Search Results - "Regina, A. La"

Role of peripheral mu, delta and kappa opioid receptors in opioid-induced inhibition of gastrointestinal transit in rats by Tavani, A, Petrillo, P, La Regina, A, Sbacchi, M

“…The roles of various types of opioid receptors in opioid-induced local inhibition of gastrointestinal transit were studied in rats 5 min after a charcoal meal,…”
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Cefepime Versus Ceftazidime in the Treatment of Lower Respiratory Tract Infections by Aufiero, A., Sturani, C., Zanona, P., Marruchella, A., Michetti, G., Nicolin, E., Sella, D., Goglio, A., Silleni, M., Regina, A. La

“…The objective of the study was to compare the safety and efficacy of cefepime and ceftazidime in the treatment of community acquired lower respiratory tract…”
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Trend in rifampicin-, multidrug- and extensively drug-resistant tuberculosis in Italy, 2009-2016 by Mustazzolu, Alessandro, Borroni, Emanuele, Cirillo, Daniela Maria, Giannoni, Federico, Iacobino, Angelo, Fattorini, Lanfranco

“…Tuberculosis (TB) caused by strains of Mycobacterium tuberculosis that are rifampicin-resistant (RR), multidrug-resistant (MDR) (strains resistant to at least…”
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Tuberculosis in migrants from 106 countries to Italy, 2008-2014 by Fattorini, Lanfranco, Mustazzolu, Alessandro, Borroni, Emanuele, Piccaro, Giovanni, Giannoni, Federico, Cirillo, Daniela Maria

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Design, Molecular Modeling, Synthesis, and Anti-HIV-1 Activity of New Indolyl Aryl Sulfones. Novel Derivatives of the Indole-2-carboxamide by Ragno, Rino, Coluccia, Antonio, La Regina, Giuseppe, De Martino, Gabriella, Piscitelli, Francesco, Lavecchia, Antonio, Novellino, Ettore, Bergamini, Alberto, Ciaprini, Chiara, Sinistro, Anna, Maga, Giovanni, Crespan, Emanuele, Artico, Marino, Silvestri, Romano

“…Molecular modeling studies and an updated highly predictive 3-D QSAR model led to the discovery of exceptionally potent indolyl aryl sulfones (IASs)…”
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Antagonism by N-methyl levallorphan-methane sulphonate (SR 58002 C) of morphine-elicited acute and chronic central and peripheral effects by Sbacchi, M, Colombo, M, La Regina, A, Petrillo, P, Tavani, A

“…The peripheral activity of the quaternary narcotic antagonist N-methyl levallorphan-methane sulphonate (SR 58002 C) at opioid sites located in the periphery…”
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Arylthioindoles, Potent Inhibitors of Tubulin Polymerization by De Martino, Gabriella, La Regina, Giuseppe, Coluccia, Antonio, Edler, Michael C, Barbera, Maria Chiara, Brancale, Andrea, Wilcox, Elizabeth, Hamel, Ernest, Artico, Marino, Silvestri, Romano

“…Several arylthioindoles had excellent activity as inhibitors both of tubulin polymerization and of the growth of MCF-7 human breast carcinoma cells. Methyl…”
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New Pyrrole Inhibitors of Monoamine Oxidase:  Synthesis, Biological Evaluation, and Structural Determinants of MAO-A and MAO-B Selectivity by La Regina, Giuseppe, Silvestri, Romano, Artico, Marino, Lavecchia, Antonio, Novellino, Ettore, Befani, Olivia, Turini, Paola, Agostinelli, Enzo

“…A series of new pyrrole derivatives have been synthesized and evaluated for their monoamine oxidase (MAO) A and B inhibitory activity and selectivity…”
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Synthesis, Cannabinoid Receptor Affinity, and Molecular Modeling Studies of Substituted 1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides by Silvestri, Romano, Cascio, Maria Grazia, La Regina, Giuseppe, Piscitelli, Francesco, Lavecchia, Antonio, Brizzi, Antonella, Pasquini, Serena, Botta, Maurizio, Novellino, Ettore, Di Marzo, Vincenzo, Corelli, Federico

“…The new 1-phenyl-5-(1H-pyrrol-1-yl)pyrazole-3-carboxamides were compared with the reference compounds AM251 and SR144528 for cannabinoid hCB1 and hCB2 receptor…”
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RIPETUTI CLUSTERS DA S. MARCESCENS IN UN REPARTO DI TERAPIA INTENSIVA NEONATALE: ASPETTI MICROBIOLOGICI E CLINICO-EPIDEMIOLOGICI by M. Pecorari, M.G. Tamassia, G. Fabio, N. Nanni, S. Tagliazucchi, E. Della Casa Muttini, G. Leporati, A. La Regina, P. Marchegiano, S. Scaltriti, E. Vecchi, C. Casolari

