Search Results - "Ruchko, E A"

Synthesis and biological properties of novel structural analogs of isothiobarbamine by Novakov, I. A., Sheikin, D. S., Ruchko, E. A., Brunilina, L. L., Vernigora, A. A., Salykin, N. A., Vostrikova, O. V., Chapurkin, V. V., Nawrozkij, M. B., Kurkin, D. V., Bakulin, D. A., Vorontsov, M. Yu, Sablina, L. A., Kovalev, N. S., Tyurenkov, I. N.

“…Novel structural analogs of isothiobarbamine, which differ from the prototype scaffold by the substituent at position 2 of the pyrimidine heterocycle, were for…”
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Pentapeptide analogs of somatostatin containing a thiazolidine fragment: synthesis and cytotoxic activity by Balaev, A. N., Osipov, V. N., Okhmanovich, K. A., Ruchko, E. A., Baryshnikova, M. A., Khachatryan, D. S.

“…Pentapeptide analogs of somatostatin containing an ( R )-1,3-thiazolidine fragment (Thz) of the general formula X—Thz—Phe—D-Trp—Lys(Y)—Thr—Z were synthesized…”
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Synthesis and cytotoxic activity of Boc-protected pentapeptide amide analogs of somatostatin by Balaev, A. N., Osipov, V. N., Okhmanovich, K. A., Ruchko, E. A., Kolotaev, A. V., Khachatryan, D. S.

“…New Boc-protected pentapeptide amides of the general formula Boc—Cys(Boc)—Phe— d -Trp—Lys(Boc)—Thr—NHR, which are analogs of the natural hormone somatostatin,…”
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Aminolysis of 6-[1-(2,6-difluorophenyl)cyclopropyl]-5-methyl-2-(nitroamino)pyrimidin-4(3H)-one by Novakov, I. A., Brunilina, L. L., Vernigora, A. A., Kirillov, I. A., Mkrtchyan, A. S., Navrotskii, M. B., Sheikin, D. S., Yablokov, A. S., Ruchko, E. A., Kachala, V. V.

“…The aminolysis of 6-[1-(2,6-difluorophenyl)cyclopropyl]-5-methyl-2-(nitroamino)pyrimidin-4(3 H )-one with various amines in butan-1-ol and under solvent-free…”
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Reactions of indolylmagnesium bromide with trans-2-phenylcyclopropane-1-carbonyl chloride by Babushkin, A. S., Brunilina, L. L., Navrotskii, M. B., Ruchko, E. A., Kachala, V. V.

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Synthesis of 3-oxoesters and functional derivatives of pyrimidin-4(3Н)-one based on 1-(2,6-dihalophenyl)cyclopropan-1-carboxylic acids by Novakov, I. A., Yablokov, A. S., Navrotskii, M. B., Mkrtchyan, A. S., Vernigora, A. A., Babushkin, A. S., Kachala, V. V., Ruchko, E. A.

“…Special features of the synthesis and chemical transformations of novel functional derivatives of 6-[1-(2,6-dihalophenyl)cyclopropyl]pyrimidin-4(3 H )-one and…”
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Structural Analogs of Umifenovir. 1. Synthesis and Biological Activity of Ethyl 5-Hydroxy-1-Methyl-2-(Trans-2-Phenylcyclopropyl)-1H-Indole-3-Carboxylate by Balzarini, J., Ruchko, E. A., Zakharova, E. K., Kameneva, I. Yu, Nawrozkij, M. B.

“…Ethyl 5-hydroxy-1-methyl-2-(trans-2-phenylcyclopropyl)-1H-indole-3-carboxylate is the first prototype of conformationally restricted analogs of umifenovir. It…”
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Specific features of amidoalkylation of 6-hydroxy-5-isopropyl-2-thioxo-2,3-dihydropyrimidin-4(1H)-one by Novakov, I. A., Sheikin, D. S., Chapurkin, V. V., Nawrozkij, M. B., Kirillov, I. A., Ruchko, E. A.

“…During the synthesis of new structural analogs of isothiobarbamine, the amidoalkylation of 6-hydroxy-5-isopropyl-2-thioxo-2,3-dihydropyrimidin-4(1 H )-one was…”
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Some Features of the Tscherniac‒Einhorn Reaction with 2-Thiouracil Derivatives by Novakov, I. A., Sheikin, D. S., Chapurkin, V. V., Navrotskii, M. B., Babushkin, A. S., Ruchko, E. A., Maryshev, A. Yu, Schols, D.

“…The Tscherniac–Einhorn reaction of 6-methyl and 6-(trifluoromethyl) derivatives of 2-thiouracil with N -(bromomethyl)phthalimide in under basic catalysis leads…”
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Some Features of the TscherniacâEinhorn Reaction with 2-Thiouracil Derivatives by Novakov, I. A, Sheikin, D. S, Chapurkin, V. V, Navrotskii, M. B, Babushkin, A. S, Ruchko, E. A, Maryshev, A. Yu

“…The Tscherniac-Einhorn reaction of 6-methyl and 6-(trifluoromethyl)derivatives of 2-thiouracil with N-(bromomethyl)phthalimide in under basic catalysis leads…”
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Some Features of the Tscherniac‒Einhorn Reaction with2-Thiouracil Derivatives by Novakov, I A, Sheikin, D S, Chapurkin, V V, Navrotskii, M B, Babushkin, A S, Ruchko, E A, Yu, Maryshev A, Schols, D

“…The Tscherniac–Einhorn reaction of 6-methyl and 6-(trifluoromethyl) derivatives of 2-thiouracil with N-(bromomethyl)phthalimide in under basic catalysis leads…”
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Experimental and quantum chemical study of the reactions of 2-methyloxirane with 5-alkyl-6-(2,6-dihalobenzyl)-2-thioxo1,2-dihydropyrimidine-4(3H)-one derivatives by Yablokov, A. S., Steglenko, D. V., Ruchko, E. A., Nawrozkij, M. B., Brunilina, L. L., Novakov, I. A., Minkin, V. I.

“…The reactions of 5-alkyl-6-(2,6-dihalobenzyl)-2-thioxo-1,2-dihydropyrimidin-4(3 H )-one with 2-methyloxirane in an alkaline medium afforded uracil and…”
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Structural Analogs of Umifenovir. 1. Synthesis and Biological Activity of Ethyl 5-Hydroxy-1-Methyl-2-( Trans -2-Phenylcyclopropyl)-1 H -Indole-3-Carboxylate by Balzarini, J, Ruchko, E A, Zakharova, E K, Kameneva, I Yu, Nawrozkij, M B

“…Ethyl 5-hydroxy-1-methyl-2-(trans-2-phenylcyclopropyl)-1H-indole-3-carboxylate is the first prototype of conformationally restricted analogs of umifenovir. It…”
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Reduction of Camphthotecine by 1,4-dihydropyridine by Ivchenko, A. N., Balaev, A. N., Ruchko, E. A., Fedorov, V. E.

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