Search Results - "Riesco, Alejandra"

Continuous Flow Synthesis of Urea‐Containing Compound Libraries Based on the Piperidin‐4‐one Scaffold by Riesco‐Domínguez, Alejandra, Blanco‐Ania, Daniel, Rutjes, Floris P. J. T.

“…The advantages of performing reactions in continuous flow vs. the classic batch processes render flow chemistry a suitable technique for library synthesis…”
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Trifluoromethyl Vinyl Sulfide: A Building Block for the Synthesis of CF3S‑Containing Isoxazolidines by Riesco-Domínguez, Alejandra, van de Wiel, Jeroen, Hamlin, Trevor A, van Beek, Bas, Lindell, Stephen D, Blanco-Ania, Daniel, Bickelhaupt, F. Matthias, Rutjes, Floris P. J. T

“…Trifluoromethyl vinyl sulfide, a potential building block for pharmaceutically and agrochemically relevant products, is prepared and used for the first time in…”
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An Enantio‐ and Diastereoselective Mannich/Pictet–Spengler Sequence To Form Spiro[piperidine‐pyridoindoles] and Application to Library Synthesis by Riesco‐Domínguez, Alejandra, van der Zwaluw, Nick, Blanco‐Ania, Daniel, Rutjes, Floris P. J. T.

“…A new tandem strategy based on a Mannich/Pictet–Spengler sequence has been developed and applied to the synthesis of a new small library (14 examples) of…”
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Exploring the size adaptability of the B ring binding zone of the colchicine site of tubulin with para-nitrogen substituted isocombretastatins by Jiménez, Carmen, Ellahioui, Younes, Álvarez, Raquel, Aramburu, Laura, Riesco, Alejandra, González, Myriam, Vicente, Alba, Dahdouh, Abdelaziz, Ibn Mansour, Ahmed, Jiménez, Carlos, Martín, Diego, Sarmiento, Rogelio G., Medarde, Manuel, Caballero, Esther, Peláez, Rafael

“…We have synthesized and assayed dimethylaminophenyl, pyrrolidin-1-ylphenyl and carbazole containing phenstatins and isocombretastatins as analogues of the…”
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Trifluoromethyl Vinyl Sulfide: A Building Block for the Synthesis of CF 3 S-Containing Isoxazolidines by Riesco-Domínguez, Alejandra, van de Wiel, Jeroen, Hamlin, Trevor A, van Beek, Bas, Lindell, Stephen D, Blanco-Ania, Daniel, Bickelhaupt, F Matthias, Rutjes, Floris P J T

“…Trifluoromethyl vinyl sulfide, a potential building block for pharmaceutically and agrochemically relevant products, is prepared and used for the first time in…”
Get full text