Search Results - "Popat, D."

Novel quinoline and naphthalene derivatives as potent antimycobacterial agents by Upadhayaya, Ram Shankar, Vandavasi, Jaya Kishore, Kardile, Ramakant A., Lahore, Santosh V., Dixit, Shailesh S., Deokar, Hemantkumar S., Shinde, Popat D., Sarmah, Manash P., Chattopadhyaya, Jyoti

“…We have designed and synthesized both the quinoline and naphthalene based molecules influenced by the unique structural make-up of mefloquine and TMC207,…”
Get full text

Study on impact of flexible endoscopy training course for surgeons in India by Sundaram, Easwaramoorthy, Chandrasekar, Sakthivel, Agarwalla, Ramesh, Govindaraj, Kanagaraj, Desarkar, Satyapriya, Yasmine, Jaseema, Khanna, Subhash, Manickavasakam, Kanagavel, Popat, Sunil

“…Context: Competence in flexible endoscopy is essential for all surgeons during this era of minimal access surgery. However, fewer surgeons have expertise in…”
Get full text

Conformationally-constrained indeno[2,1-c]quinolines--a new class of anti-mycobacterial agents by Upadhayaya, Ram Shankar, Lahore, Santosh V, Sayyed, Aftab Y, Dixit, Shailesh S, Shinde, Popat D, Chattopadhyaya, Jyoti

“…The design, synthesis and anti-mycobacterial activities of 23 conformationally-constrained indeno[2,1-c]quinolines against Mycobacterium tuberculosis H37Rv is…”
Get more information

Synthesis and antimycobacterial activity of prodrugs of indeno[2,1- c]quinoline derivatives by Upadhayaya, Ram Shankar, Shinde, Popat D., Kadam, Sandip A., Bawane, Amit N., Sayyed, Aftab Y., Kardile, Ramakant A., Gitay, Pallavi N., Lahore, Santosh V., Dixit, Shailesh S., Földesi, András, Chattopadhyaya, Jyoti

“…Recently we have reported anti-TB properties of a new class of conformationally-constrained indeno[2,1- c]quinolines, which are although considerably active…”
Get full text

Role for α-L-fucosidase in the control of Helicobacter pylori-infected gastric cancer cells by Liu, Ta-Wei, Ho, Ching-Wen, Huang, Hsin-Hung, Chang, Sue-Ming, Popat, Shide D, Wang, Yi-Ting, Wu, Ming-Shiang, Chen, Yu-Ju, Lin, Chun-Hung

“…Infecting about one-half of the global human population, Helicobacter pylori is well established as the primary cause of gastritis, duodenal ulcer, and gastric…”
Get full text

Structural Basis of α-Fucosidase Inhibition by Iminocyclitols with Ki Values in the Micro- to Picomolar Range by Wu, Hsing-Ju, Ho, Ching-Wen, Ko, Tzu-Ping, Popat, Shinde D, Lin, Chun-Hung, Wang, Andrew H.-J

“…Two loops were found to move inward toward the α‐fucosidase active site to produce a closed conformation of complexes with inhibitors with increasing Ki values…”
Get full text

Synthesis and structure of azole-fused indeno[2,1-c]quinolines and their anti-mycobacterial properties by Upadhayaya, Ram Shankar, Shinde, Popat D, Sayyed, Aftab Y, Kadam, Sandip A, Bawane, Amit N, Poddar, Avijit, Plashkevych, Oleksandr, Földesi, Andras, Chattopadhyaya, Jyoti

“…Prompted by our discovery of a new class of conformationally-locked indeno[2,1-c]quinolines as anti-mycobacterials, compounds 2a and 3a (Fig. 1; MIC < 0.39 μg…”
Get more information

Synthesis and Evaluation of 4/5-Hydroxy-2,3-diaryl(substituted)-cyclopent-2-en-1-ones as cis-Restricted Analogues of Combretastatin A-4 as Novel Anticancer Agents by Gurjar, Mukund K, Wakharkar, Radhika D, Singh, Anu T, Jaggi, Manu, Borate, Hanumant B, Shinde, Popat D, Verma, Ritu, Rajendran, Praveen, Dutt, Sarjana, Singh, Gurvinder, Sanna, Vinod K, Singh, Manoj K, Srivastava, Sanjay K, Mahajan, Vishal A, Jadhav, Vinod H, Dutta, Kakali, Krishnan, Karthik, Chaudhary, Anika, Agarwal, Shiv K, Mukherjee, Rama, Burman, Anand C

