Search Results - "ROETZ, Ralf"

Design of Annulated Pyrazoles as Inhibitors of HIV-1 Reverse Transcriptase by Sweeney, Zachary K, Harris, Seth F, Arora, Nidhi, Javanbakht, Hassan, Li, Yu, Fretland, Jennifer, Davidson, James P, Billedeau, J. Roland, Gleason, Shelley K, Hirschfeld, Donald, Kennedy-Smith, Joshua J, Mirzadegan, Taraneh, Roetz, Ralf, Smith, Mark, Sperry, Sarah, Suh, Judy M, Wu, Jeffrey, Tsing, Stan, Villaseñor, Armando G, Paul, Amber, Su, Guoping, Heilek, Gabrielle, Hang, Julie Q, Zhou, Amy S, Jernelius, Jesper A, Zhang, Fang-Jie, Klumpp, Klaus

“…Non-nucleoside reverse transcriptase inhibitors (NNRTIs) are recommended components of preferred combination antiretroviral therapies used for the treatment of…”
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2-Substituted N-aryl piperazines as novel triple reuptake inhibitors for the treatment of depression by Carter, David S., Cai, Hai-Ying, Lee, Eun Kyung, Iyer, Pravin S., Lucas, Matthew C., Roetz, Ralf, Schoenfeld, Ryan C., Weikert, Robert J.

“…The discovery and optimization of a novel series of 2-substituted N-aryl piperazine based triple reuptake inhibitors is described. Recently a class of…”
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Novel 3,3-disubstituted pyrrolidines as selective triple serotonin/norepinephrine/dopamine reuptake inhibitors by BANNWART, Linda M, CARTER, David S, LYNCH, Stephen M, MADERA, Ann Marie, MOORE, Amy, OZBOYA, Kerem, RAPTOVA, Lubica, ROETZ, Ralf, SCHOENFELD, Ryan C, STEIN, Karin Ann, STEINER, Sandra, VILLA, Marzia, CAI, Hai-Ying, WEIKERT, Robert J, YANSHENG ZHAI, CHOY, Jason C, GREENHOUSE, Robert, JAIME-FIGUEROA, Saul, LYER, Pravin S, LIN, Clara J, EUN KYUNG LEE, LUCAS, Matthew C

“…A series of 3,3-disubstituted pyrrolidine monoamine triple reuptake inhibitors were discovered. Analogues with low nanomolar potency, good human in vitro…”
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Diphenyl Ether Non-Nucleoside Reverse Transcriptase Inhibitors with Excellent Potency Against Resistant Mutant Viruses and Promising Pharmacokinetic Properties by Sweeney, Zachary K., Kennedy-Smith, Joshua J., Wu, Jeffrey, Arora, Nidhi, Billedeau, J. Roland, Davidson, James P., Fretland, Jennifer, Hang, Julie Q., Heilek, Gabrielle M., Harris, Seth F., Hirschfeld, Donald, Inbar, Petra, Javanbakht, Hassan, Jernelius, Jesper A., Jin, Qingwu, Li, Yu, Liang, Weiling, Roetz, Ralf, Sarma, Keshab, Smith, Mark, Stefanidis, Dimitrio, Su, Guoping, Suh, Judy M., Villaseñor, Armando G., Welch, Michael, Zhang, Fang-Jie, Klumpp, Klaus

“…Non‐nucleoside reverse transcriptase inhibitors (NNRTIs) are part of the preferred treatment regimens for individuals infected with HIV. These NNRTI‐based…”
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Diphenyl Ether Non-Nucleoside Reverse Transcriptase Inhibitors with Excellent Potency Against Resistant Mutant Viruses and Promising Pharmacokinetic Properties (ChemMedChem 1/2009) by Sweeney, Zachary K, Kennedy-Smith, Joshua J, Wu, Jeffrey, Arora, Nidhi, Billedeau, J Roland, Davidson, James P, Fretland, Jennifer, Hang, Julie Q, Heilek, Gabrielle M, Harris, Seth F, Hirschfeld, Donald, Inbar, Petra, Javanbakht, Hassan, Jernelius, Jesper A, Jin, Qingwu, Li, Yu, Liang, Weiling, Roetz, Ralf, Sarma, Keshab, Smith, Mark, Stefanidis, Dimitrio, Su, Guoping, Suh, Judy M, Villasenor, Armando G, Welch, Michael, Zhang, Fang-Jie, Klumpp, Klaus

“…The cover picture shows a cut-away view of a diaryl ether non-nucleoside reverse transcriptase inhibitor (cyan) bound to HIV reverse transcriptase. The cartoon…”
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Cover Picture: Diphenyl Ether Non-Nucleoside Reverse Transcriptase Inhibitors with Excellent Potency Against Resistant Mutant Viruses and Promising Pharmacokinetic Properties (ChemMedChem 1/2009) by Sweeney, Zachary K., Kennedy-Smith, Joshua J., Wu, Jeffrey, Arora, Nidhi, Billedeau, J. Roland, Davidson, James P., Fretland, Jennifer, Hang, Julie Q., Heilek, Gabrielle M., Harris, Seth F., Hirschfeld, Donald, Inbar, Petra, Javanbakht, Hassan, Jernelius, Jesper A., Jin, Qingwu, Li, Yu, Liang, Weiling, Roetz, Ralf, Sarma, Keshab, Smith, Mark, Stefanidis, Dimitrio, Su, Guoping, Suh, Judy M., Villaseñor, Armando G., Welch, Michael, Zhang, Fang-Jie, Klumpp, Klaus

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