Search Results - "Rival, Y"

An innovative method to quantitate tissue integration of hyaluronic acid-based dermal fillers by Dugaret, A S, Bertino, B, Gauthier, B, Gamboa, B, Motte, M, Rival, Y, Piwnica, D, Osman-Ponchet, H, Bourdès, V, Voegel, J J

“…Following intradermal injection, hyaluronic acid (HA)-based fillers tend to spread within the reticular dermis and to distribute between the dermal fibers…”
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Design, Synthesis, and Structure−Activity Relationships of a Series of 3-[2-(1-Benzylpiperidin-4-yl)ethylamino]pyridazine Derivatives as Acetylcholinesterase Inhibitors by Contreras, Jean-Marie, Parrot, Isabelle, Sippl, Wolfgang, Rival, Yveline M, Wermuth, Camille G

“…Starting from the 3-[2-(1-benzylpiperidin-4-yl)ethylamino]-6-phenylpyridazine 1, we performed the design, the synthesis, and the structure−activity…”
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Aminopyridazines as Acetylcholinesterase Inhibitors by Contreras, Jean-Marie, Rival, Yveline M, Chayer, Said, Bourguignon, Jean-Jacques, Wermuth, Camille G

“…Following the discovery of the weak, competitive and reversible acetylcholinesterase (AChE)-inhibiting activity of minaprine (3c) (IC50 = 85 μM on homogenized…”
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Polymorphonuclear Leukocyte Adhesion Triggers the Disorganization of Endothelial Cell-to-Cell Adherens Junctions by Del Maschio, Aldo, Zanetti, Adriana, Corada, Monica, Rival, Yves, Ruco, Luigi, Lampugnani, Maria Grazia, Dejana, Elisabetta

“…Polymorphonuclear leukocytes (PMN) infiltration into tissues is frequently accompanied by increase in vascular permeability. This suggests that PMN adhesion…”
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Synthesis and Antibacterial Activity of Some Imidazo [1, 2-α]pyrimidine Derivatives by RIVAL, Yveline, GRASSY, Gerard, MICHEL, Georges

“…A series of 75 imidazo[1, 2-α]pyrimidine derivatives were synthesized. The "in vitro" antibacterial activity of these compounds and their corresponding…”
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Inhibition of platelet endothelial cell adhesion molecule-1 synthesis and leukocyte transmigration in endothelial cells by the combined action of TNF-alpha and IFN-gamma by Rival, Y, Del Maschio, A, Rabiet, MJ, Dejana, E, Duperray, A

“…Endothelial cell (EC) junctions regulate circulating leukocyte extravasation and infiltration at inflammatory sites. Several lines of evidence show that…”
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Structure-based 3D QSAR and design of novel acetylcholinesterase inhibitors by Sippl, W, Contreras, J M, Parrot, I, Rival, Y M, Wermuth, C G

“…The paper describes the construction, validation and application of a structure-based 3D QSAR model of novel acetylcholinesterase (AChE) inhibitors. Initial…”
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W01.120 Regulation of the human $alpha;P2 promoter by PPAR modulators with various lipogenic properties by RIVAL, Y

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556 PERMIXON INHIBITS CYTOKINE-INDUCED EXPRESSION OF VCAM-1, ESSENTIAL FOR MONONUCLEAR CELL ADHESION ON HUMAN VASCULAR ENDOTHELIAL CELLS by Rival, Y, Taillandier, T, Lantoine-Adam, F, Templier, M, Junquero, D

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Evidence for a selective inhibitory effect of thrombin on megakaryocyte progenitor growth mediated by the thrombin receptor by Plantier, J L, Berthier, R, Rival, Y, Schweitzer, A, Rabiet, M J

“…An efficient method for the culture of human megakaryocyte precursors in serum-free medium has been developed facilitating study of the effect of regulators of…”
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Synthesis and antifungal activity evaluation of 3-hydroxyimidazo[1,2-a]pyridine and 3-hydroxyimidazo[1,2-a]pyrimidine derivatives by Rival, Y, Taudou, A, Ecalle, R