“…A new series of 2,3-diaryl-4/5-hydroxy-cyclopent-2-en-1-one analogues replacing the cis double bond of combretastatin A-4 (CA-4) by 4/5-hydroxy cyclopentenone…”
Get full text

Enantiomeric separation of novel anticancer agent 5-hydroxy-3-(4-methoxyphenyl)-2-(3,4,5-trimethoxyphenyl)-cyclopent-2-en-1-one by Shinde, Popat D., Jadhav, Vinod H., Borate, Hanumant B., Bhide, Sunil R., Sonawane, Kiran B., Wakharkar, Radhika D.

“…The enantiomers of 5-hydroxy-3-(4-methoxyphenyl)-2-(3,4,5-trimethoxyphenyl)-cyclopent-2-en-1-one, a novel anticancer agent, were separated by derivatisation…”
Get full text

Study on impact of flexible endoscopy training course for surgeons in India by Sundaram, Easwaramoorthy, Chandrasekar, Sakthivel, Agarwalla, Ramesh, Govindaraj, Kanagaraj, Desarkar, Satyapriya, Yasmine, Jaseema, Khanna, Subhash, Manickavasakam, Kanagavel, Popat, Sunil D

“…Competence in flexible endoscopy is essential for all surgeons during this era of minimal access surgery. However, fewer surgeons have expertise in endoscopy…”
Get full text

Comparative study on the behaviour of castellated beams provided with hexagonal, circular, and diamond-shaped web openings by Patil, Sourabh S., Kumbhar, Popat D.

Get full text

Comparative study on behaviour of castellated beams with diamond- and hexagonal-shaped openings using CFRP stiffeners by Mali, Suyash S., Kumbhar, Popat D.

Get full text

Li–X-type zeolite mediated Michael addition of thiols to cyclic enones and its application in the synthesis of 13-thiaprostaglandins by Shinde, Popat D, Mahajan, Vishal A, Borate, Hanumant B, Tillu, Vasudha H, Bal, Rajaram, Chandwadkar, Asha, Wakharkar, Radhika D

“…Michael addition of various thiols to cyclic enones in presence of Li–X-type zeolite has been described. 13-Thiaprostaglandins have been synthesized in good…”
Get full text

A convenient oxidative demasking of 1,3-dithiolanes and dithianes to carbonyl compounds with TBHP by Barhate, Nivrutti B, Shinde, Popat D, Mahajan, Vishal A, Wakharkar, Radhika D

“…Regeneration of carbonyl compounds from their 1,3-dithiolanes and dithianes was achieved using tert-butyl hydroperoxide (TBHP, aq. 70%) in high yields. Thus,…”
Get full text

Structural Basis of α‐Fucosidase Inhibition by Iminocyclitols with K i Values in the Micro‐ to Picomolar Range by Wu, Hsing‐Ju, Ho, Ching‐Wen, Ko, Tzu‐Ping, Popat, Shinde D., Lin, Chun‐Hung, Wang, Andrew H.‐J.

Get full text

Comparative study on the behaviour of conventional and pre-engineered buildings provided with different types of bracing by Bharmal, Pravin P., Kumbhar, Popat D., Gumaste, Krishnakedar S.

Get full text

Structural behavior of pre-engineered industrial buildings provided with different types of bracings in various seismic zones by Bharmal, Pravin P., Kumbhar, Popat D., Gumaste, Krishnakedar S.

Get full text

Analyzing the influence of perforations on the structural behavior of mild steel cellular beams by Kurlapkar, Rohit Rajendra, Patil, Amit Prakash, Kumbhar, Popat D.

Get full text

Immunotherapy: MECHANISMS REGULATING THE RESISTANCE OF NORMAL T-CELLS TO CD5 CAR-MEDIATED CYTOTOXICITY by Ma, R., Woods, M.L., Chaumette, A., Popat, D., Carisey, A., Brenner, M., Mamonkin, M.

Get full text

Thioacetalization of the carbonyl function, transthioacetalization of acetals, ketals, oximes and hydrazones catalysed by aqueous hydrobromic acid by Shinde, Popat D., Borate, Hanumant B., Wakharkar, Radhika D.

Get full text