Search Results - "RAO, A. Raghuram"

Synthesis, anti-inflammatory evaluation and docking studies of some new fluorinated fused quinazolines by Balakumar, C., Lamba, P., Pran Kishore, D., Lakshmi Narayana, B., Venkat Rao, K., Rajwinder, K., Raghuram Rao, A., Shireesha, B., Narsaiah, B.

“…A series of novel 8/10-trifluoromethyl-substituted-imidazo[1,2- c] quinazolines have been synthesized and evaluated in vivo (rat paw edema) for their…”
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Facile Methods for the Synthesis of 5-Aryl and 5-Iodo Pyrrolo[2,3-d]pyrimidines by Venkata Rao, K., Raghu Prasad, M., Raghuram Rao, A.

“…An efficient and environmentally benign one‐pot method has been developed for the synthesis of 4‐amino‐5‐arylpyrrolo[2,3‐d]pyrimidines. Phthalimido…”
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Synthesis and theoretical studies on energetics of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines – Their potential as adenosine receptor ligands by Sirisha, B., Narsaiah, B., Yakaiah, T., Gayatri, G., Sastry, G. Narahari, Prasad, M. Raghu, Rao, A. Raghuram

“…A series of novel N- and O- perfluoroalkyl triazole tagged thienopyrimidines 6a– c and 7a– d was synthesized in two steps from thienopyrimidin-4-ones 2 through…”
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Transesterification of trimethyl orthoacetate: an efficient protocol for the synthesis of 4-alkoxy-2-aminothiophene-3-carbonitriles by Venkata Rao, K., Balakumar, C., Lakshmi Narayana, B., Pran Kishore, D., Rajwinder, K., Raghuram Rao, A.

“…A facile one-pot method is reported for the synthesis of 4-alkoxy-2-aminothiophene-3-carbonitriles. Transesterification of trimethylorthoacetate technique…”
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QSAR study on pyridinone derivatives as HIV-1 non-nucleoside reverse transcriptase inhibitor: a mixed approach by Vasanthanathan, P, Lakshmi, M, Rao, A Raghuram

“…HIV-1 reverse transcriptase inhibitory activity of a series of substituted pyridinone derivatives (non-nucleoside) was subjected to classical QSAR study by…”
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QSAR of adenosine receptor antagonists: Exploring physicochemical requirements for binding of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives with human adenosine A(3) receptor subtype by Pran Kishore, D, Balakumar, C, Raghuram Rao, A, Roy, Partha Pratim, Roy, Kunal

“…Human adenosine A(3) receptor (A(3) AR) binding affinity of pyrazolotriazolopyrimidine derivatives (n=116) has been subjected to QSAR analyses using…”
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Liquid-Chromatographic Separation and Determination of Process-related Impurities, Including a Regio-Specific Isomer of Celecoxib on Reversed-Phase C18 Column Dynamically Coated with Hexamethyldisilazane by RAO, R. Nageswara, MEENA, S., NAGARAJU, D., RAO, A. Raghuram, RAVIKANTH, S.

“…A simple and rapid reversed-phase high-performance liquid-chromatographic method for the separation and determination of process-related impurities of…”
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An overview of the recent developments in analytical methodologies for determination of COX-2 inhibitors in bulk drugs, pharmaceuticals and biological matrices by Nageswara Rao, R., Meena, S., Raghuram Rao, A.

“…An extensive survey of the literature published in various analytical and pharmaceutical chemistry related journals has been conducted and the instrumental…”
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QSAR of adenosine receptor antagonists: Exploring physicochemical requirements for binding of pyrazolo[4,3-e]-1,2,4-triazolo[1,5-c]pyrimidine derivatives with human adenosine A₃ receptor subtype by Pran Kishore, D, Balakumar, C, Raghuram Rao, A, Roy, Partha Pratim, Roy, Kunal

“…Human adenosine A₃ receptor (A₃ AR) binding affinity of pyrazolotriazolopyrimidine derivatives (n=116) has been subjected to QSAR analyses using…”
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A facile microwave-assisted synthesis of 8,9-cycloalkathieno[3,2-e] [1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-ones by KAUR, RAJWINDER, KISHORE, D PRAN, NARAYANA, B LAKSHMI, RAO, K VENKAT, BALAKUMAR, C, RAJKUMAR, V, RAO, A RAGHURAM

“…A new series of fused thieno[3,2- e ][1,2,4]triazolo[1,5- c ]pyrimidinones was synthesized by condensation of ethyl-3-cyano-4,5,6,7-tetrahydrobenzo[ b…”
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Active site acidic residues and structural analysis of modelled human aromatase: a potential drug target for breast cancer by Murthy, J Narashima, Nagaraju, M, Sastry, G Madhavi, Rao, A Raghuram, Sastry, G Narahari

“…This study sheds new light on the role of acidic residues present in the active site cavity of human aromatase. Eight acidic residues (E129, D222, E245, E302,…”
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QSAR of adenosine receptor antagonists: Exploring physicochemical requirements for binding of pyrazolo[4,3- e]-1,2,4-triazolo[1,5- c]pyrimidine derivatives with human adenosine A 3 receptor subtype by Pran Kishore, D., Balakumar, C., Raghuram Rao, A., Roy, Partha Pratim, Roy, Kunal

“…Human adenosine A 3 receptor (A 3 AR) binding affinity of pyrazolotriazolopyrimidine derivatives ( n = 116) has been subjected to QSAR analyses using…”
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MEETING REPORT: Eleventh Frank Warren conference by Narayana, B. Lakshmi, Rao, A. Raghuram

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QSAR and docking studies of novel β-carboline derivatives as anticancer by Chourasiya, Ravindra Kumar, Rao, A. Raghuram, Agrawal, Ram Kishore

“…Quantitative structure–activity relationship (QSAR) studies were performed on β-carboline derivatives for prediction of anticancer activity. The statistically…”
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