Search Results - "Ryabova, Olga B"

Towards a new combination therapy for tuberculosis with next generation benzothiazinones by Makarov, Vadim, Lechartier, Benoit, Zhang, Ming, Neres, João, van der Sar, Astrid M, Raadsen, Susanne A, Hartkoorn, Ruben C, Ryabova, Olga B, Vocat, Anthony, Decosterd, Laurent A, Widmer, Nicolas, Buclin, Thierry, Bitter, Wilbert, Andries, Koen, Pojer, Florence, Dyson, Paul J, Cole, Stewart T

“…The benzothiazinone lead compound, BTZ043, kills Mycobacterium tuberculosis by inhibiting the essential flavo‐enzyme DprE1, decaprenylphosphoryl‐beta‐D‐ribose…”
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Finding of the low molecular weight inhibitors of resuscitation promoting factor enzymatic and resuscitation activity by Demina, Galina R, Makarov, Vadim A, Nikitushkin, Vadim D, Ryabova, Olga B, Vostroknutova, Galina N, Salina, Elena G, Shleeva, Margarita O, Goncharenko, Anna V, Kaprelyants, Arseny S

“…Resuscitation promoting factors (RPF) are secreted proteins involved in reactivation of dormant actinobacteria, including Mycobacterium tuberculosis. They have…”
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The 8-Pyrrole-Benzothiazinones Are Noncovalent Inhibitors of DprE1 from Mycobacterium tuberculosis by Makarov, Vadim, Neres, João, Hartkoorn, Ruben C, Ryabova, Olga B, Kazakova, Elena, Šarkan, Michal, Huszár, Stanislav, Piton, Jérémie, Kolly, Gaëlle S, Vocat, Anthony, Conroy, Trent M, Mikušová, Katarína, Cole, Stewart T

“…8-Nitro-benzothiazinones (BTZs), such as BTZ043 and PBTZ169, inhibit decaprenylphosphoryl-β-d-ribose 2'-oxidase (DprE1) and display nanomolar bactericidal…”
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Mechanism of action of 5-nitrothiophenes against Mycobacterium tuberculosis by Hartkoorn, Ruben C, Ryabova, Olga B, Chiarelli, Laurent R, Riccardi, Giovanna, Makarov, Vadim, Cole, Stewart T

“…On using the streptomycin-starved 18b strain as a model for nonreplicating Mycobacterium tuberculosis, we identified a 5-nitrothiophene compound as highly…”
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Structural characterization of prazosin hydrochloride and prazosin free base by Chernyshev, Vladimir V, Stephens, Peter W, Yatsenko, Alexandr V, Ryabova, Olga B, Makarov, Vadim A

“…The three-dimensional solid-state structures of prazosin hydrochloride, C19H22N5O4+.Cl- (A), and prazosin free base, C19H21N5O4 (B), have been determined by…”
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Mechanism of Action of 5-Nitrothiophenes against Mycobacterium tuberculosis by HARTKOORN, Ruben C, RYABOVA, Olga B, CHIARELLI, Laurent R, RICCARDI, Giovanna, MAKAROV, Vadim, COLE, Stewart T

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