Search Results - "Roubert, P"

α1-Adrenoceptors in testosterone-induced prostatic hypertrophy by Auger-Pourmarin, L, Roubert, P, Chabrier, P.E

“…Modifications of rat prostatic α 1-adrenoceptors were investigated in testosterone-induced prostatic hypertrophy. [ 3 H ]prazosin bound to a single class of…”
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Regulation of atrial natriuretic factor receptors by angiotensin II in rat vascular smooth muscle cells by Chabrier, P E, Roubert, P, Lonchampt, M O, Plas, P, Braquet, P

“…Atrial natriuretic factor (ANF) is actively involved in the control of blood pressure and fluid homeostasis as a physiological antagonist of the…”
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Endothelin receptor subtypes A and B are up-regulated in an experimental model of acute renal failure by Roubert, P, Gillard-Roubert, V, Pourmarin, L, Cornet, S, Guilmard, C, Plas, P, Pirotzky, E, Chabrier, P E, Braquet, P

“…The two endothelin (ET) receptor subtypes (ETA and ETB) have been characterized in rat kidney from normal rats and rats with acute renal failure induced by…”
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410 Antitumoral activity of tasquinimod is mediated through tumour immunomodulatory and antiangiogenic properties in bladder cancer by Nakhlé, J, Bauchet, A-L, Pierron, V, Plas, P, Thiongane, A, Renauleaud, C, Roubert, P, Navarrete, Ruiz A.M, Schmidlin, F

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Specific Binding of Atrial Natriuretic Factor in Brain Microvessels by Chabrier, Pierre E., Roubert, Pierre, Braquet, Pierre

“…Cerebral capillaries constitute the blood--brain barrier. Studies of specific receptors (neurotransmitters or hormones) located on this structure can be…”
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Down-regulation of atrial natriuretic factor receptors and correlation with cGMP stimulation in rat cultured vascular smooth muscle cells by Roubert, P, Lonchampt, M O, Chabrier, P E, Plas, P, Goulin, J, Braquet, P

“…The relationship between the binding of 125I-labeled rat ANF and the responsiveness in cGMP production of ANF receptors were examined in cultured rat thoracic…”
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Down-regulation of endothelin binding sites in rat vascular smooth muscle cells by Roubert, P, Gillard, V, Plas, P, Chabrier, P E, Braquet, P

“…In cultured rat aortic smooth muscle cells, [125I]endothelin (ET-1) bound to an apparent single class of high affinity recognition sites with a dissociation…”
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Upregulation of renal endothelin receptors in glycerol-induced acute renal failure in the rat by Roubert, P, Cornet, S, Plas, P, Guilmard, C, Pirotzky, E, Chabrier, P E, Braquet, P

“…Acute renal failure was induced in rat with a hypertonic glycerol solution and endothelin-1 (ET-1) binding was measured in kidney membrane preparations. In…”
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Binding characteristics of endothelin isoforms (ET-1, ET-2, and ET-3) in vascular smooth muscle cells by Roubert, P, Gillard, V, Plas, P, Chabrier, P E, Braquet, P

“…The existence of distinct endothelin (ET) receptor subtypes has been reported in several tissues. In the present study, we investigated the binding…”
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Blood-brain barrier and atrial natriuretic factor by Chabrier, P E, Roubert, P, Plas, P, Braquet, P

“…In brain, binding sites for atrial natriuretic factor (ANF) have been characterized in areas such as circumventricular organs that lack the tight capillary…”
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Identification of potent non-peptide somatostatin antagonists with sst(3) selectivity by Poitout, L, Roubert, P, Contour-Galcéra, M O, Moinet, C, Lannoy, J, Pommier, J, Plas, P, Bigg, D, Thurieau, C

“…Using a solution-phase parallel synthesis strategy, a series of non-peptide somatostatin analogues were prepared, and their binding affinities to the five…”
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Identification of Potent Non-Peptide Somatostatin Antagonists with sst3 Selectivity by Poitout, Lydie, Roubert, Pierre, Contour-Galcéra, Marie-Odile, Moinet, Christophe, Lannoy, Jacques, Pommier, Jacques, Plas, Pascale, Bigg, Dennis, Thurieau, Christophe

“…Using a solution-phase parallel synthesis strategy, a series of non-peptide somatostatin analogues were prepared, and their binding affinities to the five…”
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Cross-desensitization between angiotensin II and endothelin-1 in the pithed rat by Guillon, J M, Etiemble, E, Roubert, P, Auguet, M, Chabrier, P E, Braquet, P

“…It has been shown that in vitro angiotensin II (Ang II) potently downregulates endothelin-1 (ET-1) binding sites. In this study, we investigated in vivo the…”
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Vascular mechanism of action of endothelin-1: effect of Ca2+ antagonists by Chabrier, P E, Auguet, M, Roubert, P, Lonchampt, M O, Gillard, V, Guillon, J M, Delaflotte, S, Braquet, P

“…The vasoconstrictive properties of the endothelium-derived peptide, endothelin-1 (ET-1), were investigated on rat isolated aorta and on cultured rat aortic…”
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Des agonistes du récepteur de type 4 aux mélanocortines permettent de corriger in vitro le défaut d’activation induit par des mutations associées à l’obésité humaine by Dubern, B., Roubert, P., Plas, P., Lubrano-Berthelier, C., Alihi, R., Auger, F., DeOliveira, D.B., Dong, J.Z., Basdevant, A., Thurieau, C., Clément, K.

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Effects and specific binding sites of endothelin in human lung preparations by Brink, C, Gillard, V, Roubert, P, Mencia-Huerta, J M, Chabrier, P E, Braquet, P, Verley, J

“…Endothelin binding in human isolated lung membrane fractions revealed a single class of high affinity recognition sites with a Kd of 1.33 +/- 0.15 nM and a…”
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Comparison of the bronchopulmonary and pressor activities of endothelin isoforms ET-1, ET-2, and ET-3 and characterization of their binding sites in guinea pig lung by Pons, F, Loquet, I, Touvay, C, Roubert, P, Chabrier, P E, Mencia-Huerta, J M, Braquet, P

“…In anesthetized and ventilated guinea pigs intravenous injection of ET-1, ET-2, or ET-3 (1 or 2 nmol/kg) induced similar dose-dependent increases in pulmonary…”
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Receptor regulation of atrial natriuretic factor by Chabrier, P E, Roubert, P, Lonchampt, M O, Plas, P, Braquet, P

“…Two atrial natriuretic factor (ANF) receptor subtypes are present in vascular smooth muscle cells: the B receptors (or biologically active) coupled to a…”
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Endothelin-secreting angiosarcoma occurring at the site of an arteriovenous fistula for haemodialysis in a renal transplant recipient by Bessis, D, Sotto, A, Roubert, P, Chabrier, P E, Mourad, G, Guilhou, J J

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Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5 by Contour-Galcéra, Marie-Odile, Poitout, Lydie, Moinet, Christophe, Morgan, Barry, Gordon, Tom, Roubert, Pierre, Thurieau, Christophe

“…A new preparation of trisubstituted imidazopyrazines and dihydroimidazopyrazines via parallel synthesis using aminoacids and bromoketones resulted in the…”
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