl}-6-chloro-1H-indole), a dopamine D 4 receptor antagonist and serotonin reuptake inhibitor: Characterisation of its in vitro profile and pre-clinical antipsychotic potential by Hertel, Peter, Didriksen, Michael, Pouzet, Bruno, Brennum, Lise T., Søby, Karina K., Larsen, Anna Kirstine, Christoffersen, Claus T., Ramirez, Teresa, Marcus, Monica M., Svensson, Torgny H., Di Matteo, Vincenzo, Esposito, Ennio, Bang-Andersen, Benny, Arnt, Jørn

“…The present study describes the pharmacological profile of the putative antipsychotic drug Lu 35-138…”
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Aryl and cycloalkyl analogues of AMPA: synthetic, pharmacological and stereochemical aspects by Skjærbæk, Niels, Brehm, Lotte, Johansen, Tommy N., Hansen, Lene M., Nielsen, Birgitte, Ebert, Bjarke, Søby, Karina K., Stensbøl, Tine B., Falch, Erik, Krogsgaard-Larsen, Povl

“…We have previously shown that ( RS)-2-amino-3-(3-hydroxy-5-phenylisoxazol-4-yl)propionic acid (APPA, 2) is a functional partial agonist at the (…”
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FUNCTIONAL PARTIAL AGONISM AT IONOTROPIC EXCITATORY AMINO ACID RECEPTORS by EBERT, BJARKE, MADSEN, ULF, SØBY, KARINA K., KROGSGAARD-LARSEN, POVL

“…( RS)-2-Amino-3-(3-hydroxy-5-phenyl-4-isoxazolyl)propionic acid (APPA), which is an analogue of ( RS)-2-amino-3-(3-hydroxy-5-methyl-4-isoxazolyl)propionic acid…”
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