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Italian multicentre study of didanosine compassionate use in advanced HIV infection by D'ARMINIO MONFORTE, A, MUSICCO, M, MAZZOTTA, F, VISCO, G, AIUTI, F, MORONI, M, GALLI, M, PAGA, C, LA REGINA, A, LAZZARIN, A, ANGARANO, G, MILAZZO, F, GRITTI, F, ARLOTTI, M

“…The aim of the present study, a multicentre trial of didanosine (ddI) compassionate use, was to identify factors associated with a better outcome in patients…”
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D-optimal design applied to binding saturation curves of an enkephalin analog in rat brain by Verotta, D, Petrillo, P, La Regina, A, Rocchetti, M, Tavani, A

“…The D-optimal design, a minimal sample design that minimizes the volume of the joint confidence region for the parameters, was used to evaluate binding…”
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Safety and efficacy of low‐dose fondaparinux (1.5 mg) for the prevention of venous thromboembolism in acutely ill medical patients with renal impairment: the FONDAIR study by AGENO, W., RIVA, N., NORIS, P., DI NISIO, M., LA REGINA, M., ARIOLI, D., RIA, L., MONZANI, V., CUPPINI, S., LUPIA, E., GIORGI PIERFRANCESCHI, M., DENTALI, F.

“…Background:  Renal impairment is common, affecting around 40% of acutely ill medical patients, and is associated with an increased risk of both venous…”
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Development of dopaminergic drugs for the chronic treatment of congestive heart failure by Casagrande, C, Merlo, L, La Regina, A

“…1. The search of orally active dopaminergic drugs for the chronic treatment of congestive heart failure has followed two different approaches. 2. On the one…”
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A ESFINGE, A TEIA E O ENREDO: LETRAMENTO E CAMINHOS DA DEMOCRACIA NO BRASIL by REGINA, ANNE GREICE SOARES LA

“…RESUMO: Este trabalho objetiva analisar as possibilidades do letramento para uma pedagogia cidadã. Parte-se da ideia de Educação como emancipação, associando-a…”
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In vitro binding profile and in vivo pharmacological properties of the K-opioid compound PD 117302 by Colombo, M, Petrillo, P, La Regina, A, Bianchi, G, Tavani, A

“…The in vitro binding profile and some in vivo pharmacological properties of (+/-)trans-N-Methyl-N-[2-(1-pyrrolidinyl)-cyclohexyl]benzo[b]-thiophene-…”
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The role of mu- and delta- opioid receptors on the intestinal propulsion in rats by Sbacchi, M, La Regina, A, Petrillo, P, Tavani, A

“…The agonist effects on intestinal transit of relatively selective mu- and delta- ligands, administered intraperitoneally, and their antagonism by the…”
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Novel 1-[2-(Diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. A Structure−Activity Relationship Investigation by De Martino, Gabriella, La Regina, Giuseppe, Di Pasquali, Alessandra, Ragno, Rino, Bergamini, Alberto, Ciaprini, Chiara, Sinistro, Anna, Maga, Giovanni, Crespan, Emmanuele, Artico, Marino, Silvestri, Romano

“…1-[2-(Diarylmethoxy)ethyl]-2-methyl-5-nitroimidazoles (DAMNIs) is a novel family of HIV-1 non-nucleoside reverse transcriptase inhibitors (NNRTIs) active at…”
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Simple, Short Peptide Derivatives of a Sulfonylindolecarboxamide (L-737,126) Active in Vitro against HIV-1 Wild Type and Variants Carrying Non-Nucleoside Reverse Transcriptase Inhibitor Resistance Mutations by Silvestri, Romano, Artico, Marino, De Martino, Gabriella, La Regina, Giuseppe, Loddo, Roberta, La Colla, Massimiliano, La Colla, Paolo

“…Non-nucleoside reverse transcriptase inhibitors (NNRTIs) active against NNRTI-resistant mutants were obtained by introducing two methyl groups at positions 3…”
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Novel Indolyl Aryl Sulfones Active against HIV-1 Carrying NNRTI Resistance Mutations:  Synthesis and SAR Studies by Silvestri, Romano, De Martino, Gabriella, La Regina, Giuseppe, Artico, Marino, Massa, Silvio, Vargiu, Laura, Mura, Massimo, Loi, Anna Giulia, Marceddu, Tiziana, La Colla, Paolo

“…The potent anti-HIV-1 activities of L-737,126 (2) and PAS sulfones prompted us to design and test against HIV-1 in acutely infected MT-4 cells a number of…”
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