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PPARα and PPARδ activators inhibit cytokine-induced nuclear translocation of NF-κB and expression of VCAM-1 in EAhy926 endothelial cells by Rival, Yves, Benéteau, Nathalie, Taillandier, Thierry, Pezet, Mylène, Dupont-Passelaigue, Elisabeth, Patoiseau, Jean-François, Junquéro, Didier, Colpaert, Francis C., Delhon, André

“…Endothelium injury is a primary event in atherogenesis, which is followed by monocyte infiltration, macrophage differentiation, and smooth muscle cell…”
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Thrombin-induced increase in endothelial permeability is associated with changes in cell-to-cell junction organization by RABIET, M.-J, PLANTIER, J.-L, RIVAL, Y, GENOUX, Y, LAMPUGNANI, M.-G, DEJANA, E

“…Thrombin increases endothelial permeability in a rapid and reversible way. This effect requires the catalytic activity of the enzyme and thrombin receptor…”
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Human adipocyte fatty acid-binding protein (aP2) gene promoter-driven reporter assay discriminates nonlipogenic peroxisome proliferator-activated receptor gamma ligands by Rival, Yves, Stennevin, Aline, Puech, Laurence, Rouquette, Anne, Cathala, Claudie, Lestienne, Fabrice, Dupont-Passelaigue, Elisabeth, Patoiseau, Jean-François, Wurch, Thierry, Junquéro, Didier

“…Peroxisome proliferator-activated receptors (PPARs) regulate storage and catabolism of fats and carbohydrates. PPARgamma activity increases insulin sensitivity…”
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Metabolic syndrome: which definition for what treatment(s)? by Junquero, Didier, Rival, Yves

“…Metabolic syndrome is asymptomatic and results from the increasing prevalence of obesity. Although several definitions exist and complicate its diagnosis,…”
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Comparative sensitivity study of Clostridium perfringens towards 16 antibiotics from different classes by Rival, Y, Grassy, G, Simeon de Buochberg, M, Dusart, G

“…A series of 16 antibiotics from different classes (5-nitro imidazoles, beta-lactams, cyclins, macrolids, chloramphenicol) was examined for their bacteriostatic…”
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L’étude du transcriptome des peaux de patients souffrant de vitiligo montre une altération de la voie de WNT et révèle une cible thérapeutique nouvelle pour repigmenter les lésions de vitiligo by Regazzetti, C., Joly, F., Marty, C., Rivier, M., Mehul, B., Reniche, P., Mounier, C., Rival, Y., Piwnica, D., Cavalié, M., Chignon-Sicard, B., Ballotti, R., Voegel, J., Passeron, T.

“…Le vitiligo touche environ 1 % de la population mondiale. Stopper l’évolutivité de la maladie et repigmenter les zones lésionnelles sont les deux challenges…”
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Efficient one-step synthesis of 3-amino-6-arylpyridazines by Guery, Sébastien, Parrot, Isabelle, Rival, Yveline, Wermuth, Camille G

“…Starting from the commercially available 3-amino-6-chloropyridazine, 3-amino-6-arylpyridazines were prepared in good yields by means of a Suzuki cross-coupling…”
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Cardiovascular drugs inhibit MMP-9 activity from human THP-1 macrophages by Rival, Yves, Benéteau, Nathalie, Chapuis, Violaine, Taillandier, Thierry, Lestienne, Fabrice, Dupont-Passelaigue, Elisabeth, Patoiseau, Jean-François, Colpaert, Francis C, Junquéro, Didier

“…It is now recognized that atherosclerosis complications are related to the unstable character of the plaque rather than its volume. Vulnerable plaques often…”
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5-HT3 Antagonists Derived from Aminopyridazine-type Muscarinic M1 Agonists by Rival, Yveline, Hoffmann, Rémy, Didier, Bruno, Rybaltchenko, Volodymyr, Bourguignon, Jean-Jacques, Wermuth, Camille G

“…A conformational analysis, performed on muscarinic M1 agonists, identified four structural features characteristic of the muscarinic M1 pharmacophore:  (i) a…”
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