Search Results - "Pundeer, Rashmi"
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Green Synthesis of Pyrazoles: Recent Developments in Aqueous Methods
Published in SynOpen (2017) (01-08-2023)“…Organic syntheses by adopting green protocols such as sonochemical procedures, microwave technologies, solvent-free conditions, green solvents, heterogeneous…”
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Recent advances in the synthesis of cholesterol-based triazoles and their biological applications
Published in Steroids (01-11-2024)“…•Synthetic strategies of cholesterol-based triazoles is provided.•33 Different synthetic schemes are provided.•Cholesterol-triazole hybrid are prepared by…”
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3
Chalcone and pyrazoline derivatives of dehydroacetic acid as digestive enzyme effectors and In silico studies
Published in Journal of molecular structure (05-11-2023)“…•Synthesis of DHA chalcones and pyrazolines.•Enzymatic activities of α-Amylase, Lipase, Trypsin, Pepsin and BSA were performed.•In silico studies of DHA…”
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4
Synergistic corrosion inhibition of mild steel by chalcone derivatives and KI in acidic media via computational and experimental methods
Published in Progress in organic coatings (01-01-2025)“…The corrosion inhibition characteristics of chalcone 4-hydroxy-6-methyl-3-(3-phenylacryloyl)-2H-pyran-2-one derivatives with different functional groups (H,…”
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5
Developments in the synthesis of α,α-dibromoacetophenones and related compounds
Published in Synthetic communications (18-06-2019)“…Increasing demand of α,α-dibromoketones, as highly reactive and easy-to-handle precursors to carry out selective organic transformations, to synthesize…”
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Development of potential cathepsin B inhibitors: Synthesis of new bithiazole derivatives, in vitro studies supported with theoretical docking studies
Published in International journal of biological macromolecules (01-11-2024)“…Cysteine cathepsins play a crucial role in cancer, inflammation, and the regulation of degenerative processes such as apoptosis, making them significant…”
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Insights of newly synthesized novel pyrazole compounds for mild steel corrosion inhibition in an acidic environment by experimental and computational calculations
Published in Journal of molecular structure (15-11-2024)“…•Novel pyrazole derivatives synthesized and evaluated as corrosion inhibitor.•Pyrazoles Pz-a (84.47 %) and Pz-b (89.85 %) are good inhibitors for mild steel in…”
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8
Dehydroacetic acid hydrazones as potent enzyme inhibitors: design, synthesis and computational studies
Published in Computational toxicology (01-11-2022)“…•Designing and in silico studies on hydrazones of DHA.•Synthesis of most potent derivative.•Evaluation against amylase, lipase, trypsin, BSA, cathepsin B and…”
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α,α‐Dibromoketone precursors in the synthesis of some new thiazole derivatives: Thiazol‐2‐yl hydrazonobutanoates, thiazol‐2‐yl pyrazole‐4‐carboxylates and acids
Published in Journal of heterocyclic chemistry (01-05-2020)“…In the present study, α,α‐dibromoacetophenones are used as efficient precursors for the facile synthesis of several new hydrazonothiazoles, ethyl…”
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10
Pyrazole-thiazole hybrids: Synthesis, computational studies and impact on digestive enzymes
Published in Journal of molecular structure (15-11-2024)“…•A series of pyrazole-thiazole hybrids were synthesized and characterized by IR, 1H NMR, 13C NMR, and LC-MS.•All the synthesized compounds were tested for…”
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Some New Pyrazolyl Pyrazolones and Cyanopyrazolyl Acrylates: Design, Synthesis and Biological Evaluation
Published in ChemistrySelect (Weinheim) (21-06-2019)“…The present work is aimed to report several new synthetically and medicinally important pyrazole derivatives. Herein, a series of new…”
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12
A Facile Synthesis of Some New 1-Benzothiazolyl-3-aryl/Hetaryl-5-(3-aryl-1-phenyl-4-pyrazolyl) Pyrazoles and Their Antimicrobial Activity
Published in Journal of heterocyclic chemistry (01-11-2015)“…Some new derivatives of 1‐benzothiazolyl‐3‐aryl/hetaryl‐5‐(3‐aryl‐1‐phenyl‐4‐pyrazolyl) pyrazoles were synthesized by the cyclocondensation of…”
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13
Synthesis and evaluation of antibacterial and antifungal activities of new (Z)-3-bromo-4-(1,3-diaryl-1H-pyrazol-4-yl)but-3-en-2-ones and 4-(3-methyl-1-phenyl-1H-pyrazol-5-yl)-1,3-diaryl-1H-pyrazoles
Published in Medicinal chemistry research (01-10-2013)“…Bromination of 4-(1, 3-diaryl-1 H -pyrazol-4-yl) but-3-en-2-ones, triggered by a combination of potassium bromide and cerium(IV) ammonium nitrate in a biphasic…”
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14
One-Pot Synthesis of Some New Semicarbazone, Thiosemicarbazone, and Hydrazone Derivatives of 1-Phenyl-3-Arylpyrazole-4-Carboxaldehyde from Acetophenone Phenylhydrazones Using Vilsmeier-Haack Reagent
Published in Synthetic communications (01-01-2009)“…Semicarbazone derivatives 3 of 1,3-diphenylpyrazole-4-carboxaldehyde have been synthesized in high yields through a one-pot procedure involving acetophenone…”
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α,α-Dibromoacetophenones mediated synthesis of some new 7H-7-alkoxy-3-alkyl/phenyl-6-aryl-s-triazolo[3,4-b][1,3,4]thiadiazines and their antimicrobial evaluation
Published in Medicinal chemistry research (01-12-2012)“…A series of new 7 H -7-alkoxy-3-alkyl/phenyl-6-aryl- s -triazolo[3,4-b][1,3,4]thiadiazines (3 , 4) were synthesized by the reaction of various…”
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A novel and facile iodine(III)-mediated approach for C(5)-acetoxylation of 6-hydroxyflavone and 6-hydroxyflavanones
Published in Tetrahedron letters (29-11-2004)“…Oxidation of 6-hydroxyflavone and 6-hydroxyflavanones with iodobenzene diacetate in acetic acid leads to regioselective acetoxylation, thereby providing a…”
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A Facile Synthesis of Thiazole-2(3H)-thiones Through [Hydroxy(tosyloxy)iodo]benzene
Published in Synthetic communications (2004)“…A one-pot facile synthesis of thiazole-2(3H)-thiones (4) has been achieved by hypervalent iodine oxidation of ketones (1) using [hydroxy(tosyloxy)iodo]benzene,…”
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An Improved Iodine(III) Mediated Method for Thiocyanation of 2-Arylindan-1,3-diones, Phenols, and Anilines
Published in Synthetic communications (01-12-2003)“…An improved method for thiocyanation of 2-arylindan-1,3-diones, phenols, and anilines using a reagent combination of (dichloroiodo)benzene and potassium…”
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