Search Results - "Riyadh, Sayed M."
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Clean Grinding Technique: A Facile Synthesis and In Silico Antiviral Activity of Hydrazones, Pyrazoles, and Pyrazines Bearing Thiazole Moiety against SARS-CoV-2 Main Protease (M pro )
Published in Molecules (Basel, Switzerland) (06-10-2020)“…A novel series of some hydrazones bearing thiazole moiety were generated via solvent-drop grinding of thiazole carbohydrazide with various carbonyl compounds…”
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Enaminones as building blocks for the synthesis of substituted pyrazoles with antitumor and antimicrobial activities
Published in Molecules (Basel, Switzerland) (22-02-2011)“…Novel N-arylpyrazole-containing enaminones 2a,b were synthesized as key intermediates. Reactions of 2a,b with active methylene compounds in acetic acid in the…”
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Synthesis, Molecular Docking Study, and Cytotoxic Activity against MCF Cells of New Thiazole–Thiophene Scaffolds
Published in Molecules (Basel, Switzerland) (20-07-2022)“…Investigating novel compounds that may be useful in designing new, less toxic, selective, and potent breast anticancer agents is still the main challenge for…”
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Synthesis under microwave irradiation of [1,2,4]triazolo[3,4-b] [1,3,4]thiadiazoles and other diazoles bearing indole moieties and their antimicrobial evaluation
Published in Molecules (Basel, Switzerland) (28-09-2011)“…Microwave-assisted synthesis of some novel compounds, namely, 3-(2-methyl-1H-indol-3-yl)-6-aryl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles 5a,b was accomplished…”
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A Literature Review Focusing on the Antiviral Activity of [1,2,4] and [1,2,3]-triazoles
Published in Mini reviews in medicinal chemistry (01-01-2024)“…Out of a variety of heterocycles, triazole scaffolds have been shown to play a significant part in a wide array of biological functions. Many drug compounds…”
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Synthesis of Chitosan-La2O3 Nanocomposite and Its Utility as a Powerful Catalyst in the Synthesis of Pyridines and Pyrazoles
Published in Molecules (Basel, Switzerland) (17-06-2021)“…Recently, the development of nanocatalysts based on naturally occurring polysaccharides has received a lot of attention. Chitosan (CS), as a biodegradable and…”
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Potential COVID-19 Drug Candidates Based on Diazinyl-Thiazol-Imine Moieties: Synthesis and Greener Pastures Biological Study
Published in Molecules (Basel, Switzerland) (13-01-2022)“…A novel series of 1-aryl- -[4-phenyl-5-(arylazo)thiazol-2-yl)methanimines has been synthesized via the condensation of 2-amino-4-phenyl-5-arylazothiazole with…”
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Bio-Based (Chitosan-ZnO) Nanocomposite: Synthesis, Characterization, and Its Use as Recyclable, Ecofriendly Biocatalyst for Synthesis of Thiazoles Tethered Azo Groups
Published in Polymers (19-01-2022)“…In recent years, nanotechnology has become a considerable research interest in the area of preparation of nanocatalysts based on naturally occurring…”
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Synthesis and greener pastures biological study of bis-thiadiazoles as potential Covid-19 drug candidates
Published in Arabian journal of chemistry (01-09-2022)“…A novel series of bis- (Abdelhamid et al., 2017; Banerjee et al., 2018; Bharanidharan et al., 2022)thiadiazoles was synthesized from the reaction of precursor…”
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Chitosan-Strontium Oxide Nanocomposite: Preparation, Characterization, and Catalytic Potency in Thiadiazoles Synthesis
Published in Polymers (12-07-2022)“…Recently, Strontium oxide (SrO) nanoparticles (NPs) and hybrids outperformed older commercial catalysts in terms of catalytic performance. Herein, we present a…”
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Synthesis, DPPH Radical Scavenging, Cytotoxic Activity, and Apoptosis Induction Efficacy of Novel Thiazoles and Bis-thiazoles
Published in Current organic synthesis (01-01-2024)“…Heterocyclic materials-containing thiazoles exhibited incredible importance in pharmaceutical chemistry and drug design due to their extensive biological…”
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Structural Properties and Catalytic Activity of Binary Poly (vinyl alcohol)/Al2O3 Nanocomposite Film for Synthesis of Thiazoles
Published in Catalysts (01-01-2020)“…A solution casting technique was applied to prepare a binary poly (vinyl alcohol)/Al2O3 nanocomposite. The structural properties of nanocomposite were…”
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Chitosan-MgO Nanocomposite: One Pot Preparation and Its Utility as an Ecofriendly Biocatalyst in the Synthesis of Thiazoles and [1,3,4]thiadiazoles
Published in Nanomaterials (Basel, Switzerland) (08-11-2018)“…A chitosan-MgO hybrid nanocomposite was prepared using a simple chemical precipitation method and characterized using Fourier transform spectroscopy (FTIR),…”
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Green Synthetic Approaches of 2-Hydrazonothiazol-4(5H)-ones Using Sustainable Barium Oxide-Chitosan Nanocomposite Catalyst
Published in Polymers (01-09-2023)“…The diverse applications of metal oxide-biopolymer matrix as a nanocomposite heterogenous catalyst have caused many researches to scrutinize the potential of…”
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Investigation of inhibition efficiencies of Novel bis-oxindole and bis(spiro(triazole-oxindole)) for the corrosion of copper in sulfuric acid medium
Published in Polycyclic aromatic compounds (07-02-2024)“…The condensation reaction of bis-oxindole with aniline derivatives produced three derivatives of…”
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Synthesis and In Silico Study of Some New bis -[1,3,4]thiadiazolimines and bis -Thiazolimines as Potential Inhibitors for SARS-CoV-2 Main Protease
Published in Current issues in molecular biology (30-09-2022)“…A novel series of -[1,3,4]thiadiazolimines, and -thiazolimines, with alkyl linker, were synthesized through general routes from cyclization of…”
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Effect of solvent on the regioselective synthesis of spiropyrazoles
Published in Tetrahedron (04-11-2012)“…1,3-Dipolarcycloaddition reactions of 6-arylmethylene-6,7,8,9-tetrahydro-5H-benzocyclohepten-5-ones (1) with nitrilimines 3 were investigated in benzene and…”
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Green Route Synthesis and Molecular Docking of Azines Using Cellulose Sulfuric Acid under Microwave Irradiation
Published in Crystals (Basel) (01-02-2023)“…A novel catalytic approach for the synthesis of symmetric and asymmetric azines has been developed. The environmentally benign protocol was achieved via…”
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Synthesis, Biological Evaluation, and Molecular Docking of Novel Azolylhydrazonothiazoles as Potential Anticancer Agents
Published in ACS omega (19-09-2023)“…A novel set of thiazolylhydrazonothiazoles bearing an indole moiety were synthesized by subjection reactions of carbothioamide derivative and hydrazonoyl…”
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